| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DA | P21802 | 467 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8853 | 13.9149 | BLAminus | -147.5, -176.54 | 60.37, 88.47 | -102.26, 25.1 | 300.92, 154.4 | -57.13, -34.04 | in-in | in | 7.8251 | Saltbr-in | 2.7968 | HRD-in | -84.9, -54.51 | 77.26, 0.33 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8575 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.98, 12.82 | APE9-dihe-in | -97.28, 131.96 | APE8-dihe-in | -62.75, 115.5 | APE8-rot-na | 335.68 | APE67-dihe-in | -74.05, -8.17 | -56.13, -41.02 | APE12-dist-na | 10.0605 | APE11-dist-na | 11.1727 | APE10-dist-na | 7.3858 | APE9-dist-in | 4.9839 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | A | 324.0 | 298.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8w3d | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DB | P21802 | 463 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8319 | 14.0174 | BLAminus | -148.34, -176.74 | 60.99, 88.17 | -102.41, 24.87 | 299.72, 154.97 | -58.18, -33.84 | in-in | in | 7.7871 | Saltbr-in | 2.7649 | HRD-in | -83.96, -54.88 | 76.41, -0.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8516 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.87, 19.37 | APE9-dihe-in | -95.98, 132.29 | APE8-dihe-in | -61.49, 116.39 | APE8-rot-na | 335.8 | APE67-dihe-in | -74.83, -7.73 | -55.74, -41.43 | APE12-dist-na | 10.8074 | APE11-dist-na | 10.9135 | APE10-dist-na | 7.4654 | APE9-dist-in | 4.9702 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | B | 324.0 | 286.0 | 16 | 30 | 23 | 7 | [[481, 759]] | 1.0 | 8w3d | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DC | P21802 | 467 | 766 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8552 | 13.9002 | BLAminus | -147.64, -176.09 | 60.07, 88.49 | -102.13, 25.05 | 300.63, 154.01 | -57.64, -33.63 | in-in | in | 7.7725 | Saltbr-in | 2.7934 | HRD-in | -84.16, -54.95 | 77.08, 0.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8542 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.76, 14.01 | APE9-dihe-in | -96.42, 131.36 | APE8-dihe-in | -63.38, 115.02 | APE8-rot-na | 334.88 | APE67-dihe-in | -73.92, -8.44 | -56.07, -40.69 | APE12-dist-na | 10.1128 | APE11-dist-na | 11.132 | APE10-dist-na | 7.4256 | APE9-dist-in | 4.9863 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | C | 324.0 | 300.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8w3d | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DD | P21802 | 463 | 765 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8116 | 14.007 | BLAminus | -147.99, -176.89 | 61.0, 88.35 | -102.2, 24.75 | 299.43, 154.83 | -57.77, -34.3 | in-in | in | 7.7731 | Saltbr-in | 2.7585 | HRD-in | -84.08, -54.96 | 76.09, 0.5 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.846 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.21, 21.5 | APE9-dihe-in | -95.42, 132.82 | APE8-dihe-in | -60.81, 115.91 | APE8-rot-na | 335.81 | APE67-dihe-in | -74.61, -8.25 | -55.74, -40.98 | APE12-dist-na | 10.7994 | APE11-dist-na | 10.9249 | APE10-dist-na | 7.5894 | APE9-dist-in | 4.9671 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | D | 324.0 | 296.0 | 7 | 30 | 28 | 2 | [[481, 759]] | 1.0 | 8w3d | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DA | P21802 | 467 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8853 | 13.9149 | BLAminus | -147.5, -176.54 | 60.37, 88.47 | -102.26, 25.1 | 300.92, 154.4 | -57.13, -34.04 | in-in | in | 7.8251 | Saltbr-in | 2.7968 | HRD-in | -84.9, -54.51 | 77.26, 0.33 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8575 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.98, 12.82 | APE9-dihe-in | -97.28, 131.96 | APE8-dihe-in | -62.75, 115.5 | APE8-rot-na | 335.68 | APE67-dihe-in | -74.05, -8.17 | -56.13, -41.02 | APE12-dist-na | 10.0605 | APE11-dist-na | 11.1727 | APE10-dist-na | 7.3858 | APE9-dist-in | 4.9839 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | A | 324.0 | 298.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8w3d | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DB | P21802 | 463 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8319 | 14.0174 | BLAminus | -148.34, -176.74 | 60.99, 88.17 | -102.41, 24.87 | 299.72, 154.97 | -58.18, -33.84 | in-in | in | 7.7871 | Saltbr-in | 2.7649 | HRD-in | -83.96, -54.88 | 76.41, -0.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8516 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.87, 19.37 | APE9-dihe-in | -95.98, 132.29 | APE8-dihe-in | -61.49, 116.39 | APE8-rot-na | 335.8 | APE67-dihe-in | -74.83, -7.73 | -55.74, -41.43 | APE12-dist-na | 10.8074 | APE11-dist-na | 10.9135 | APE10-dist-na | 7.4654 | APE9-dist-in | 4.9702 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | B | 324.0 | 286.0 | 16 | 30 | 23 | 7 | [[481, 759]] | 1.0 | 8w3d | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DC | P21802 | 467 | 766 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8552 | 13.9002 | BLAminus | -147.64, -176.09 | 60.07, 88.49 | -102.13, 25.05 | 300.63, 154.01 | -57.64, -33.63 | in-in | in | 7.7725 | Saltbr-in | 2.7934 | HRD-in | -84.16, -54.95 | 77.08, 0.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8542 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.76, 14.01 | APE9-dihe-in | -96.42, 131.36 | APE8-dihe-in | -63.38, 115.02 | APE8-rot-na | 334.88 | APE67-dihe-in | -73.92, -8.44 | -56.07, -40.69 | APE12-dist-na | 10.1128 | APE11-dist-na | 11.132 | APE10-dist-na | 7.4256 | APE9-dist-in | 4.9863 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | C | 324.0 | 300.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8w3d | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W3DD | P21802 | 463 | 765 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.8116 | 14.007 | BLAminus | -147.99, -176.89 | 61.0, 88.35 | -102.2, 24.75 | 299.43, 154.83 | -57.77, -34.3 | in-in | in | 7.7731 | Saltbr-in | 2.7585 | HRD-in | -84.08, -54.96 | 76.09, 0.5 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.846 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.21, 21.5 | APE9-dihe-in | -95.42, 132.82 | APE8-dihe-in | -60.81, 115.91 | APE8-rot-na | 335.81 | APE67-dihe-in | -74.61, -8.25 | -55.74, -40.98 | APE12-dist-na | 10.7994 | APE11-dist-na | 10.9249 | APE10-dist-na | 7.5894 | APE9-dist-in | 4.9671 | N549K,D650V | None | None | XRAY | 2.04 | 0.22 | 0.25 | D | 324.0 | 296.0 | 7 | 30 | 28 | 2 | [[481, 759]] | 1.0 | 8w3d | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 6.7e-104 | 352.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|