| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 5UGXA | P21802 | 468 | 764 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.6569 | 14.0485 | BLAminus | -131.13, -166.11 | 46.79, 87.05 | -100.0, 21.89 | 288.47, 85.57 | -64.83, -24.6 | in-in | in | 7.6085 | Saltbr-in | 2.9922 | HRD-in | -78.16, -51.21 | 73.9, -1.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8666 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.33, 9.75 | APE9-dihe-in | -97.42, 138.88 | APE8-dihe-in | -59.74, 121.4 | APE8-rot-na | 334.26 | APE67-dihe-in | -70.7, -5.46 | -65.5, -39.78 | APE12-dist-na | 15.029 | APE11-dist-na | 11.1765 | APE10-dist-na | 7.4581 | APE9-dist-in | 4.8037 | C491A,E565A | None | None | XRAY | 2.349 | 0.22 | 0.275 | A | 324.0 | 297.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5ugx | TYR_FGFR2_HUMAN | TYR | 4.5e-103 | 350.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 5UGXB | P21802 | 468 | 764 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.7107 | 13.9229 | BLAminus | -132.31, -170.71 | 52.3, 81.71 | -96.0, 22.25 | 292.25, 87.7 | -65.69, -25.27 | in-in | in | 7.3927 | Saltbr-in | 3.1538 | HRD-in | -75.61, -53.17 | 73.28, -1.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9195 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.49, 16.52 | APE9-dihe-in | -100.17, 138.41 | APE8-dihe-in | -61.9, 122.99 | APE8-rot-na | 336.36 | APE67-dihe-in | -71.64, -5.56 | -62.65, -38.67 | APE12-dist-na | 10.081 | APE11-dist-na | 10.7661 | APE10-dist-na | 7.2815 | APE9-dist-in | 4.828 | C491A,E565A | None | None | XRAY | 2.349 | 0.22 | 0.275 | B | 324.0 | 282.0 | 15 | 30 | 20 | 10 | [[481, 759]] | 1.0 | 5ugx | TYR_FGFR2_HUMAN | TYR | 4.5e-103 | 350.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 5UGXA | P21802 | 468 | 764 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.6569 | 14.0485 | BLAminus | -131.13, -166.11 | 46.79, 87.05 | -100.0, 21.89 | 288.47, 85.57 | -64.83, -24.6 | in-in | in | 7.6085 | Saltbr-in | 2.9922 | HRD-in | -78.16, -51.21 | 73.9, -1.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8666 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.33, 9.75 | APE9-dihe-in | -97.42, 138.88 | APE8-dihe-in | -59.74, 121.4 | APE8-rot-na | 334.26 | APE67-dihe-in | -70.7, -5.46 | -65.5, -39.78 | APE12-dist-na | 15.029 | APE11-dist-na | 11.1765 | APE10-dist-na | 7.4581 | APE9-dist-in | 4.8037 | C491A,E565A | None | None | XRAY | 2.349 | 0.22 | 0.275 | A | 324.0 | 297.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5ugx | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 4.5e-103 | 350.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 5UGXB | P21802 | 468 | 764 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.7107 | 13.9229 | BLAminus | -132.31, -170.71 | 52.3, 81.71 | -96.0, 22.25 | 292.25, 87.7 | -65.69, -25.27 | in-in | in | 7.3927 | Saltbr-in | 3.1538 | HRD-in | -75.61, -53.17 | 73.28, -1.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9195 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.49, 16.52 | APE9-dihe-in | -100.17, 138.41 | APE8-dihe-in | -61.9, 122.99 | APE8-rot-na | 336.36 | APE67-dihe-in | -71.64, -5.56 | -62.65, -38.67 | APE12-dist-na | 10.081 | APE11-dist-na | 10.7661 | APE10-dist-na | 7.2815 | APE9-dist-in | 4.828 | C491A,E565A | None | None | XRAY | 2.349 | 0.22 | 0.275 | B | 324.0 | 282.0 | 15 | 30 | 20 | 10 | [[481, 759]] | 1.0 | 5ugx | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 4.5e-103 | 350.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|