| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J96B | P21802 | 462 | 766 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.422 | 14.0694 | BLAminus | -135.07, -171.17 | 49.96, 77.75 | -93.13, 20.28 | 283.65, 85.2 | -66.67, -18.8 | in-out | in | 7.205 | Saltbr-out | 3.6908 | HRD-in | -86.85, -47.88 | 76.0, -13.66 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8113 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.69, 28.85 | APE9-dihe-in | -99.38, 128.67 | APE8-dihe-in | -54.56, 125.51 | APE8-rot-na | 329.88 | APE67-dihe-in | -70.35, -5.29 | -58.48, -39.96 | APE12-dist-na | 14.7243 | APE11-dist-na | 10.1541 | APE10-dist-na | 7.5072 | APE9-dist-in | 4.9304 | C491A,K659M | None | None | XRAY | 2.297 | 0.178 | 0.219 | B | 324.0 | 305.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j96 | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J96A | P21802 | 461 | 766 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8978 | 14.2428 | BLAminus | -129.08, -173.93 | 55.13, 75.05 | -93.92, 17.08 | 285.11, 85.16 | -64.81, -20.47 | in-in | in | 7.2911 | Saltbr-in | 3.1055 | HRD-in | -86.2, -46.65 | 77.15, -15.27 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8459 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.58, 28.84 | APE9-dihe-in | -101.23, 126.83 | APE8-dihe-in | -54.36, 124.63 | APE8-rot-na | 330.34 | APE67-dihe-in | -70.0, -5.4 | -59.65, -38.1 | APE12-dist-na | 14.9329 | APE11-dist-na | 10.2923 | APE10-dist-na | 7.4434 | APE9-dist-in | 4.9133 | C491A,K659M | None | None | XRAY | 2.297 | 0.178 | 0.219 | A | 324.0 | 302.0 | 4 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j96 | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J96B | P21802 | 462 | 766 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.422 | 14.0694 | BLAminus | -135.07, -171.17 | 49.96, 77.75 | -93.13, 20.28 | 283.65, 85.2 | -66.67, -18.8 | in-out | in | 7.205 | Saltbr-out | 3.6908 | HRD-in | -86.85, -47.88 | 76.0, -13.66 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8113 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.69, 28.85 | APE9-dihe-in | -99.38, 128.67 | APE8-dihe-in | -54.56, 125.51 | APE8-rot-na | 329.88 | APE67-dihe-in | -70.35, -5.29 | -58.48, -39.96 | APE12-dist-na | 14.7243 | APE11-dist-na | 10.1541 | APE10-dist-na | 7.5072 | APE9-dist-in | 4.9304 | C491A,K659M | None | None | XRAY | 2.297 | 0.178 | 0.219 | B | 324.0 | 305.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j96 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J96A | P21802 | 461 | 766 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8978 | 14.2428 | BLAminus | -129.08, -173.93 | 55.13, 75.05 | -93.92, 17.08 | 285.11, 85.16 | -64.81, -20.47 | in-in | in | 7.2911 | Saltbr-in | 3.1055 | HRD-in | -86.2, -46.65 | 77.15, -15.27 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8459 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.58, 28.84 | APE9-dihe-in | -101.23, 126.83 | APE8-dihe-in | -54.36, 124.63 | APE8-rot-na | 330.34 | APE67-dihe-in | -70.0, -5.4 | -59.65, -38.1 | APE12-dist-na | 14.9329 | APE11-dist-na | 10.2923 | APE10-dist-na | 7.4434 | APE9-dist-in | 4.9133 | C491A,K659M | None | None | XRAY | 2.297 | 0.178 | 0.219 | A | 324.0 | 302.0 | 4 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j96 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|