| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J97A | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.5502 | 14.1232 | BLAminus | -139.14, -173.61 | 59.78, 71.54 | -95.85, 23.3 | 290.64, 88.77 | -67.56, -16.73 | in-in | in | 7.3156 | Saltbr-in | 3.0041 | HRD-in | -83.97, -47.07 | 72.51, -7.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8773 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.39, 21.13 | APE9-dihe-in | -97.79, 130.15 | APE8-dihe-in | -58.11, 126.83 | APE8-rot-na | 332.95 | APE67-dihe-in | -66.85, -7.34 | -61.56, -42.87 | APE12-dist-na | 15.3363 | APE11-dist-na | 10.6921 | APE10-dist-na | 7.7435 | APE9-dist-in | 4.8822 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | A | 324.0 | 282.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J97B | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6186 | 14.1611 | BLAminus | -137.2, -170.97 | 56.98, 77.11 | -102.2, 28.96 | 291.71, 89.32 | -70.08, -17.2 | in-in | in | 7.4319 | Saltbr-in | 2.6835 | HRD-in | -92.02, -43.47 | 71.93, -10.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.882 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.22, 28.28 | APE9-dihe-in | -102.89, 130.04 | APE8-dihe-in | -52.94, 125.61 | APE8-rot-na | 331.88 | APE67-dihe-in | -68.38, -8.99 | -59.09, -43.64 | APE12-dist-na | 15.3327 | APE11-dist-na | 10.6375 | APE10-dist-na | 7.7777 | APE9-dist-in | 4.8875 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | B | 324.0 | 283.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J97C | P21802 | 467 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6453 | 13.9457 | BLAminus | -135.48, -176.12 | 59.98, 78.76 | -103.0, 29.61 | 294.18, 85.28 | -73.23, -9.75 | in-in | in | 7.3695 | Saltbr-in | 2.7717 | HRD-in | -84.13, -44.14 | 69.93, -6.04 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8366 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.47, 19.13 | APE9-dihe-in | -91.95, 123.86 | APE8-dihe-in | -53.96, 120.55 | APE8-rot-na | 330.23 | APE67-dihe-in | -67.12, -15.11 | -56.46, -44.57 | APE12-dist-na | 15.2845 | APE11-dist-na | 10.8279 | APE10-dist-na | 7.6387 | APE9-dist-in | 4.8499 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | C | 324.0 | 283.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J97D | P21802 | 466 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.5998 | 13.9519 | BLAminus | -140.55, -174.15 | 59.58, 71.6 | -94.76, 28.97 | 293.72, 82.5 | -71.76, -12.96 | in-in | in | 7.3264 | Saltbr-in | 3.2878 | HRD-in | -86.64, -45.82 | 71.0, -4.65 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9764 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.43, 15.17 | APE9-dihe-in | -92.91, 126.7 | APE8-dihe-in | -55.77, 123.75 | APE8-rot-na | 332.18 | APE67-dihe-in | -67.8, -5.5 | -58.98, -44.55 | APE12-dist-na | 15.1752 | APE11-dist-na | 10.8096 | APE10-dist-na | 7.6532 | APE9-dist-in | 4.7736 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | D | 324.0 | 285.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J97A | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.5502 | 14.1232 | BLAminus | -139.14, -173.61 | 59.78, 71.54 | -95.85, 23.3 | 290.64, 88.77 | -67.56, -16.73 | in-in | in | 7.3156 | Saltbr-in | 3.0041 | HRD-in | -83.97, -47.07 | 72.51, -7.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8773 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.39, 21.13 | APE9-dihe-in | -97.79, 130.15 | APE8-dihe-in | -58.11, 126.83 | APE8-rot-na | 332.95 | APE67-dihe-in | -66.85, -7.34 | -61.56, -42.87 | APE12-dist-na | 15.3363 | APE11-dist-na | 10.6921 | APE10-dist-na | 7.7435 | APE9-dist-in | 4.8822 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | A | 324.0 | 282.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J97B | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6186 | 14.1611 | BLAminus | -137.2, -170.97 | 56.98, 77.11 | -102.2, 28.96 | 291.71, 89.32 | -70.08, -17.2 | in-in | in | 7.4319 | Saltbr-in | 2.6835 | HRD-in | -92.02, -43.47 | 71.93, -10.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.882 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.22, 28.28 | APE9-dihe-in | -102.89, 130.04 | APE8-dihe-in | -52.94, 125.61 | APE8-rot-na | 331.88 | APE67-dihe-in | -68.38, -8.99 | -59.09, -43.64 | APE12-dist-na | 15.3327 | APE11-dist-na | 10.6375 | APE10-dist-na | 7.7777 | APE9-dist-in | 4.8875 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | B | 324.0 | 283.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J97C | P21802 | 467 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6453 | 13.9457 | BLAminus | -135.48, -176.12 | 59.98, 78.76 | -103.0, 29.61 | 294.18, 85.28 | -73.23, -9.75 | in-in | in | 7.3695 | Saltbr-in | 2.7717 | HRD-in | -84.13, -44.14 | 69.93, -6.04 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8366 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.47, 19.13 | APE9-dihe-in | -91.95, 123.86 | APE8-dihe-in | -53.96, 120.55 | APE8-rot-na | 330.23 | APE67-dihe-in | -67.12, -15.11 | -56.46, -44.57 | APE12-dist-na | 15.2845 | APE11-dist-na | 10.8279 | APE10-dist-na | 7.6387 | APE9-dist-in | 4.8499 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | C | 324.0 | 283.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J97D | P21802 | 466 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.5998 | 13.9519 | BLAminus | -140.55, -174.15 | 59.58, 71.6 | -94.76, 28.97 | 293.72, 82.5 | -71.76, -12.96 | in-in | in | 7.3264 | Saltbr-in | 3.2878 | HRD-in | -86.64, -45.82 | 71.0, -4.65 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9764 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.43, 15.17 | APE9-dihe-in | -92.91, 126.7 | APE8-dihe-in | -55.77, 123.75 | APE8-rot-na | 332.18 | APE67-dihe-in | -67.8, -5.5 | -58.98, -44.55 | APE12-dist-na | 15.1752 | APE11-dist-na | 10.8096 | APE10-dist-na | 7.6532 | APE9-dist-in | 4.7736 | C491A,K659E | None | None | XRAY | 2.548 | 0.202 | 0.257 | D | 324.0 | 285.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j97 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 353.9 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|