| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 7DUAA | P07949 | 712 | 1011 | 1114.0 | HJ0:61101 | Type1.5_Back | Inactive | DFGin | 7.0159 | 13.8138 | BLAminus | -133.17, -175.88 | 62.46, 70.06 | -88.8, 12.02 | 286.56, 80.96 | -63.0, -32.79 | in-in | in | 7.2365 | Saltbr-in | 2.6085 | HRD-in | -71.94, -44.64 | 75.36, -32.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.912 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.88, 16.82 | APE9-dihe-in | -86.9, 135.07 | APE8-dihe-in | -52.13, 133.31 | APE8-rot-na | 327.44 | APE67-dihe-in | -66.8, -11.83 | -51.98, -41.62 | APE12-dist-na | 13.4533 | APE11-dist-na | 9.0582 | APE10-dist-na | 7.4546 | APE9-dist-in | 5.3827 | None | None | None | XRAY | 1.64 | 0.192 | 0.218 | A | 314.0 | 287.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 7dua | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 7DUAB | P07949 | 705 | 1012 | 1114.0 | HJ0:61101 | Type1.5_Back | Inactive | DFGin | 6.8596 | 13.9741 | BLAminus | -133.96, -176.89 | 64.96, 70.22 | -90.12, 11.04 | 287.56, 76.53 | -62.89, -28.63 | in-in | in | 7.3058 | Saltbr-in | 2.746 | HRD-in | -70.74, -43.98 | 77.73, -36.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8286 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.25, 10.02 | APE9-dihe-in | -84.68, 132.89 | APE8-dihe-in | -55.12, 134.64 | APE8-rot-na | 329.21 | APE67-dihe-in | -67.4, -15.3 | -50.29, -41.81 | APE12-dist-na | 12.4118 | APE11-dist-na | 9.2712 | APE10-dist-na | 7.2352 | APE9-dist-in | 5.3643 | None | None | None | XRAY | 1.64 | 0.192 | 0.218 | B | 314.0 | 269.0 | 36 | 30 | 20 | 10 | [[724, 1007]] | 1.0 | 7dua | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 7DUAA | P07949 | 712 | 1011 | 1114.0 | HJ0:61101 | Type1.5_Back | Inactive | DFGin | 7.0159 | 13.8138 | BLAminus | -133.17, -175.88 | 62.46, 70.06 | -88.8, 12.02 | 286.56, 80.96 | -63.0, -32.79 | in-in | in | 7.2365 | Saltbr-in | 2.6085 | HRD-in | -71.94, -44.64 | 75.36, -32.55 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.912 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.88, 16.82 | APE9-dihe-in | -86.9, 135.07 | APE8-dihe-in | -52.13, 133.31 | APE8-rot-na | 327.44 | APE67-dihe-in | -66.8, -11.83 | -51.98, -41.62 | APE12-dist-na | 13.4533 | APE11-dist-na | 9.0582 | APE10-dist-na | 7.4546 | APE9-dist-in | 5.3827 | None | None | None | XRAY | 1.64 | 0.192 | 0.218 | A | 314.0 | 287.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 7dua | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 7DUAB | P07949 | 705 | 1012 | 1114.0 | HJ0:61101 | Type1.5_Back | Inactive | DFGin | 6.8596 | 13.9741 | BLAminus | -133.96, -176.89 | 64.96, 70.22 | -90.12, 11.04 | 287.56, 76.53 | -62.89, -28.63 | in-in | in | 7.3058 | Saltbr-in | 2.746 | HRD-in | -70.74, -43.98 | 77.73, -36.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8286 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.25, 10.02 | APE9-dihe-in | -84.68, 132.89 | APE8-dihe-in | -55.12, 134.64 | APE8-rot-na | 329.21 | APE67-dihe-in | -67.4, -15.3 | -50.29, -41.81 | APE12-dist-na | 12.4118 | APE11-dist-na | 9.2712 | APE10-dist-na | 7.2352 | APE9-dist-in | 5.3643 | None | None | None | XRAY | 1.64 | 0.192 | 0.218 | B | 314.0 | 269.0 | 36 | 30 | 20 | 10 | [[724, 1007]] | 1.0 | 7dua | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|