| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 7DU9A | P07949 | 714 | 1011 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.9494 | 14.1208 | BLAminus | -130.33, -174.42 | 58.73, 65.36 | -86.19, 8.31 | 283.62, 87.3 | -63.28, -29.26 | in-in | in | 7.2978 | Saltbr-in | 2.8438 | HRD-in | -74.67, -44.9 | 78.94, -42.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8619 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.78, 19.67 | APE9-dihe-in | -82.89, 134.45 | APE8-dihe-in | -52.33, 137.21 | APE8-rot-na | 323.27 | APE67-dihe-in | -68.72, -8.49 | -59.25, -37.83 | APE12-dist-na | 13.5407 | APE11-dist-na | 9.167 | APE10-dist-na | 7.5 | APE9-dist-in | 5.4743 | None | None | None | XRAY | 2.31 | 0.22 | 0.249 | A | 314.0 | 285.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 7du9 | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 7DU9B | P07949 | 705 | 1012 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.9424 | 14.8146 | BLAminus | -140.75, -174.14 | 57.44, 65.56 | -90.9, 8.95 | 281.01, 87.37 | -61.32, -27.02 | in-in | in | 7.623 | Saltbr-in | 2.94 | HRD-in | -75.71, -46.65 | 86.04, -41.97 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9371 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.69, 12.26 | APE9-dihe-in | -84.37, 136.33 | APE8-dihe-in | -56.91, 135.68 | APE8-rot-na | 327.83 | APE67-dihe-in | -66.72, -12.27 | -52.77, -41.0 | APE12-dist-na | 12.8048 | APE11-dist-na | 9.5848 | APE10-dist-na | 7.7592 | APE9-dist-in | 5.511 | None | None | None | XRAY | 2.31 | 0.22 | 0.249 | B | 314.0 | 268.0 | 36 | 30 | 20 | 10 | [[724, 1007]] | 1.0 | 7du9 | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 7DU9A | P07949 | 714 | 1011 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.9494 | 14.1208 | BLAminus | -130.33, -174.42 | 58.73, 65.36 | -86.19, 8.31 | 283.62, 87.3 | -63.28, -29.26 | in-in | in | 7.2978 | Saltbr-in | 2.8438 | HRD-in | -74.67, -44.9 | 78.94, -42.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8619 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.78, 19.67 | APE9-dihe-in | -82.89, 134.45 | APE8-dihe-in | -52.33, 137.21 | APE8-rot-na | 323.27 | APE67-dihe-in | -68.72, -8.49 | -59.25, -37.83 | APE12-dist-na | 13.5407 | APE11-dist-na | 9.167 | APE10-dist-na | 7.5 | APE9-dist-in | 5.4743 | None | None | None | XRAY | 2.31 | 0.22 | 0.249 | A | 314.0 | 285.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 7du9 | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 7DU9B | P07949 | 705 | 1012 | 1114.0 | Q4J:61101 | Type1 | Inactive | DFGin | 6.9424 | 14.8146 | BLAminus | -140.75, -174.14 | 57.44, 65.56 | -90.9, 8.95 | 281.01, 87.37 | -61.32, -27.02 | in-in | in | 7.623 | Saltbr-in | 2.94 | HRD-in | -75.71, -46.65 | 86.04, -41.97 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9371 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.69, 12.26 | APE9-dihe-in | -84.37, 136.33 | APE8-dihe-in | -56.91, 135.68 | APE8-rot-na | 327.83 | APE67-dihe-in | -66.72, -12.27 | -52.77, -41.0 | APE12-dist-na | 12.8048 | APE11-dist-na | 9.5848 | APE10-dist-na | 7.7592 | APE9-dist-in | 5.511 | None | None | None | XRAY | 2.31 | 0.22 | 0.249 | B | 314.0 | 268.0 | 36 | 30 | 20 | 10 | [[724, 1007]] | 1.0 | 7du9 | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|