| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 6NECA | P07949 | 713 | 1012 | 1114.0 | XIN:61101 | Type1.5_Back | Inactive | DFGin | 6.9546 | 14.2179 | BLAminus | -133.91, -174.29 | 60.89, 71.58 | -95.62, 14.14 | 281.92, 78.83 | -63.28, -30.8 | in-in | in | 7.4452 | Saltbr-in | 2.7339 | HRD-in | -64.75, -44.44 | 74.89, -24.66 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.808 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.85, 14.06 | APE9-dihe-in | -80.07, 133.09 | APE8-dihe-in | -50.98, 131.84 | APE8-rot-na | 329.18 | APE67-dihe-in | -66.23, -12.23 | -51.13, -39.97 | APE12-dist-na | 13.539 | APE11-dist-na | 9.1655 | APE10-dist-na | 7.4943 | APE9-dist-in | 5.3838 | None | None | None | XRAY | 1.87 | 0.196 | 0.232 | A | 314.0 | 287.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 6nec | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 6NECC | P07949 | 705 | 1012 | 1114.0 | XIN:61102 | Type1.5_Back | Inactive | DFGin | 6.9109 | 14.5461 | BLAminus | -127.42, -177.46 | 57.73, 73.5 | -96.06, 13.56 | 281.45, 72.28 | -58.66, -26.62 | in-in | in | 7.651 | Saltbr-in | 2.6262 | HRD-in | -74.42, -46.81 | 83.36, -28.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9345 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.6, 14.75 | APE9-dihe-in | -87.1, 131.84 | APE8-dihe-in | -50.39, 132.72 | APE8-rot-na | 328.71 | APE67-dihe-in | -69.0, -12.61 | -52.04, -41.84 | APE12-dist-na | 13.8521 | APE11-dist-na | 9.5393 | APE10-dist-na | 7.6385 | APE9-dist-in | 5.4708 | None | None | None | XRAY | 1.87 | 0.196 | 0.232 | C | 314.0 | 279.0 | 29 | 30 | 21 | 9 | [[724, 1007]] | 1.0 | 6nec | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 6NECA | P07949 | 713 | 1012 | 1114.0 | XIN:61101 | Type1.5_Back | Inactive | DFGin | 6.9546 | 14.2179 | BLAminus | -133.91, -174.29 | 60.89, 71.58 | -95.62, 14.14 | 281.92, 78.83 | -63.28, -30.8 | in-in | in | 7.4452 | Saltbr-in | 2.7339 | HRD-in | -64.75, -44.44 | 74.89, -24.66 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.808 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.85, 14.06 | APE9-dihe-in | -80.07, 133.09 | APE8-dihe-in | -50.98, 131.84 | APE8-rot-na | 329.18 | APE67-dihe-in | -66.23, -12.23 | -51.13, -39.97 | APE12-dist-na | 13.539 | APE11-dist-na | 9.1655 | APE10-dist-na | 7.4943 | APE9-dist-in | 5.3838 | None | None | None | XRAY | 1.87 | 0.196 | 0.232 | A | 314.0 | 287.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 6nec | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 6NECC | P07949 | 705 | 1012 | 1114.0 | XIN:61102 | Type1.5_Back | Inactive | DFGin | 6.9109 | 14.5461 | BLAminus | -127.42, -177.46 | 57.73, 73.5 | -96.06, 13.56 | 281.45, 72.28 | -58.66, -26.62 | in-in | in | 7.651 | Saltbr-in | 2.6262 | HRD-in | -74.42, -46.81 | 83.36, -28.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9345 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.6, 14.75 | APE9-dihe-in | -87.1, 131.84 | APE8-dihe-in | -50.39, 132.72 | APE8-rot-na | 328.71 | APE67-dihe-in | -69.0, -12.61 | -52.04, -41.84 | APE12-dist-na | 13.8521 | APE11-dist-na | 9.5393 | APE10-dist-na | 7.6385 | APE9-dist-in | 5.4708 | None | None | None | XRAY | 1.87 | 0.196 | 0.232 | C | 314.0 | 279.0 | 29 | 30 | 21 | 9 | [[724, 1007]] | 1.0 | 6nec | Homo sapiens | TYR_RET_HUMAN | TYR | 4.1e-101 | 343.6 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|