| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | JAK1-12 | JAK1_MOUSE | 8EWYA | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | None | 999.0 | 999.0 | None | -138.68, -158.74 | 57.84, 53.41 | -86.5, 17.2 | 999.0, 999.0 | -66.33, -21.83 | in-none | in | 8.0785 | Saltbr-none | 999.0 | HRD-in | -63.86, -38.24 | 65.99, -1.42 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.8414 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.88, 139.03 | APE9-dihe-in | -137.63, 148.1 | APE8-dihe-in | -70.82, 80.23 | APE8-rot-na | 999.0 | APE67-dihe-in | -71.32, -12.38 | -60.07, -30.97 | APE12-dist-na | 13.0021 | APE11-dist-na | 7.9281 | APE10-dist-na | 11.009 | APE9-dist-in | 6.3419 | V657F | None | None | EM | 5.5 | 999.0 | 999.0 | A | 1173.0 | 1047.0 | 19 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 8ewy | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |
| TYR | JAK1-12 | JAK1_MOUSE | 8EWYB | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | None | 999.0 | 999.0 | None | -138.65, -158.76 | 57.86, 53.37 | -86.37, 17.05 | 999.0, 999.0 | -66.24, -21.9 | in-none | in | 8.0788 | Saltbr-none | 999.0 | HRD-in | -63.87, -38.25 | 66.06, -1.5 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.8419 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.87, 139.06 | APE9-dihe-in | -137.62, 148.16 | APE8-dihe-in | -70.91, 80.26 | APE8-rot-na | 999.0 | APE67-dihe-in | -71.25, -12.38 | -60.08, -31.01 | APE12-dist-na | 13.0021 | APE11-dist-na | 7.9285 | APE10-dist-na | 11.0086 | APE9-dist-in | 6.3412 | V657F | None | None | EM | 5.5 | 999.0 | 999.0 | B | 1173.0 | 1047.0 | 19 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 8ewy | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | JAK1-12 | JAK1_MOUSE | 8EWYA | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | None | 999.0 | 999.0 | None | -138.68, -158.74 | 57.84, 53.41 | -86.5, 17.2 | 999.0, 999.0 | -66.33, -21.83 | in-none | in | 8.0785 | Saltbr-none | 999.0 | HRD-in | -63.86, -38.24 | 65.99, -1.42 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.8414 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.88, 139.03 | APE9-dihe-in | -137.63, 148.1 | APE8-dihe-in | -70.82, 80.23 | APE8-rot-na | 999.0 | APE67-dihe-in | -71.32, -12.38 | -60.07, -30.97 | APE12-dist-na | 13.0021 | APE11-dist-na | 7.9281 | APE10-dist-na | 11.009 | APE9-dist-in | 6.3419 | V657F | None | None | EM | 5.5 | 999.0 | 999.0 | A | 1173.0 | 1047.0 | 19 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 8ewy | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |
| TYR | JAK1-12 | JAK1_MOUSE | 8EWYB | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | None | 999.0 | 999.0 | None | -138.65, -158.76 | 57.86, 53.37 | -86.37, 17.05 | 999.0, 999.0 | -66.24, -21.9 | in-none | in | 8.0788 | Saltbr-none | 999.0 | HRD-in | -63.87, -38.25 | 66.06, -1.5 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.8419 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.87, 139.06 | APE9-dihe-in | -137.62, 148.16 | APE8-dihe-in | -70.91, 80.26 | APE8-rot-na | 999.0 | APE67-dihe-in | -71.25, -12.38 | -60.08, -31.01 | APE12-dist-na | 13.0021 | APE11-dist-na | 7.9285 | APE10-dist-na | 11.0086 | APE9-dist-in | 6.3412 | V657F | None | None | EM | 5.5 | 999.0 | 999.0 | B | 1173.0 | 1047.0 | 19 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 8ewy | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |