| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYA | P48730 | 4 | 294 | 415.0 | UX2:301 | Type1 | Active | DFGin | 6.5594 | 14.8855 | BLAminus | -133.96, 167.79 | 70.83, 96.95 | -106.29, 25.68 | 291.55, 83.04 | -66.18, -24.86 | in-in | in | 8.0753 | Saltbr-in | 3.0163 | HRD-in | -78.9, -49.6 | 75.24, 4.27 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8129 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.05, -40.09 | APE9-dihe-na | -82.1, -153.64 | APE8-dihe-in | -93.91, 137.61 | APE8-rot-in | 310.79 | APE67-dihe-in | -56.87, -39.19 | -67.48, -35.89 | APE12-dist-in | 12.8045 | APE11-dist-in | 11.4735 | APE10-dist-in | 5.9635 | APE9-dist-in | 3.855 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | A | 314.0 | 286.0 | 5 | 35 | 30 | 5 | [[9, 275]] | 1.0 | 7nzy | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYB | P48730 | 2 | 294 | 415.0 | UX2:301 | Type1 | None | DFGin | 6.5575 | 14.8824 | BLAminus | -133.2, 168.2 | 69.93, 96.11 | -104.78, 25.32 | 292.5, 81.62 | -64.88, -24.78 | in-in | in | 8.1357 | Saltbr-in | 2.965 | HRD-in | -79.22, -50.76 | 76.11, 7.31 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8899 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -70.52, -73.6 | APE9-dihe-na | -68.02, -150.38 | APE8-dihe-in | -91.32, 139.07 | APE8-rot-in | 311.34 | APE67-dihe-in | -57.14, -39.91 | -68.37, -36.29 | APE12-dist-none | 999.0 | APE11-dist-in | 11.8132 | APE10-dist-in | 6.8722 | APE9-dist-in | 3.7311 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | B | 314.0 | 286.0 | 7 | 35 | 28 | 7 | [[9, 275]] | 1.0 | 7nzy | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYC | P48730 | 3 | 294 | 415.0 | UX2:301 | Type1 | Active | DFGin | 6.2176 | 14.7908 | BLAminus | -136.64, 167.98 | 72.37, 97.2 | -107.4, 23.39 | 293.87, 95.12 | -65.21, -24.66 | in-in | in | 8.0998 | Saltbr-in | 2.7699 | HRD-in | -79.48, -51.87 | 75.69, 7.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9286 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.57, 101.78 | APE9-dihe-na | 127.22, -154.68 | APE8-dihe-in | -96.66, 135.72 | APE8-rot-in | 310.5 | APE67-dihe-in | -59.23, -39.9 | -66.83, -34.06 | APE12-dist-in | 12.3803 | APE11-dist-in | 11.857 | APE10-dist-in | 6.4832 | APE9-dist-in | 3.7789 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | C | 314.0 | 283.0 | 9 | 35 | 35 | 0 | [[9, 275]] | 1.0 | 7nzy | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYD | P48730 | 3 | 294 | 415.0 | UX2:301 | Type1 | Active | DFGin | 6.464 | 14.9368 | BLAminus | -138.25, 167.9 | 72.5, 98.99 | -108.83, 24.01 | 292.41, 92.73 | -66.77, -25.48 | in-in | in | 8.1322 | Saltbr-in | 2.8235 | HRD-in | -79.6, -51.19 | 75.63, 6.47 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8171 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -102.03, 112.87 | APE9-dihe-na | 117.74, -155.19 | APE8-dihe-in | -96.88, 133.52 | APE8-rot-in | 309.51 | APE67-dihe-in | -57.81, -40.27 | -67.41, -34.56 | APE12-dist-in | 12.5975 | APE11-dist-in | 12.323 | APE10-dist-in | 6.7621 | APE9-dist-in | 3.9211 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | D | 314.0 | 285.0 | 7 | 35 | 35 | 0 | [[9, 275]] | 1.0 | 7nzy | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYA | P48730 | 4 | 294 | 415.0 | UX2:301 | Type1 | Active | DFGin | 6.5594 | 14.8855 | BLAminus | -133.96, 167.79 | 70.83, 96.95 | -106.29, 