| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PZRA | P21802 | 468 | 765 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.5281 | 14.0867 | BLAminus | -124.48, -173.68 | 60.99, 80.27 | -100.69, 20.88 | 290.45, 81.11 | -57.12, -25.75 | in-in | in | 7.4182 | Saltbr-in | 2.6479 | HRD-in | -69.22, -43.88 | 65.36, -10.35 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8333 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.95, 17.65 | APE9-dihe-in | -96.03, 130.55 | APE8-dihe-in | -55.73, 111.71 | APE8-rot-na | 326.73 | APE67-dihe-in | -57.11, -22.38 | -39.78, -52.21 | APE12-dist-na | 9.9733 | APE11-dist-na | 10.692 | APE10-dist-na | 7.3862 | APE9-dist-in | 4.7337 | C491A,K641R | None | None | XRAY | 3.0 | 0.201 | 0.268 | A | 324.0 | 280.0 | 18 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pzr | TYR_FGFR2_HUMAN | TYR | 8.4e-104 | 352.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PZRB | P21802 | 467 | 766 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.4464 | 14.1347 | BLAminus | -124.12, -169.42 | 57.57, 72.92 | -93.39, 13.68 | 295.44, 82.57 | -53.73, -21.74 | in-in | in | 7.6343 | Saltbr-in | 2.7058 | HRD-in | -69.55, -51.19 | 76.09, -22.69 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9447 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.28, 13.02 | APE9-dihe-in | -94.85, 132.36 | APE8-dihe-in | -55.27, 118.14 | APE8-rot-na | 326.76 | APE67-dihe-in | -72.22, 2.52 | -57.29, -38.32 | APE12-dist-na | 9.9488 | APE11-dist-na | 10.9786 | APE10-dist-na | 7.5192 | APE9-dist-in | 5.0157 | C491A,K641R | None | None | XRAY | 3.0 | 0.201 | 0.268 | B | 324.0 | 282.0 | 18 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pzr | TYR_FGFR2_HUMAN | TYR | 8.4e-104 | 352.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PZRA | P21802 | 468 | 765 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.5281 | 14.0867 | BLAminus | -124.48, -173.68 | 60.99, 80.27 | -100.69, 20.88 | 290.45, 81.11 | -57.12, -25.75 | in-in | in | 7.4182 | Saltbr-in | 2.6479 | HRD-in | -69.22, -43.88 | 65.36, -10.35 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8333 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.95, 17.65 | APE9-dihe-in | -96.03, 130.55 | APE8-dihe-in | -55.73, 111.71 | APE8-rot-na | 326.73 | APE67-dihe-in | -57.11, -22.38 | -39.78, -52.21 | APE12-dist-na | 9.9733 | APE11-dist-na | 10.692 | APE10-dist-na | 7.3862 | APE9-dist-in | 4.7337 | C491A,K641R | None | None | XRAY | 3.0 | 0.201 | 0.268 | A | 324.0 | 280.0 | 18 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pzr | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 8.4e-104 | 352.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PZRB | P21802 | 467 | 766 | 821.0 | ACP:803 | ATPlike | Inactive | DFGin | 6.4464 | 14.1347 | BLAminus | -124.12, -169.42 | 57.57, 72.92 | -93.39, 13.68 | 295.44, 82.57 | -53.73, -21.74 | in-in | in | 7.6343 | Saltbr-in | 2.7058 | HRD-in | -69.55, -51.19 | 76.09, -22.69 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9447 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.28, 13.02 | APE9-dihe-in | -94.85, 132.36 | APE8-dihe-in | -55.27, 118.14 | APE8-rot-na | 326.76 | APE67-dihe-in | -72.22, 2.52 | -57.29, -38.32 | APE12-dist-na | 9.9488 | APE11-dist-na | 10.9786 | APE10-dist-na | 7.5192 | APE9-dist-in | 5.0157 | C491A,K641R | None | None | XRAY | 3.0 | 0.201 | 0.268 | B | 324.0 | 282.0 | 18 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pzr | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 8.4e-104 | 352.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|