| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 7KHKA | P10721 | 566 | 931 | 976.0 | WEJ:61001 | Type1 | Active | DFGin | 6.6215 | 14.2719 | BLAminus | -140.87, -169.56 | 54.53, 74.43 | -96.38, 20.12 | 284.39, 79.52 | -61.52, -34.11 | in-in | in | 7.7962 | Saltbr-in | 2.955 | HRD-in | -71.94, -49.6 | 78.21, -7.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7743 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.36, 145.92 | APE9-dihe-in | -134.49, 154.24 | APE8-dihe-in | -84.47, 81.8 | APE8-rot-na | 31.31 | APE67-dihe-in | -63.63, -25.49 | -58.99, -41.55 | APE12-dist-na | 999.0 | APE11-dist-na | 9.1055 | APE10-dist-na | 11.1533 | APE9-dist-in | 7.1628 | None | None | None | XRAY | 2.34 | 0.247 | 0.285 | A | 335.0 | 291.0 | 17 | 30 | 28 | 2 | [[589, 926]] | 1.0 | 7khk | TYR_KIT_HUMAN | TYR | 1.1e-104 | 355.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 7KHKB | P10721 | 567 | 929 | 976.0 | WEJ:61001 | Type1.5_Back | Active | DFGin | 6.4978 | 14.2352 | BLAminus | -142.53, -172.25 | 54.51, 74.71 | -95.93, 18.48 | 280.18, 76.12 | -61.98, -36.28 | in-in | in | 7.9458 | Saltbr-in | 2.743 | HRD-in | -68.07, -48.48 | 77.89, -8.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0286 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.55, 143.65 | APE9-dihe-in | -140.59, 157.12 | APE8-dihe-in | -84.72, 84.57 | APE8-rot-na | 30.89 | APE67-dihe-in | -62.7, -33.9 | -56.2, -38.85 | APE12-dist-na | 14.3028 | APE11-dist-na | 9.1622 | APE10-dist-na | 11.3832 | APE9-dist-in | 7.1129 | None | None | None | XRAY | 2.34 | 0.247 | 0.285 | B | 335.0 | 266.0 | 39 | 30 | 28 | 2 | [[589, 926]] | 1.0 | 7khk | TYR_KIT_HUMAN | TYR | 1.1e-104 | 355.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 7KHKA | P10721 | 566 | 931 | 976.0 | WEJ:61001 | Type1 | Active | DFGin | 6.6215 | 14.2719 | BLAminus | -140.87, -169.56 | 54.53, 74.43 | -96.38, 20.12 | 284.39, 79.52 | -61.52, -34.11 | in-in | in | 7.7962 | Saltbr-in | 2.955 | HRD-in | -71.94, -49.6 | 78.21, -7.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7743 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -69.36, 145.92 | APE9-dihe-in | -134.49, 154.24 | APE8-dihe-in | -84.47, 81.8 | APE8-rot-na | 31.31 | APE67-dihe-in | -63.63, -25.49 | -58.99, -41.55 | APE12-dist-na | 999.0 | APE11-dist-na | 9.1055 | APE10-dist-na | 11.1533 | APE9-dist-in | 7.1628 | None | None | None | XRAY | 2.34 | 0.247 | 0.285 | A | 335.0 | 291.0 | 17 | 30 | 28 | 2 | [[589, 926]] | 1.0 | 7khk | Homo sapiens | TYR_KIT_HUMAN | TYR | 1.1e-104 | 355.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 7KHKB | P10721 | 567 | 929 | 976.0 | WEJ:61001 | Type1.5_Back | Active | DFGin | 6.4978 | 14.2352 | BLAminus | -142.53, -172.25 | 54.51, 74.71 | -95.93, 18.48 | 280.18, 76.12 | -61.98, -36.28 | in-in | in | 7.9458 | Saltbr-in | 2.743 | HRD-in | -68.07, -48.48 | 77.89, -8.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0286 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.55, 143.65 | APE9-dihe-in | -140.59, 157.12 | APE8-dihe-in | -84.72, 84.57 | APE8-rot-na | 30.89 | APE67-dihe-in | -62.7, -33.9 | -56.2, -38.85 | APE12-dist-na | 14.3028 | APE11-dist-na | 9.1622 | APE10-dist-na | 11.3832 | APE9-dist-in | 7.1129 | None | None | None | XRAY | 2.34 | 0.247 | 0.285 | B | 335.0 | 266.0 | 39 | 30 | 28 | 2 | [[589, 926]] | 1.0 | 7khk | Homo sapiens | TYR_KIT_HUMAN | TYR | 1.1e-104 | 355.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|