| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SYK | KSYK_HUMAN | 5LMBA | P43405 | 364 | 634 | 635.0 | 6ZF:701 | Type1 | Active | DFGin | 6.4476 | 14.2826 | BLAminus | -131.02, -173.87 | 62.28, 69.39 | -93.16, 19.0 | 290.08, 82.25 | -59.68, -28.46 | in-in | in | 7.6957 | Saltbr-in | 2.454 | HRD-in | -78.06, -53.9 | 76.38, 4.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9631 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.66, 104.96 | APE9-dihe-in | -108.73, 152.4 | APE8-dihe-in | -79.7, 70.25 | APE8-rot-na | 31.84 | APE67-dihe-in | -69.34, -16.13 | -51.43, -34.69 | APE12-dist-na | 13.0735 | APE11-dist-na | 10.546 | APE10-dist-na | 11.4482 | APE9-dist-in | 6.9588 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | A | 277.0 | 265.0 | 6 | 31 | 31 | 0 | [[370, 628]] | 1.0 | 5lmb | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 5LMBB | P43405 | 364 | 630 | 635.0 | 6ZF:701 | Type1 | None | DFGin | 6.5417 | 14.2074 | BLAminus | -133.05, -174.7 | 62.98, 72.21 | -97.02, 21.38 | 290.54, 88.36 | -62.52, -32.46 | in-in | in | 7.7365 | Saltbr-in | 2.5556 | HRD-in | -77.26, -52.74 | 74.6, 8.57 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.872 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 129.43 | APE8-dihe-in | -80.7, 73.18 | APE8-rot-na | 30.16 | APE67-dihe-in | -64.42, -18.25 | -49.18, -37.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.9476 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | B | 277.0 | 262.0 | 5 | 31 | 26 | 5 | [[370, 628]] | 1.0 | 5lmb | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SYK | KSYK_HUMAN | 5LMBA | P43405 | 364 | 634 | 635.0 | 6ZF:701 | Type1 | Active | DFGin | 6.4476 | 14.2826 | BLAminus | -131.02, -173.87 | 62.28, 69.39 | -93.16, 19.0 | 290.08, 82.25 | -59.68, -28.46 | in-in | in | 7.6957 | Saltbr-in | 2.454 | HRD-in | -78.06, -53.9 | 76.38, 4.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9631 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.66, 104.96 | APE9-dihe-in | -108.73, 152.4 | APE8-dihe-in | -79.7, 70.25 | APE8-rot-na | 31.84 | APE67-dihe-in | -69.34, -16.13 | -51.43, -34.69 | APE12-dist-na | 13.0735 | APE11-dist-na | 10.546 | APE10-dist-na | 11.4482 | APE9-dist-in | 6.9588 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | A | 277.0 | 265.0 | 6 | 31 | 31 | 0 | [[370, 628]] | 1.0 | 5lmb | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 5LMBB | P43405 | 364 | 630 | 635.0 | 6ZF:701 | Type1 | None | DFGin | 6.5417 | 14.2074 | BLAminus | -133.05, -174.7 | 62.98, 72.21 | -97.02, 21.38 | 290.54, 88.36 | -62.52, -32.46 | in-in | in | 7.7365 | Saltbr-in | 2.5556 | HRD-in | -77.26, -52.74 | 74.6, 8.57 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.872 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 129.43 | APE8-dihe-in | -80.7, 73.18 | APE8-rot-na | 30.16 | APE67-dihe-in | -64.42, -18.25 | -49.18, -37.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.9476 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.178 | 0.228 | B | 277.0 | 262.0 | 5 | 31 | 26 | 5 | [[370, 628]] | 1.0 | 5lmb | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|