| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8S1AA | P10721 | 565 | 931 | 976.0 | 6T2:61001 | Type1 | Active | DFGin | 7.4808 | 13.4537 | BLAminus | -130.25, 174.66 | 66.24, 93.25 | -105.72, 18.63 | 285.4, 75.09 | -61.16, -30.32 | in-in | in | 8.3211 | Saltbr-in | 3.005 | HRD-in | -89.71, -45.27 | 75.21, -0.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8512 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.31, 143.6 | APE9-dihe-in | -122.04, 151.68 | APE8-dihe-in | -82.91, 74.45 | APE8-rot-na | 35.68 | APE67-dihe-in | -72.93, -9.14 | -57.9, -42.62 | APE12-dist-na | 13.9398 | APE11-dist-na | 9.4995 | APE10-dist-na | 12.9558 | APE9-dist-in | 7.5844 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.188 | 0.208 | A | 327.0 | 286.0 | 3 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s1a | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S1AB | P10721 | 566 | 931 | 976.0 | 6T2:61001 | Type1 | Active | DFGin | 7.4323 | 13.5642 | BLAminus | -134.77, 174.81 | 62.68, 90.66 | -103.62, 20.87 | 285.06, 74.67 | -61.54, -35.7 | in-in | in | 8.3104 | Saltbr-in | 2.716 | HRD-in | -95.21, -44.44 | 74.01, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8065 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.03, 139.89 | APE9-dihe-in | -118.65, 149.04 | APE8-dihe-in | -82.35, 75.62 | APE8-rot-na | 34.69 | APE67-dihe-in | -73.13, -6.18 | -57.98, -42.32 | APE12-dist-na | 14.1507 | APE11-dist-na | 9.6536 | APE10-dist-na | 13.1267 | APE9-dist-in | 7.6697 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.188 | 0.208 | B | 327.0 | 288.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s1a | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8S1AA | P10721 | 565 | 931 | 976.0 | 6T2:61001 | Type1 | Active | DFGin | 7.4808 | 13.4537 | BLAminus | -130.25, 174.66 | 66.24, 93.25 | -105.72, 18.63 | 285.4, 75.09 | -61.16, -30.32 | in-in | in | 8.3211 | Saltbr-in | 3.005 | HRD-in | -89.71, -45.27 | 75.21, -0.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8512 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.31, 143.6 | APE9-dihe-in | -122.04, 151.68 | APE8-dihe-in | -82.91, 74.45 | APE8-rot-na | 35.68 | APE67-dihe-in | -72.93, -9.14 | -57.9, -42.62 | APE12-dist-na | 13.9398 | APE11-dist-na | 9.4995 | APE10-dist-na | 12.9558 | APE9-dist-in | 7.5844 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.188 | 0.208 | A | 327.0 | 286.0 | 3 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s1a | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S1AB | P10721 | 566 | 931 | 976.0 | 6T2:61001 | Type1 | Active | DFGin | 7.4323 | 13.5642 | BLAminus | -134.77, 174.81 | 62.68, 90.66 | -103.62, 20.87 | 285.06, 74.67 | -61.54, -35.7 | in-in | in | 8.3104 | Saltbr-in | 2.716 | HRD-in | -95.21, -44.44 | 74.01, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8065 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.03, 139.89 | APE9-dihe-in | -118.65, 149.04 | APE8-dihe-in | -82.35, 75.62 | APE8-rot-na | 34.69 | APE67-dihe-in | -73.13, -6.18 | -57.98, -42.32 | APE12-dist-na | 14.1507 | APE11-dist-na | 9.6536 | APE10-dist-na | 13.1267 | APE9-dist-in | 7.6697 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.188 | 0.208 | B | 327.0 | 288.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s1a | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|