| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J99A | P21802 | 466 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.7153 | 14.1397 | BLAminus | -130.96, -174.69 | 58.83, 77.45 | -92.73, 19.29 | 291.78, 87.39 | -60.03, -34.11 | in-in | in | 7.6098 | Saltbr-in | 2.8446 | HRD-in | -78.19, -48.52 | 73.01, -4.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8606 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.36, 29.03 | APE9-dihe-in | -109.75, 138.54 | APE8-dihe-in | -57.3, 116.33 | APE8-rot-na | 330.48 | APE67-dihe-in | -70.7, -10.42 | -57.47, -40.52 | APE12-dist-na | 15.0402 | APE11-dist-na | 11.232 | APE10-dist-na | 7.9723 | APE9-dist-in | 5.1297 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | A | 324.0 | 280.0 | 19 | 30 | 26 | 4 | [[481, 759]] | 1.0 | 4j99 | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J99B | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.666 | 14.1883 | BLAminus | -133.21, -176.0 | 58.56, 76.97 | -94.04, 15.78 | 292.83, 99.53 | -58.91, -32.83 | in-in | in | 7.584 | Saltbr-in | 2.6156 | HRD-in | -76.65, -48.86 | 73.31, -6.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9004 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -118.89, 30.62 | APE9-dihe-in | -108.84, 137.25 | APE8-dihe-in | -57.12, 118.19 | APE8-rot-na | 330.19 | APE67-dihe-in | -70.1, -10.12 | -57.01, -39.76 | APE12-dist-na | 14.1481 | APE11-dist-na | 11.074 | APE10-dist-na | 8.0074 | APE9-dist-in | 5.1802 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | B | 324.0 | 291.0 | 7 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j99 | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J99C | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.8355 | 14.168 | BLAminus | -131.87, -175.54 | 59.17, 75.71 | -91.42, 19.92 | 291.67, 85.71 | -59.92, -32.59 | in-in | in | 7.6282 | Saltbr-in | 2.9134 | HRD-in | -76.88, -47.72 | 74.23, -7.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8938 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.66, 30.6 | APE9-dihe-in | -110.19, 138.06 | APE8-dihe-in | -55.44, 118.46 | APE8-rot-na | 330.51 | APE67-dihe-in | -70.73, -10.29 | -57.12, -38.65 | APE12-dist-na | 14.1212 | APE11-dist-na | 10.9538 | APE10-dist-na | 8.0502 | APE9-dist-in | 5.3615 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | C | 324.0 | 291.0 | 7 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j99 | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J99D | P21802 | 465 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5929 | 14.159 | BLAminus | -133.66, -174.57 | 58.72, 78.56 | -92.61, 20.44 | 290.96, 82.99 | -59.4, -33.38 | in-in | in | 7.6313 | Saltbr-in | 2.6395 | HRD-in | -78.38, -50.11 | 73.68, -6.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8934 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.76, 31.03 | APE9-dihe-in | -108.34, 137.61 | APE8-dihe-in | -55.35, 118.06 | APE8-rot-na | 330.85 | APE67-dihe-in | -71.9, -11.56 | -55.67, -38.95 | APE12-dist-na | 999.0 | APE11-dist-na | 11.135 | APE10-dist-na | 7.8592 | APE9-dist-in | 4.9921 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | D | 324.0 | 281.0 | 19 | 30 | 27 | 3 | [[481, 759]] | 1.0 | 4j99 | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J99A | P21802 | 466 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.7153 | 14.1397 | BLAminus | -130.96, -174.69 | 58.83, 77.45 | -92.73, 19.29 | 291.78, 87.39 | -60.03, -34.11 | in-in | in | 7.6098 | Saltbr-in | 2.8446 | HRD-in | -78.19, -48.52 | 73.01, -4.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8606 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.36, 29.03 | APE9-dihe-in | -109.75, 138.54 | APE8-dihe-in | -57.3, 116.33 | APE8-rot-na | 330.48 | APE67-dihe-in | -70.7, -10.42 | -57.47, -40.52 | APE12-dist-na | 15.0402 | APE11-dist-na | 11.232 | APE10-dist-na | 7.9723 | APE9-dist-in | 5.1297 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | A | 324.0 | 280.0 | 19 | 30 | 26 | 4 | [[481, 759]] | 1.0 | 4j99 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J99B | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.666 | 14.1883 | BLAminus | -133.21, -176.0 | 58.56, 76.97 | -94.04, 15.78 | 292.83, 99.53 | -58.91, -32.83 | in-in | in | 7.584 | Saltbr-in | 2.6156 | HRD-in | -76.65, -48.86 | 73.31, -6.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9004 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -118.89, 30.62 | APE9-dihe-in | -108.84, 137.25 | APE8-dihe-in | -57.12, 118.19 | APE8-rot-na | 330.19 | APE67-dihe-in | -70.1, -10.12 | -57.01, -39.76 | APE12-dist-na | 14.1481 | APE11-dist-na | 11.074 | APE10-dist-na | 8.0074 | APE9-dist-in | 5.1802 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | B | 324.0 | 291.0 | 7 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j99 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J99C | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.8355 | 14.168 | BLAminus | -131.87, -175.54 | 59.17, 75.71 | -91.42, 19.92 | 291.67, 85.71 | -59.92, -32.59 | in-in | in | 7.6282 | Saltbr-in | 2.9134 | HRD-in | -76.88, -47.72 | 74.23, -7.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8938 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.66, 30.6 | APE9-dihe-in | -110.19, 138.06 | APE8-dihe-in | -55.44, 118.46 | APE8-rot-na | 330.51 | APE67-dihe-in | -70.73, -10.29 | -57.12, -38.65 | APE12-dist-na | 14.1212 | APE11-dist-na | 10.9538 | APE10-dist-na | 8.0502 | APE9-dist-in | 5.3615 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | C | 324.0 | 291.0 | 7 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j99 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J99D | P21802 | 465 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5929 | 14.159 | BLAminus | -133.66, -174.57 | 58.72, 78.56 | -92.61, 20.44 | 290.96, 82.99 | -59.4, -33.38 | in-in | in | 7.6313 | Saltbr-in | 2.6395 | HRD-in | -78.38, -50.11 | 73.68, -6.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8934 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.76, 31.03 | APE9-dihe-in | -108.34, 137.61 | APE8-dihe-in | -55.35, 118.06 | APE8-rot-na | 330.85 | APE67-dihe-in | -71.9, -11.56 | -55.67, -38.95 | APE12-dist-na | 999.0 | APE11-dist-na | 11.135 | APE10-dist-na | 7.8592 | APE9-dist-in | 4.9921 | C491A,K659T | None | None | XRAY | 1.847 | 0.206 | 0.24 | D | 324.0 | 281.0 | 19 | 30 | 27 | 3 | [[481, 759]] | 1.0 | 4j99 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|