PDB: 8H75 — TYR FGFR2_HUMAN

Total number of chains: 4
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 4 100.0% 8H75A

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
TYR FGFR2 FGFR2_HUMAN 8H75A P21802 467 765 821.0 KX0:1001 Type1 Inactive DFGin 7.213 14.585 BLAminus -154.63, 179.57 55.91, 54.1 -74.79, -3.2 274.96, 68.76 -58.48, -41.04 in-out in 7.417 Saltbr-out 4.811 HRD-out -96.67, 103.01 -67.39, -41.62 out-in-in SNCoii in-in ActLoopNT-in 3.141 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -162.98, 72.34 APE9-dihe-in -137.73, 148.36 APE8-dihe-in -71.99, 141.14 APE8-rot-na 343.8 APE67-dihe-in -63.34, -38.73 -70.52, -42.38 APE12-dist-na 13.018 APE11-dist-na 9.408 APE10-dist-na 7.3 APE9-dist-in 6.868 None PTR656 PTR656 XRAY 3.75 0.216 0.238 A 312 285 14 0 0 0 [[481, 759]] 1.0 8h75 TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8H75B P21802 467 764 821.0 KX0:1001 Type1 Inactive DFGin 7.114 15.321 BLAminus -140.03, -170.55 50.75, 50.66 -73.91, -10.21 273.73, 91.58 -58.96, -39.4 in-out in 7.468 Saltbr-out 4.436 HRD-in -64.7, -43.07 75.93, -2.73 out-in-out SNCoio in-out ActLoopNT-in 3.383 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -63.7, -40.57 APE9-dihe-in -143.97, 156.51 APE8-dihe-in -61.01, 137.3 APE8-rot-na 23.2 APE67-dihe-in -61.01, -38.56 -64.05, -38.82 APE12-dist-na 14.092 APE11-dist-na 11.287 APE10-dist-na 7.446 APE9-dist-in 5.738 None PTR656 PTR656 XRAY 3.75 0.216 0.238 B 312 283 15 0 0 0 [[481, 759]] 1.0 8h75 TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8H75C P21802 467 763 821.0 KX0:1001 Type1 Inactive DFGin 6.415 13.942 BLAminus -139.77, -171.25 51.94, 53.82 -68.52, 7.4 288.78, 82.18 -59.71, -35.71 in-in in 7.763 Saltbr-in 2.579 HRD-in -64.69, -38.41 67.2, 3.13 in-out-out SNCioo out-out ActLoopNT-out 3.788 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -86.06, 23.54 APE9-dihe-in -123.01, 141.76 APE8-dihe-in -64.83, 140.92 APE8-rot-na 351.7 APE67-dihe-in -63.43, -39.45 -65.53, -40.64 APE12-dist-na 10.784 APE11-dist-na 10.944 APE10-dist-na 7.514 APE9-dist-in 5.382 None PTR656 PTR656 XRAY 3.75 0.216 0.238 C 312 275 22 0 0 6 [[481, 759]] 1.0 8h75 TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8H75D P21802 467 764 821.0 KX0:1001 Type1 Inactive DFGin 6.719 14.006 BLAminus -145.79, -169.72 52.31, 64.06 -85.42, 2.67 285.45, 103.44 -59.5, -38.29 in-out in 7.69 Saltbr-out 4.357 HRD-in -66.94, -45.53 78.8, 0.63 out-in-out SNCoio in-out ActLoopNT-in 3.389 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out 55.78, 41.43 APE9-dihe-in -144.13, 151.96 APE8-dihe-in -70.01, 128.38 APE8-rot-na 29.85 APE67-dihe-in -54.94, -35.54 -65.88, -42.6 APE12-dist-na 10.994 APE11-dist-na 11.053 APE10-dist-na 8.829 APE9-dist-in 5.759 None PTR656 PTR656 XRAY 3.75 0.216 0.238 D 312 277 21 0 0 4 [[481, 759]] 1.0 8h75 TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2

PDB: 8H75 — TYR FGFR2_HUMAN

Total number of chains: 4
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 4 100.0% 8H75A