25.68 | 291.55, 83.04 | -66.18, -24.86 | in-in | in | 8.0753 | Saltbr-in | 3.0163 | HRD-in | -78.9, -49.6 | 75.24, 4.27 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8129 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.05, -40.09 | APE9-dihe-na | -82.1, -153.64 | APE8-dihe-in | -93.91, 137.61 | APE8-rot-in | 310.79 | APE67-dihe-in | -56.87, -39.19 | -67.48, -35.89 | APE12-dist-in | 12.8045 | APE11-dist-in | 11.4735 | APE10-dist-in | 5.9635 | APE9-dist-in | 3.855 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | A | 314.0 | 286.0 | 5 | 35 | 30 | 5 | [[9, 275]] | 1.0 | 7nzy | Homo sapiens | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYB | P48730 | 2 | 294 | 415.0 | UX2:301 | Type1 | None | DFGin | 6.5575 | 14.8824 | BLAminus | -133.2, 168.2 | 69.93, 96.11 | -104.78, 25.32 | 292.5, 81.62 | -64.88, -24.78 | in-in | in | 8.1357 | Saltbr-in | 2.965 | HRD-in | -79.22, -50.76 | 76.11, 7.31 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8899 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -70.52, -73.6 | APE9-dihe-na | -68.02, -150.38 | APE8-dihe-in | -91.32, 139.07 | APE8-rot-in | 311.34 | APE67-dihe-in | -57.14, -39.91 | -68.37, -36.29 | APE12-dist-none | 999.0 | APE11-dist-in | 11.8132 | APE10-dist-in | 6.8722 | APE9-dist-in | 3.7311 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | B | 314.0 | 286.0 | 7 | 35 | 28 | 7 | [[9, 275]] | 1.0 | 7nzy | Homo sapiens | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYC | P48730 | 3 | 294 | 415.0 | UX2:301 | Type1 | Active | DFGin | 6.2176 | 14.7908 | BLAminus | -136.64, 167.98 | 72.37, 97.2 | -107.4, 23.39 | 293.87, 95.12 | -65.21, -24.66 | in-in | in | 8.0998 | Saltbr-in | 2.7699 | HRD-in | -79.48, -51.87 | 75.69, 7.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9286 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.57, 101.78 | APE9-dihe-na | 127.22, -154.68 | APE8-dihe-in | -96.66, 135.72 | APE8-rot-in | 310.5 | APE67-dihe-in | -59.23, -39.9 | -66.83, -34.06 | APE12-dist-in | 12.3803 | APE11-dist-in | 11.857 | APE10-dist-in | 6.4832 | APE9-dist-in | 3.7789 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | C | 314.0 | 283.0 | 9 | 35 | 35 | 0 | [[9, 275]] | 1.0 | 7nzy | Homo sapiens | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| CK1 | CSNK1D | KC1D_HUMAN | 7NZYD | P48730 | 3 | 294 | 415.0 | UX2:301 | Type1 | Active | DFGin | 6.464 | 14.9368 | BLAminus | -138.25, 167.9 | 72.5, 98.99 | -108.83, 24.01 | 292.41, 92.73 | -66.77, -25.48 | in-in | in | 8.1322 | Saltbr-in | 2.8235 | HRD-in | -79.6, -51.19 | 75.63, 6.47 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8171 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -102.03, 112.87 | APE9-dihe-na | 117.74, -155.19 | APE8-dihe-in | -96.88, 133.52 | APE8-rot-in | 309.51 | APE67-dihe-in | -57.81, -40.27 | -67.41, -34.56 | APE12-dist-in | 12.5975 | APE11-dist-in | 12.323 | APE10-dist-in | 6.7621 | APE9-dist-in | 3.9211 | None | TPO220 | TPO220 | XRAY | 1.85 | 0.205 | 0.229 | D | 314.0 | 285.0 | 7 | 35 | 35 | 0 | [[9, 275]] | 1.0 | 7nzy | Homo sapiens | CK1_CSNK1D_HUMAN | CK1 | 1.9e-122 | 413.6 | 1.0 | 262.0 | 262.0 | 148 | 149 | 150 | 152 | 154 | 38 | 52 | 56 | 125 | 127 | 126 | 128.0 | 195 | 183 | 178 | 177 | 176 | 175 | 174 | 173 | 172 | 83 | Casein kinase I isoform delta |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|