| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SYK | KSYK_HUMAN | 3SRVA | P43405 | 364 | 634 | 635.0 | S19:1 | Type1 | Active | DFGin | 6.2782 | 14.0241 | BLAminus | -137.61, -172.24 | 65.42, 72.28 | -96.27, 25.84 | 296.23, 89.02 | -63.12, -26.69 | in-in | in | 7.7479 | Saltbr-in | 2.717 | HRD-in | -84.44, -49.93 | 72.25, 5.56 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9734 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.48, 113.26 | APE9-dihe-in | -101.68, 153.86 | APE8-dihe-in | -78.64, 68.9 | APE8-rot-na | 34.87 | APE67-dihe-in | -67.25, -14.96 | -56.26, -32.84 | APE12-dist-na | 12.9309 | APE11-dist-na | 10.491 | APE10-dist-na | 11.935 | APE9-dist-in | 7.2164 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.188 | 0.241 | A | 277.0 | 263.0 | 8 | 31 | 31 | 0 | [[370, 628]] | 1.0 | 3srv | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 3SRVB | P43405 | 364 | 632 | 635.0 | S19:2 | Type1 | Active | DFGin | 6.2831 | 14.2364 | BLAminus | -130.89, -171.96 | 62.47, 72.82 | -96.45, 25.83 | 293.72, 91.52 | -65.61, -26.16 | in-in | in | 7.6629 | Saltbr-in | 2.9666 | HRD-in | -72.4, -57.08 | 74.0, 8.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9744 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -91.35, 90.32 | APE9-dihe-in | -97.42, 146.07 | APE8-dihe-in | -79.19, 69.07 | APE8-rot-na | 34.2 | APE67-dihe-in | -70.71, -15.69 | -52.0, -32.14 | APE12-dist-na | 13.2109 | APE11-dist-na | 10.2607 | APE10-dist-na | 10.8708 | APE9-dist-in | 6.9838 | None | None | None | XRAY | 1.95 | 0.188 | 0.241 | B | 277.0 | 263.0 | 6 | 31 | 31 | 0 | [[370, 628]] | 1.0 | 3srv | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | SYK | KSYK_HUMAN | 3SRVA | P43405 | 364 | 634 | 635.0 | S19:1 | Type1 | Active | DFGin | 6.2782 | 14.0241 | BLAminus | -137.61, -172.24 | 65.42, 72.28 | -96.27, 25.84 | 296.23, 89.02 | -63.12, -26.69 | in-in | in | 7.7479 | Saltbr-in | 2.717 | HRD-in | -84.44, -49.93 | 72.25, 5.56 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9734 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.48, 113.26 | APE9-dihe-in | -101.68, 153.86 | APE8-dihe-in | -78.64, 68.9 | APE8-rot-na | 34.87 | APE67-dihe-in | -67.25, -14.96 | -56.26, -32.84 | APE12-dist-na | 12.9309 | APE11-dist-na | 10.491 | APE10-dist-na | 11.935 | APE9-dist-in | 7.2164 | None | PTR525 | PTR525 | XRAY | 1.95 | 0.188 | 0.241 | A | 277.0 | 263.0 | 8 | 31 | 31 | 0 | [[370, 628]] | 1.0 | 3srv | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| TYR | SYK | KSYK_HUMAN | 3SRVB | P43405 | 364 | 632 | 635.0 | S19:2 | Type1 | Active | DFGin | 6.2831 | 14.2364 | BLAminus | -130.89, -171.96 | 62.47, 72.82 | -96.45, 25.83 | 293.72, 91.52 | -65.61, -26.16 | in-in | in | 7.6629 | Saltbr-in | 2.9666 | HRD-in | -72.4, -57.08 | 74.0, 8.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9744 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -91.35, 90.32 | APE9-dihe-in | -97.42, 146.07 | APE8-dihe-in | -79.19, 69.07 | APE8-rot-na | 34.2 | APE67-dihe-in | -70.71, -15.69 | -52.0, -32.14 | APE12-dist-na | 13.2109 | APE11-dist-na | 10.2607 | APE10-dist-na | 10.8708 | APE9-dist-in | 6.9838 | None | None | None | XRAY | 1.95 | 0.188 | 0.241 | B | 277.0 | 263.0 | 6 | 31 | 31 | 0 | [[370, 628]] | 1.0 | 3srv | Homo sapiens | TYR_SYK_HUMAN | TYR | 4.6e-90 | 307.4 | 5.0 | 260.0 | 256.0 | 511 | 512 | 513 | 515 | 517 | 402 | 420 | 424 | 491 | 493 | 492 | 494.0 | 554 | 542 | 537 | 536 | 535 | 534 | 533 | 532 | 531 | 449 | Tyrosine-protein kinase SYK |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|