| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8PQCA | P10721 | 566 | 932 | 976.0 | 9OO:61001 | Type1 | Active | DFGin | 7.3203 | 13.7282 | BLAminus | -124.52, 177.4 | 59.32, 88.07 | -98.4, 24.69 | 287.2, 70.41 | -61.62, -29.61 | in-in | in | 7.8146 | Saltbr-in | 2.7673 | HRD-in | -93.83, -42.0 | 73.11, -0.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.888 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.91, 142.75 | APE9-dihe-in | -125.5, 151.35 | APE8-dihe-in | -83.13, 70.57 | APE8-rot-na | 37.57 | APE67-dihe-in | -73.25, -7.87 | -53.76, -43.02 | APE12-dist-na | 14.0422 | APE11-dist-na | 9.7008 | APE10-dist-na | 13.0233 | APE9-dist-in | 7.718 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.77 | 0.183 | 0.206 | A | 327.0 | 287.0 | 2 | 30 | 28 | 2 | [[589, 926]] | 1.0 | 8pqc | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8PQCB | P10721 | 566 | 931 | 976.0 | 9OO:61001 | Type1 | Active | DFGin | 7.283 | 13.8349 | BLAminus | -128.31, 173.51 | 60.11, 89.0 | -97.68, 23.86 | 286.68, 71.19 | -63.1, -28.82 | in-in | in | 7.9711 | Saltbr-in | 2.8275 | HRD-in | -94.17, -44.79 | 74.42, -0.63 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.29, 141.63 | APE9-dihe-in | -125.35, 153.08 | APE8-dihe-in | -84.91, 76.41 | APE8-rot-na | 34.61 | APE67-dihe-in | -73.13, -6.88 | -58.59, -41.47 | APE12-dist-na | 14.0973 | APE11-dist-na | 9.7391 | APE10-dist-na | 13.1187 | APE9-dist-in | 7.6922 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.77 | 0.183 | 0.206 | B | 327.0 | 287.0 | 1 | 30 | 29 | 1 | [[589, 926]] | 1.0 | 8pqc | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8PQCA | P10721 | 566 | 932 | 976.0 | 9OO:61001 | Type1 | Active | DFGin | 7.3203 | 13.7282 | BLAminus | -124.52, 177.4 | 59.32, 88.07 | -98.4, 24.69 | 287.2, 70.41 | -61.62, -29.61 | in-in | in | 7.8146 | Saltbr-in | 2.7673 | HRD-in | -93.83, -42.0 | 73.11, -0.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.888 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.91, 142.75 | APE9-dihe-in | -125.5, 151.35 | APE8-dihe-in | -83.13, 70.57 | APE8-rot-na | 37.57 | APE67-dihe-in | -73.25, -7.87 | -53.76, -43.02 | APE12-dist-na | 14.0422 | APE11-dist-na | 9.7008 | APE10-dist-na | 13.0233 | APE9-dist-in | 7.718 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.77 | 0.183 | 0.206 | A | 327.0 | 287.0 | 2 | 30 | 28 | 2 | [[589, 926]] | 1.0 | 8pqc | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8PQCB | P10721 | 566 | 931 | 976.0 | 9OO:61001 | Type1 | Active | DFGin | 7.283 | 13.8349 | BLAminus | -128.31, 173.51 | 60.11, 89.0 | -97.68, 23.86 | 286.68, 71.19 | -63.1, -28.82 | in-in | in | 7.9711 | Saltbr-in | 2.8275 | HRD-in | -94.17, -44.79 | 74.42, -0.63 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.29, 141.63 | APE9-dihe-in | -125.35, 153.08 | APE8-dihe-in | -84.91, 76.41 | APE8-rot-na | 34.61 | APE67-dihe-in | -73.13, -6.88 | -58.59, -41.47 | APE12-dist-na | 14.0973 | APE11-dist-na | 9.7391 | APE10-dist-na | 13.1187 | APE9-dist-in | 7.6922 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.77 | 0.183 | 0.206 | B | 327.0 | 287.0 | 1 | 30 | 29 | 1 | [[589, 926]] | 1.0 | 8pqc | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|