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
TYR FGFR2 FGFR2_HUMAN 8H75A P21802 467 765 821.0 KX0:1001 Type1 Inactive DFGin 7.213 14.585 BLAminus -154.63, 179.57 55.91, 54.1 -74.79, -3.2 274.96, 68.76 -58.48, -41.04 in-out in 7.417 Saltbr-out 4.811 HRD-out -96.67, 103.01 -67.39, -41.62 out-in-in SNCoii in-in ActLoopNT-in 3.141 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -162.98, 72.34 APE9-dihe-in -137.73, 148.36 APE8-dihe-in -71.99, 141.14 APE8-rot-na 343.8 APE67-dihe-in -63.34, -38.73 -70.52, -42.38 APE12-dist-na 13.018 APE11-dist-na 9.408 APE10-dist-na 7.3 APE9-dist-in 6.868 None PTR656 PTR656 XRAY 3.75 0.216 0.238 A 312 285 14 0 0 0 [[481, 759]] 1.0 8h75 Homo sapiens TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8H75B P21802 467 764 821.0 KX0:1001 Type1 Inactive DFGin 7.114 15.321 BLAminus -140.03, -170.55 50.75, 50.66 -73.91, -10.21 273.73, 91.58 -58.96, -39.4 in-out in 7.468 Saltbr-out 4.436 HRD-in -64.7, -43.07 75.93, -2.73 out-in-out SNCoio in-out ActLoopNT-in 3.383 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -63.7, -40.57 APE9-dihe-in -143.97, 156.51 APE8-dihe-in -61.01, 137.3 APE8-rot-na 23.2 APE67-dihe-in -61.01, -38.56 -64.05, -38.82 APE12-dist-na 14.092 APE11-dist-na 11.287 APE10-dist-na 7.446 APE9-dist-in 5.738 None PTR656 PTR656 XRAY 3.75 0.216 0.238 B 312 283 15 0 0 0 [[481, 759]] 1.0 8h75 Homo sapiens TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8H75C P21802 467 763 821.0 KX0:1001 Type1 Inactive DFGin 6.415 13.942 BLAminus -139.77, -171.25 51.94, 53.82 -68.52, 7.4 288.78, 82.18 -59.71, -35.71 in-in in 7.763 Saltbr-in 2.579 HRD-in -64.69, -38.41 67.2, 3.13 in-out-out SNCioo out-out ActLoopNT-out 3.788 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -86.06, 23.54 APE9-dihe-in -123.01, 141.76 APE8-dihe-in -64.83, 140.92 APE8-rot-na 351.7 APE67-dihe-in -63.43, -39.45 -65.53, -40.64 APE12-dist-na 10.784 APE11-dist-na 10.944 APE10-dist-na 7.514 APE9-dist-in 5.382 None PTR656 PTR656 XRAY 3.75 0.216 0.238 C 312 275 22 0 0 6 [[481, 759]] 1.0 8h75 Homo sapiens TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8H75D P21802 467 764 821.0 KX0:1001 Type1 Inactive DFGin 6.719 14.006 BLAminus -145.79, -169.72 52.31, 64.06 -85.42, 2.67 285.45, 103.44 -59.5, -38.29 in-out in 7.69 Saltbr-out 4.357 HRD-in -66.94, -45.53 78.8, 0.63 out-in-out SNCoio in-out ActLoopNT-in 3.389 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out 55.78, 41.43 APE9-dihe-in -144.13, 151.96 APE8-dihe-in -70.01, 128.38 APE8-rot-na 29.85 APE67-dihe-in -54.94, -35.54 -65.88, -42.6 APE12-dist-na 10.994 APE11-dist-na 11.053 APE10-dist-na 8.829 APE9-dist-in 5.759 None PTR656 PTR656 XRAY 3.75 0.216 0.238 D 312 277 21 0 0 4 [[481, 759]] 1.0 8h75 Homo sapiens TYR_FGFR2_HUMAN TYR 2.5e-104 354.1 1 260 260 643 644 645 647 649 517 534 538 623 625 624 626 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2

PDB: 8H75 — TYR FGFR2_HUMAN

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name