| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 5IA0A | P29317 | 604 | 889 | 976.0 | A5B:1001 | Type1 | None | DFGin | 5.7495 | 15.2251 | BLAminus | -131.01, -155.76 | 61.65, 69.41 | -104.69, 91.97 | 299.22, 100.6 | -172.83, 999.0 | in-in | in | 7.988 | Saltbr-in | 3.0566 | HRD-in | -80.45, -46.02 | 73.5, -13.13 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 103.13 | APE8-dihe-in | -95.39, 103.1 | APE8-rot-na | 22.72 | APE67-dihe-in | -72.64, -3.49 | -61.44, -50.98 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.6378 | None | None | None | XRAY | 1.948 | 0.194 | 0.225 | A | 306.0 | 263.0 | 23 | 31 | 12 | 19 | [[613, 873]] | 1.0 | 5ia0 | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 5IA0B | P29317 | 600 | 882 | 976.0 | A5B:1001 | Type1 | Inactive | DFGin | 5.5534 | 15.3842 | BLBminus | -126.96, -156.55 | 64.03, 67.0 | -103.77, 142.3 | 299.95, 99.48 | 123.44, 148.27 | in-in | in | 8.0855 | Saltbr-in | 3.2301 | HRD-in | -74.38, -46.39 | 76.24, -14.79 | in-out-none | SNCion | out-none | ActLoopNT-out | 10.8366 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 107.19 | APE8-dihe-in | -66.68, 140.21 | APE8-rot-na | 27.23 | APE67-dihe-in | -76.07, -2.43 | -63.36, -38.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.3318 | None | None | None | XRAY | 1.948 | 0.194 | 0.225 | B | 306.0 | 266.0 | 17 | 31 | 17 | 14 | [[613, 873]] | 1.0 | 5ia0 | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 5IA0C | P29317 | 600 | 890 | 976.0 | A5B:1001 | Type1 | Inactive | DFGin | 6.3391 | 15.0267 | BLBminus | -132.95, -162.71 | 63.9, 70.2 | -105.45, 159.62 | 303.48, 101.06 | 149.65, -160.59 | in-in | in | 8.3563 | Saltbr-in | 2.6417 | HRD-in | -77.84, -43.14 | 69.2, -7.06 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 48.26 | APE8-rot-na | 27.02 | APE67-dihe-in | -80.71, 0.8 | -57.19, -48.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.948 | 0.194 | 0.225 | C | 306.0 | 269.0 | 22 | 31 | 13 | 18 | [[613, 873]] | 1.0 | 5ia0 | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 5IA0A | P29317 | 604 | 889 | 976.0 | A5B:1001 | Type1 | None | DFGin | 5.7495 | 15.2251 | BLAminus | -131.01, -155.76 | 61.65, 69.41 | -104.69, 91.97 | 299.22, 100.6 | -172.83, 999.0 | in-in | in | 7.988 | Saltbr-in | 3.0566 | HRD-in | -80.45, -46.02 | 73.5, -13.13 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 103.13 | APE8-dihe-in | -95.39, 103.1 | APE8-rot-na | 22.72 | APE67-dihe-in | -72.64, -3.49 | -61.44, -50.98 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.6378 | None | None | None | XRAY | 1.948 | 0.194 | 0.225 | A | 306.0 | 263.0 | 23 | 31 | 12 | 19 | [[613, 873]] | 1.0 | 5ia0 | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 5IA0B | P29317 | 600 | 882 | 976.0 | A5B:1001 | Type1 | Inactive | DFGin | 5.5534 | 15.3842 | BLBminus | -126.96, -156.55 | 64.03, 67.0 | -103.77, 142.3 | 299.95, 99.48 | 123.44, 148.27 | in-in | in | 8.0855 | Saltbr-in | 3.2301 | HRD-in | -74.38, -46.39 | 76.24, -14.79 | in-out-none | SNCion | out-none | ActLoopNT-out | 10.8366 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 107.19 | APE8-dihe-in | -66.68, 140.21 | APE8-rot-na | 27.23 | APE67-dihe-in | -76.07, -2.43 | -63.36, -38.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 5.3318 | None | None | None | XRAY | 1.948 | 0.194 | 0.225 | B | 306.0 | 266.0 | 17 | 31 | 17 | 14 | [[613, 873]] | 1.0 | 5ia0 | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 5IA0C | P29317 | 600 | 890 | 976.0 | A5B:1001 | Type1 | Inactive | DFGin | 6.3391 | 15.0267 | BLBminus | -132.95, -162.71 | 63.9, 70.2 | -105.45, 159.62 | 303.48, 101.06 | 149.65, -160.59 | in-in | in | 8.3563 | Saltbr-in | 2.6417 | HRD-in | -77.84, -43.14 | 69.2, -7.06 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 48.26 | APE8-rot-na | 27.02 | APE67-dihe-in | -80.71, 0.8 | -57.19, -48.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.948 | 0.194 | 0.225 | C | 306.0 | 269.0 | 22 | 31 | 13 | 18 | [[613, 873]] | 1.0 | 5ia0 | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|