| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 7KIEA | P21802 | 466 | 766 | 821.0 | WF7:801 | Type1 | Inactive | DFGin | 6.9767 | 14.8481 | BLAminus | -131.39, -169.16 | 54.75, 74.84 | -95.86, 20.26 | 282.29, 75.53 | -45.07, -46.66 | in-in | in | 7.6108 | Saltbr-in | 3.0478 | HRD-in | -91.29, -46.71 | 82.94, -9.97 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9875 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -125.11, 21.7 | APE9-dihe-in | -95.02, 131.64 | APE8-dihe-in | -52.4, 118.95 | APE8-rot-na | 324.83 | APE67-dihe-in | -75.99, -13.6 | -53.13, -38.79 | APE12-dist-na | 10.0333 | APE11-dist-na | 10.7047 | APE10-dist-na | 7.4828 | APE9-dist-in | 4.8386 | V564F | None | None | XRAY | 2.47 | 0.202 | 0.229 | A | 308.0 | 291.0 | 10 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7kie | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 7KIEB | P21802 | 466 | 767 | 821.0 | WF7:801 | Type1 | Inactive | DFGin | 7.0353 | 14.8094 | BLAminus | -137.38, -176.99 | 66.42, 65.65 | -89.69, 13.43 | 284.31, 71.08 | -48.41, -38.08 | in-in | in | 7.448 | Saltbr-in | 3.2322 | HRD-in | -77.26, -55.81 | 80.7, -9.45 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8513 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.89, 17.38 | APE9-dihe-in | -97.25, 125.97 | APE8-dihe-in | -52.01, 125.72 | APE8-rot-na | 329.53 | APE67-dihe-in | -76.39, -7.41 | -69.78, -34.58 | APE12-dist-na | 10.0898 | APE11-dist-na | 10.7358 | APE10-dist-na | 7.3318 | APE9-dist-in | 4.9379 | V564F | None | None | XRAY | 2.47 | 0.202 | 0.229 | B | 308.0 | 292.0 | 10 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7kie | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 7KIEA | P21802 | 466 | 766 | 821.0 | WF7:801 | Type1 | Inactive | DFGin | 6.9767 | 14.8481 | BLAminus | -131.39, -169.16 | 54.75, 74.84 | -95.86, 20.26 | 282.29, 75.53 | -45.07, -46.66 | in-in | in | 7.6108 | Saltbr-in | 3.0478 | HRD-in | -91.29, -46.71 | 82.94, -9.97 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9875 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -125.11, 21.7 | APE9-dihe-in | -95.02, 131.64 | APE8-dihe-in | -52.4, 118.95 | APE8-rot-na | 324.83 | APE67-dihe-in | -75.99, -13.6 | -53.13, -38.79 | APE12-dist-na | 10.0333 | APE11-dist-na | 10.7047 | APE10-dist-na | 7.4828 | APE9-dist-in | 4.8386 | V564F | None | None | XRAY | 2.47 | 0.202 | 0.229 | A | 308.0 | 291.0 | 10 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7kie | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 7KIEB | P21802 | 466 | 767 | 821.0 | WF7:801 | Type1 | Inactive | DFGin | 7.0353 | 14.8094 | BLAminus | -137.38, -176.99 | 66.42, 65.65 | -89.69, 13.43 | 284.31, 71.08 | -48.41, -38.08 | in-in | in | 7.448 | Saltbr-in | 3.2322 | HRD-in | -77.26, -55.81 | 80.7, -9.45 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8513 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.89, 17.38 | APE9-dihe-in | -97.25, 125.97 | APE8-dihe-in | -52.01, 125.72 | APE8-rot-na | 329.53 | APE67-dihe-in | -76.39, -7.41 | -69.78, -34.58 | APE12-dist-na | 10.0898 | APE11-dist-na | 10.7358 | APE10-dist-na | 7.3318 | APE9-dist-in | 4.9379 | V564F | None | None | XRAY | 2.47 | 0.202 | 0.229 | B | 308.0 | 292.0 | 10 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7kie | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|