| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | JAK2-2 | JAK2_HUMAN | 3JY9A | O60674 | 842 | 1130 | 1132.0 | JZH:1 | Type1.5_Back | Active | DFGin | 6.3129 | 14.2533 | BLAminus | -123.65, -154.99 | 17.68, 87.85 | -86.97, 19.54 | 286.71, 84.2 | -50.28, -36.18 | in-in | in | 8.3206 | Saltbr-in | 2.8189 | HRD-in | -57.47, -44.36 | 69.83, -15.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.835 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.55, 129.55 | APE9-dihe-in | -129.25, 135.47 | APE8-dihe-in | -83.14, 70.63 | APE8-rot-na | 34.02 | APE67-dihe-in | -70.23, -8.08 | -50.19, -35.53 | APE12-dist-na | 10.8699 | APE11-dist-na | 9.6937 | APE10-dist-na | 9.9765 | APE9-dist-in | 7.2063 | None | PTR1007,PTR1008 | PTR1007,PTR1008 | XRAY | 2.1 | 0.201 | 0.271 | A | 311.0 | 284.0 | 5 | 31 | 31 | 0 | [[545, 807], [849, 1125]] | 2.0 | 3jy9 | TYR_JAK2-2_HUMAN | TYR | 3e-87 | 298.2 | 1.0 | 260.0 | 260.0 | 993 | 994 | 995 | 997 | 999 | 882 | 898 | 902 | 973 | 975 | 974 | 976.0 | 1036 | 1024 | 1019 | 1018 | 1017 | 1016 | 1015 | 1014 | 1013 | 930 | Tyrosine-protein kinase JAK2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | JAK2-2 | JAK2_HUMAN | 3JY9A | O60674 | 842 | 1130 | 1132.0 | JZH:1 | Type1.5_Back | Active | DFGin | 6.3129 | 14.2533 | BLAminus | -123.65, -154.99 | 17.68, 87.85 | -86.97, 19.54 | 286.71, 84.2 | -50.28, -36.18 | in-in | in | 8.3206 | Saltbr-in | 2.8189 | HRD-in | -57.47, -44.36 | 69.83, -15.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.835 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.55, 129.55 | APE9-dihe-in | -129.25, 135.47 | APE8-dihe-in | -83.14, 70.63 | APE8-rot-na | 34.02 | APE67-dihe-in | -70.23, -8.08 | -50.19, -35.53 | APE12-dist-na | 10.8699 | APE11-dist-na | 9.6937 | APE10-dist-na | 9.9765 | APE9-dist-in | 7.2063 | None | PTR1007,PTR1008 | PTR1007,PTR1008 | XRAY | 2.1 | 0.201 | 0.271 | A | 311.0 | 284.0 | 5 | 31 | 31 | 0 | [[545, 807], [849, 1125]] | 2.0 | 3jy9 | Homo sapiens | TYR_JAK2-2_HUMAN | TYR | 3e-87 | 298.2 | 1.0 | 260.0 | 260.0 | 993 | 994 | 995 | 997 | 999 | 882 | 898 | 902 | 973 | 975 | 974 | 976.0 | 1036 | 1024 | 1019 | 1018 | 1017 | 1016 | 1015 | 1014 | 1013 | 930 | Tyrosine-protein kinase JAK2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|