| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J95A | P21802 | 467 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6906 | 14.0578 | BLAminus | -131.56, -174.19 | 63.25, 76.63 | -98.25, 22.24 | 292.31, 85.68 | -64.6, -23.3 | in-in | in | 7.7521 | Saltbr-in | 2.8109 | HRD-in | -79.93, -52.54 | 74.87, -4.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9917 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.79, 21.67 | APE9-dihe-in | -99.53, 131.21 | APE8-dihe-in | -54.93, 120.24 | APE8-rot-na | 331.68 | APE67-dihe-in | -73.86, -8.05 | -61.39, -39.09 | APE12-dist-na | 14.7733 | APE11-dist-na | 10.9527 | APE10-dist-na | 7.48 | APE9-dist-in | 4.8674 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | A | 324.0 | 279.0 | 19 | 30 | 26 | 4 | [[481, 759]] | 1.0 | 4j95 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J95B | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6767 | 14.3781 | BLAminus | -131.79, -176.38 | 62.78, 77.42 | -96.59, 21.6 | 290.19, 86.46 | -65.99, -23.31 | in-in | in | 7.797 | Saltbr-in | 2.9027 | HRD-in | -80.06, -52.15 | 74.05, -5.91 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8975 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.95, 20.73 | APE9-dihe-in | -101.19, 131.88 | APE8-dihe-in | -53.9, 121.25 | APE8-rot-na | 331.03 | APE67-dihe-in | -73.96, -6.54 | -59.67, -39.95 | APE12-dist-na | 14.9774 | APE11-dist-na | 11.0211 | APE10-dist-na | 7.7091 | APE9-dist-in | 4.8559 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | B | 324.0 | 282.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j95 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J95C | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.762 | 14.3167 | BLAminus | -132.19, -176.54 | 63.57, 76.14 | -98.34, 23.39 | 290.03, 85.39 | -65.87, -22.89 | in-in | in | 7.7358 | Saltbr-in | 2.8246 | HRD-in | -79.64, -52.73 | 75.27, -7.0 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9588 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.5, 23.85 | APE9-dihe-in | -97.28, 128.27 | APE8-dihe-in | -54.92, 121.79 | APE8-rot-na | 330.61 | APE67-dihe-in | -73.19, -7.42 | -60.17, -39.19 | APE12-dist-na | 14.7321 | APE11-dist-na | 10.3649 | APE10-dist-na | 7.4131 | APE9-dist-in | 4.9058 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | C | 324.0 | 281.0 | 16 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j95 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J95D | P21802 | 467 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6005 | 14.0737 | BLAminus | -131.84, -175.28 | 62.91, 77.06 | -96.79, 22.82 | 289.52, 85.1 | -64.56, -22.95 | in-in | in | 7.6408 | Saltbr-in | 2.7469 | HRD-in | -80.37, -53.3 | 74.73, -6.2 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0328 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.03, 23.13 | APE9-dihe-in | -98.93, 130.46 | APE8-dihe-in | -52.66, 122.62 | APE8-rot-na | 330.72 | APE67-dihe-in | -75.07, -8.74 | -59.5, -40.3 | APE12-dist-na | 999.0 | APE11-dist-na | 10.8037 | APE10-dist-na | 7.616 | APE9-dist-in | 4.8025 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | D | 324.0 | 271.0 | 27 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 4j95 | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J95A | P21802 | 467 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6906 | 14.0578 | BLAminus | -131.56, -174.19 | 63.25, 76.63 | -98.25, 22.24 | 292.31, 85.68 | -64.6, -23.3 | in-in | in | 7.7521 | Saltbr-in | 2.8109 | HRD-in | -79.93, -52.54 | 74.87, -4.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9917 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.79, 21.67 | APE9-dihe-in | -99.53, 131.21 | APE8-dihe-in | -54.93, 120.24 | APE8-rot-na | 331.68 | APE67-dihe-in | -73.86, -8.05 | -61.39, -39.09 | APE12-dist-na | 14.7733 | APE11-dist-na | 10.9527 | APE10-dist-na | 7.48 | APE9-dist-in | 4.8674 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | A | 324.0 | 279.0 | 19 | 30 | 26 | 4 | [[481, 759]] | 1.0 | 4j95 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J95B | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6767 | 14.3781 | BLAminus | -131.79, -176.38 | 62.78, 77.42 | -96.59, 21.6 | 290.19, 86.46 | -65.99, -23.31 | in-in | in | 7.797 | Saltbr-in | 2.9027 | HRD-in | -80.06, -52.15 | 74.05, -5.91 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8975 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.95, 20.73 | APE9-dihe-in | -101.19, 131.88 | APE8-dihe-in | -53.9, 121.25 | APE8-rot-na | 331.03 | APE67-dihe-in | -73.96, -6.54 | -59.67, -39.95 | APE12-dist-na | 14.9774 | APE11-dist-na | 11.0211 | APE10-dist-na | 7.7091 | APE9-dist-in | 4.8559 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | B | 324.0 | 282.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j95 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J95C | P21802 | 468 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.762 | 14.3167 | BLAminus | -132.19, -176.54 | 63.57, 76.14 | -98.34, 23.39 | 290.03, 85.39 | -65.87, -22.89 | in-in | in | 7.7358 | Saltbr-in | 2.8246 | HRD-in | -79.64, -52.73 | 75.27, -7.0 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9588 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.5, 23.85 | APE9-dihe-in | -97.28, 128.27 | APE8-dihe-in | -54.92, 121.79 | APE8-rot-na | 330.61 | APE67-dihe-in | -73.19, -7.42 | -60.17, -39.19 | APE12-dist-na | 14.7321 | APE11-dist-na | 10.3649 | APE10-dist-na | 7.4131 | APE9-dist-in | 4.9058 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | C | 324.0 | 281.0 | 16 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j95 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J95D | P21802 | 467 | 764 | 821.0 | ACP:801 | ATPlike | Inactive | DFGin | 6.6005 | 14.0737 | BLAminus | -131.84, -175.28 | 62.91, 77.06 | -96.79, 22.82 | 289.52, 85.1 | -64.56, -22.95 | in-in | in | 7.6408 | Saltbr-in | 2.7469 | HRD-in | -80.37, -53.3 | 74.73, -6.2 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0328 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.03, 23.13 | APE9-dihe-in | -98.93, 130.46 | APE8-dihe-in | -52.66, 122.62 | APE8-rot-na | 330.72 | APE67-dihe-in | -75.07, -8.74 | -59.5, -40.3 | APE12-dist-na | 999.0 | APE11-dist-na | 10.8037 | APE10-dist-na | 7.616 | APE9-dist-in | 4.8025 | C491A,K659N | None | None | XRAY | 2.377 | 0.214 | 0.255 | D | 324.0 | 271.0 | 27 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 4j95 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|