| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 7JU5A | P07949 | 705 | 1013 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.8787 | 14.8343 | BLAminus | -128.61, -171.91 | 57.52, 65.29 | -87.28, 11.68 | 279.55, 79.31 | -66.81, -20.12 | in-in | in | 7.6321 | Saltbr-in | 2.8002 | HRD-in | -84.47, -40.33 | 77.23, -28.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9549 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.3, 14.29 | APE9-dihe-in | -89.88, 135.82 | APE8-dihe-in | -53.54, 134.95 | APE8-rot-na | 328.22 | APE67-dihe-in | -68.32, -11.15 | -49.93, -45.95 | APE12-dist-na | 13.4717 | APE11-dist-na | 9.5116 | APE10-dist-na | 7.5863 | APE9-dist-in | 5.4137 | None | None | None | XRAY | 1.9 | 0.191 | 0.247 | A | 314.0 | 282.0 | 27 | 30 | 22 | 8 | [[724, 1007]] | 1.0 | 7ju5 | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 7JU5B | P07949 | 710 | 1012 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.8391 | 14.3423 | BLAminus | -134.43, -173.06 | 58.09, 64.61 | -89.98, 9.88 | 284.05, 81.83 | -62.24, -29.8 | in-in | in | 7.4654 | Saltbr-in | 2.8098 | HRD-in | -72.03, -43.23 | 72.95, -28.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8668 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.77, 15.0 | APE9-dihe-in | -82.46, 132.21 | APE8-dihe-in | -46.89, 130.57 | APE8-rot-na | 330.41 | APE67-dihe-in | -67.96, -11.33 | -51.31, -40.09 | APE12-dist-na | 13.4796 | APE11-dist-na | 9.2567 | APE10-dist-na | 7.5867 | APE9-dist-in | 5.3559 | None | None | None | XRAY | 1.9 | 0.191 | 0.247 | B | 314.0 | 290.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 7ju5 | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 7JU5A | P07949 | 705 | 1013 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.8787 | 14.8343 | BLAminus | -128.61, -171.91 | 57.52, 65.29 | -87.28, 11.68 | 279.55, 79.31 | -66.81, -20.12 | in-in | in | 7.6321 | Saltbr-in | 2.8002 | HRD-in | -84.47, -40.33 | 77.23, -28.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9549 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.3, 14.29 | APE9-dihe-in | -89.88, 135.82 | APE8-dihe-in | -53.54, 134.95 | APE8-rot-na | 328.22 | APE67-dihe-in | -68.32, -11.15 | -49.93, -45.95 | APE12-dist-na | 13.4717 | APE11-dist-na | 9.5116 | APE10-dist-na | 7.5863 | APE9-dist-in | 5.4137 | None | None | None | XRAY | 1.9 | 0.191 | 0.247 | A | 314.0 | 282.0 | 27 | 30 | 22 | 8 | [[724, 1007]] | 1.0 | 7ju5 | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 7JU5B | P07949 | 710 | 1012 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.8391 | 14.3423 | BLAminus | -134.43, -173.06 | 58.09, 64.61 | -89.98, 9.88 | 284.05, 81.83 | -62.24, -29.8 | in-in | in | 7.4654 | Saltbr-in | 2.8098 | HRD-in | -72.03, -43.23 | 72.95, -28.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8668 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.77, 15.0 | APE9-dihe-in | -82.46, 132.21 | APE8-dihe-in | -46.89, 130.57 | APE8-rot-na | 330.41 | APE67-dihe-in | -67.96, -11.33 | -51.31, -40.09 | APE12-dist-na | 13.4796 | APE11-dist-na | 9.2567 | APE10-dist-na | 7.5867 | APE9-dist-in | 5.3559 | None | None | None | XRAY | 1.9 | 0.191 | 0.247 | B | 314.0 | 290.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 7ju5 | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|