| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8PQGA | P10721 | 566 | 931 | 976.0 | 9JI:61001 | Type1 | Active | DFGin | 7.0429 | 14.1671 | BLAminus | -124.55, -174.12 | 54.99, 78.46 | -96.45, 26.87 | 280.71, 70.71 | -64.48, -33.68 | in-in | in | 8.0418 | Saltbr-in | 2.847 | HRD-in | -90.54, -41.04 | 71.94, -5.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0249 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.66, 135.23 | APE9-dihe-in | -115.63, 149.54 | APE8-dihe-in | -83.89, 83.11 | APE8-rot-na | 25.85 | APE67-dihe-in | -70.62, -11.93 | -61.47, -41.45 | APE12-dist-na | 999.0 | APE11-dist-na | 9.8657 | APE10-dist-na | 13.0316 | APE9-dist-in | 7.6588 | I563S,V569S,Y609Q,L631S,M651E,I662H,T670I,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.4 | 0.207 | 0.231 | A | 327.0 | 283.0 | 5 | 30 | 25 | 5 | [[589, 926]] | 1.0 | 8pqg | TYR_KIT_HUMAN | TYR | 4.7e-104 | 353.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8PQGC | P10721 | 565 | 932 | 976.0 | 9JI:61001 | Type1 | Active | DFGin | 6.9981 | 13.7774 | BLAminus | -125.01, -177.18 | 59.69, 81.81 | -99.94, 28.85 | 284.0, 66.15 | -68.84, -20.03 | in-in | in | 7.8376 | Saltbr-in | 2.8929 | HRD-in | -87.34, -47.72 | 75.4, 1.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9945 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.89, 137.72 | APE9-dihe-in | -124.07, 148.98 | APE8-dihe-in | -81.48, 76.95 | APE8-rot-na | 33.1 | APE67-dihe-in | -72.2, -11.85 | -56.44, -41.57 | APE12-dist-na | 14.3671 | APE11-dist-na | 10.0194 | APE10-dist-na | 12.9788 | APE9-dist-in | 7.6471 | I563S,V569S,Y609Q,L631S,M651E,I662H,T670I,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.4 | 0.207 | 0.231 | C | 327.0 | 290.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8pqg | TYR_KIT_HUMAN | TYR | 4.7e-104 | 353.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8PQGA | P10721 | 566 | 931 | 976.0 | 9JI:61001 | Type1 | Active | DFGin | 7.0429 | 14.1671 | BLAminus | -124.55, -174.12 | 54.99, 78.46 | -96.45, 26.87 | 280.71, 70.71 | -64.48, -33.68 | in-in | in | 8.0418 | Saltbr-in | 2.847 | HRD-in | -90.54, -41.04 | 71.94, -5.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0249 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.66, 135.23 | APE9-dihe-in | -115.63, 149.54 | APE8-dihe-in | -83.89, 83.11 | APE8-rot-na | 25.85 | APE67-dihe-in | -70.62, -11.93 | -61.47, -41.45 | APE12-dist-na | 999.0 | APE11-dist-na | 9.8657 | APE10-dist-na | 13.0316 | APE9-dist-in | 7.6588 | I563S,V569S,Y609Q,L631S,M651E,I662H,T670I,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.4 | 0.207 | 0.231 | A | 327.0 | 283.0 | 5 | 30 | 25 | 5 | [[589, 926]] | 1.0 | 8pqg | Homo sapiens | TYR_KIT_HUMAN | TYR | 4.7e-104 | 353.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8PQGC | P10721 | 565 | 932 | 976.0 | 9JI:61001 | Type1 | Active | DFGin | 6.9981 | 13.7774 | BLAminus | -125.01, -177.18 | 59.69, 81.81 | -99.94, 28.85 | 284.0, 66.15 | -68.84, -20.03 | in-in | in | 7.8376 | Saltbr-in | 2.8929 | HRD-in | -87.34, -47.72 | 75.4, 1.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9945 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.89, 137.72 | APE9-dihe-in | -124.07, 148.98 | APE8-dihe-in | -81.48, 76.95 | APE8-rot-na | 33.1 | APE67-dihe-in | -72.2, -11.85 | -56.44, -41.57 | APE12-dist-na | 14.3671 | APE11-dist-na | 10.0194 | APE10-dist-na | 12.9788 | APE9-dist-in | 7.6471 | I563S,V569S,Y609Q,L631S,M651E,I662H,T670I,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.4 | 0.207 | 0.231 | C | 327.0 | 290.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8pqg | Homo sapiens | TYR_KIT_HUMAN | TYR | 4.7e-104 | 353.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|