| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 6I82A | P07949 | 705 | 1012 | 1114.0 | H6W:61101 | Type1 | Inactive | DFGin | 6.8494 | 14.4712 | BLAminus | -128.14, -174.21 | 67.72, 61.92 | -90.26, 13.04 | 282.77, 85.15 | -61.02, -37.96 | in-in | in | 7.2917 | Saltbr-in | 2.7328 | HRD-in | -81.64, -39.67 | 73.25, -26.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8046 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -116.27, 0.25 | APE9-dihe-in | -89.57, 135.4 | APE8-dihe-in | -54.02, 135.51 | APE8-rot-na | 331.24 | APE67-dihe-in | -70.23, -12.8 | -60.25, -35.58 | APE12-dist-na | 8.5471 | APE11-dist-na | 10.359 | APE10-dist-na | 7.3971 | APE9-dist-in | 5.4905 | V804M | PTR928 | PTR928 | XRAY | 2.05 | 0.179 | 0.229 | A | 314.0 | 276.0 | 32 | 30 | 21 | 9 | [[724, 1007]] | 1.0 | 6i82 | TYR_RET_HUMAN | TYR | 2.2e-101 | 344.5 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 6I82B | P07949 | 714 | 1012 | 1114.0 | H6W:61102 | Type1 | Inactive | DFGin | 6.9541 | 13.8651 | BLAminus | -130.06, -175.77 | 62.79, 72.73 | -97.62, 2.52 | 278.58, 93.96 | -55.94, -34.07 | in-in | in | 7.211 | Saltbr-in | 3.1159 | HRD-in | -79.75, -46.53 | 78.6, -22.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.841 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.41, 14.52 | APE9-dihe-in | -83.53, 127.81 | APE8-dihe-in | -46.22, 130.06 | APE8-rot-na | 326.46 | APE67-dihe-in | -73.49, -7.07 | -47.41, -42.33 | APE12-dist-na | 13.7165 | APE11-dist-na | 9.1189 | APE10-dist-na | 7.7345 | APE9-dist-in | 5.4834 | V804M | PTR928 | PTR928 | XRAY | 2.05 | 0.179 | 0.229 | B | 314.0 | 286.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 6i82 | TYR_RET_HUMAN | TYR | 2.2e-101 | 344.5 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | RET | RET_HUMAN | 6I82A | P07949 | 705 | 1012 | 1114.0 | H6W:61101 | Type1 | Inactive | DFGin | 6.8494 | 14.4712 | BLAminus | -128.14, -174.21 | 67.72, 61.92 | -90.26, 13.04 | 282.77, 85.15 | -61.02, -37.96 | in-in | in | 7.2917 | Saltbr-in | 2.7328 | HRD-in | -81.64, -39.67 | 73.25, -26.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8046 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -116.27, 0.25 | APE9-dihe-in | -89.57, 135.4 | APE8-dihe-in | -54.02, 135.51 | APE8-rot-na | 331.24 | APE67-dihe-in | -70.23, -12.8 | -60.25, -35.58 | APE12-dist-na | 8.5471 | APE11-dist-na | 10.359 | APE10-dist-na | 7.3971 | APE9-dist-in | 5.4905 | V804M | PTR928 | PTR928 | XRAY | 2.05 | 0.179 | 0.229 | A | 314.0 | 276.0 | 32 | 30 | 21 | 9 | [[724, 1007]] | 1.0 | 6i82 | Homo sapiens | TYR_RET_HUMAN | TYR | 2.2e-101 | 344.5 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| TYR | RET | RET_HUMAN | 6I82B | P07949 | 714 | 1012 | 1114.0 | H6W:61102 | Type1 | Inactive | DFGin | 6.9541 | 13.8651 | BLAminus | -130.06, -175.77 | 62.79, 72.73 | -97.62, 2.52 | 278.58, 93.96 | -55.94, -34.07 | in-in | in | 7.211 | Saltbr-in | 3.1159 | HRD-in | -79.75, -46.53 | 78.6, -22.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.841 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.41, 14.52 | APE9-dihe-in | -83.53, 127.81 | APE8-dihe-in | -46.22, 130.06 | APE8-rot-na | 326.46 | APE67-dihe-in | -73.49, -7.07 | -47.41, -42.33 | APE12-dist-na | 13.7165 | APE11-dist-na | 9.1189 | APE10-dist-na | 7.7345 | APE9-dist-in | 5.4834 | V804M | PTR928 | PTR928 | XRAY | 2.05 | 0.179 | 0.229 | B | 314.0 | 286.0 | 13 | 30 | 30 | 0 | [[724, 1007]] | 1.0 | 6i82 | Homo sapiens | TYR_RET_HUMAN | TYR | 2.2e-101 | 344.5 | 1.0 | 261.0 | 261.0 | 891 | 892 | 893 | 895 | 897 | 758 | 775 | 779 | 871 | 873 | 872 | 874.0 | 933 | 921 | 916 | 915 | 914 | 913 | 912 | 911 | 910 | 805 | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|