| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SYK | KSYK_HUMAN | 8WYWA | P43405 | 364 | 633 | 635.0 | XFB:701 | Type1 | None | DFGin | 6.2371 | 14.4668 | BLAminus | -132.59, -164.71 | 66.23, 68.08 | -96.88, 23.52 | 293.79, 90.86 | -58.6, -30.92 | in-in | in | 8.0458 | Saltbr-in | 2.7999 | HRD-in | -78.12, -54.08 | 75.86, 6.55 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.953 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 61.34 | APE8-rot-na | 31.52 | APE67-dihe-in | -65.01, -13.06 | -58.71, -34.21 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.9 | 0.202 | 0.242 | A | 293.0 | 264.0 | 6 | 31 | 25 | 6 | [[370, 628]] | 1.0 | 8wyw | TYR_SYK_HUMAN | TYR | 5.7e-90 | 307.1 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 8WYWB | P43405 | 365 | 633 | 635.0 | XFB:701 | Type1 | None | DFGin | 6.298 | 14.4316 | BLAminus | -136.18, -166.23 | 64.92, 68.41 | -94.85, 24.26 | 293.81, 88.05 | -62.54, -27.54 | in-in | in | 8.0999 | Saltbr-in | 2.7616 | HRD-in | -75.21, -53.42 | 72.9, 5.68 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9696 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 56.28 | APE8-rot-na | 30.56 | APE67-dihe-in | -70.56, -10.12 | -50.08, -35.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.9 | 0.202 | 0.242 | B | 293.0 | 263.0 | 6 | 31 | 25 | 6 | [[370, 628]] | 1.0 | 8wyw | TYR_SYK_HUMAN | TYR | 5.7e-90 | 307.1 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SYK | KSYK_HUMAN | 8WYWA | P43405 | 364 | 633 | 635.0 | XFB:701 | Type1 | None | DFGin | 6.2371 | 14.4668 | BLAminus | -132.59, -164.71 | 66.23, 68.08 | -96.88, 23.52 | 293.79, 90.86 | -58.6, -30.92 | in-in | in | 8.0458 | Saltbr-in | 2.7999 | HRD-in | -78.12, -54.08 | 75.86, 6.55 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.953 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 61.34 | APE8-rot-na | 31.52 | APE67-dihe-in | -65.01, -13.06 | -58.71, -34.21 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.9 | 0.202 | 0.242 | A | 293.0 | 264.0 | 6 | 31 | 25 | 6 | [[370, 628]] | 1.0 | 8wyw | Homo sapiens | TYR_SYK_HUMAN | TYR | 5.7e-90 | 307.1 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 8WYWB | P43405 | 365 | 633 | 635.0 | XFB:701 | Type1 | None | DFGin | 6.298 | 14.4316 | BLAminus | -136.18, -166.23 | 64.92, 68.41 | -94.85, 24.26 | 293.81, 88.05 | -62.54, -27.54 | in-in | in | 8.0999 | Saltbr-in | 2.7616 | HRD-in | -75.21, -53.42 | 72.9, 5.68 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9696 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 56.28 | APE8-rot-na | 30.56 | APE67-dihe-in | -70.56, -10.12 | -50.08, -35.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.9 | 0.202 | 0.242 | B | 293.0 | 263.0 | 6 | 31 | 25 | 6 | [[370, 628]] | 1.0 | 8wyw | Homo sapiens | TYR_SYK_HUMAN | TYR | 5.7e-90 | 307.1 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|