| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 6LVKA | P21802 | 468 | 766 | 821.0 | EVC:801 | Type1 | Inactive | DFGin | 6.619 | 14.5428 | BLAminus | -141.93, -174.02 | 55.34, 76.62 | -90.82, 24.34 | 285.38, 77.37 | -62.85, -30.59 | in-in | in | 7.7301 | Saltbr-in | 2.6843 | HRD-in | -81.18, -49.18 | 75.66, -4.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7961 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.17, 17.9 | APE9-dihe-in | -89.66, 132.44 | APE8-dihe-in | -56.46, 117.97 | APE8-rot-na | 336.42 | APE67-dihe-in | -71.4, -11.53 | -57.14, -41.35 | APE12-dist-na | 10.0448 | APE11-dist-na | 10.8094 | APE10-dist-na | 7.4432 | APE9-dist-in | 4.9356 | None | PTR561 | PTR561 | XRAY | 2.29 | 0.206 | 0.247 | A | 313.0 | 288.0 | 11 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvk | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 6LVKB | P21802 | 468 | 765 | 821.0 | EVC:801 | Type1 | Inactive | DFGin | 6.4241 | 14.4286 | BLAminus | -142.63, -167.55 | 46.22, 79.21 | -86.53, 20.35 | 286.19, 75.54 | -62.27, -23.76 | in-in | in | 7.4486 | Saltbr-in | 2.6441 | HRD-in | -74.06, -49.98 | 75.98, -4.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8063 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -116.0, 16.4 | APE9-dihe-in | -92.04, 132.11 | APE8-dihe-in | -55.72, 122.03 | APE8-rot-na | 331.04 | APE67-dihe-in | -82.5, -6.39 | -64.61, -25.66 | APE12-dist-na | 10.1609 | APE11-dist-na | 10.8497 | APE10-dist-na | 7.4958 | APE9-dist-in | 4.862 | None | PTR561 | PTR561 | XRAY | 2.29 | 0.206 | 0.247 | B | 313.0 | 286.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvk | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 6LVKA | P21802 | 468 | 766 | 821.0 | EVC:801 | Type1 | Inactive | DFGin | 6.619 | 14.5428 | BLAminus | -141.93, -174.02 | 55.34, 76.62 | -90.82, 24.34 | 285.38, 77.37 | -62.85, -30.59 | in-in | in | 7.7301 | Saltbr-in | 2.6843 | HRD-in | -81.18, -49.18 | 75.66, -4.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7961 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.17, 17.9 | APE9-dihe-in | -89.66, 132.44 | APE8-dihe-in | -56.46, 117.97 | APE8-rot-na | 336.42 | APE67-dihe-in | -71.4, -11.53 | -57.14, -41.35 | APE12-dist-na | 10.0448 | APE11-dist-na | 10.8094 | APE10-dist-na | 7.4432 | APE9-dist-in | 4.9356 | None | PTR561 | PTR561 | XRAY | 2.29 | 0.206 | 0.247 | A | 313.0 | 288.0 | 11 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvk | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 6LVKB | P21802 | 468 | 765 | 821.0 | EVC:801 | Type1 | Inactive | DFGin | 6.4241 | 14.4286 | BLAminus | -142.63, -167.55 | 46.22, 79.21 | -86.53, 20.35 | 286.19, 75.54 | -62.27, -23.76 | in-in | in | 7.4486 | Saltbr-in | 2.6441 | HRD-in | -74.06, -49.98 | 75.98, -4.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8063 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -116.0, 16.4 | APE9-dihe-in | -92.04, 132.11 | APE8-dihe-in | -55.72, 122.03 | APE8-rot-na | 331.04 | APE67-dihe-in | -82.5, -6.39 | -64.61, -25.66 | APE12-dist-na | 10.1609 | APE11-dist-na | 10.8497 | APE10-dist-na | 7.4958 | APE9-dist-in | 4.862 | None | PTR561 | PTR561 | XRAY | 2.29 | 0.206 | 0.247 | B | 313.0 | 286.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvk | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|