| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PWLA | P21802 | 467 | 764 | 821.0 | ACP:300 | ATPlike | Inactive | DFGin | 6.4511 | 14.1775 | BLAminus | -131.61, -167.38 | 56.51, 73.64 | -92.98, 26.06 | 293.6, 74.93 | -63.45, -20.7 | in-in | in | 7.5864 | Saltbr-in | 2.8562 | HRD-in | -77.4, -49.09 | 71.28, -7.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8847 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.03, 20.75 | APE9-dihe-in | -94.74, 135.38 | APE8-dihe-in | -58.69, 123.68 | APE8-rot-na | 326.81 | APE67-dihe-in | -69.99, -5.92 | -52.74, -45.54 | APE12-dist-na | 10.002 | APE11-dist-na | 10.6782 | APE10-dist-na | 7.4317 | APE9-dist-in | 4.749 | C491A,N549H | None | None | XRAY | 2.4 | 0.21 | 0.238 | A | 324.0 | 284.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pwl | TYR_FGFR2_HUMAN | TYR | 3.1e-104 | 353.8 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PWLB | P21802 | 468 | 765 | 821.0 | ACP:300 | ATPlike | Inactive | DFGin | 6.4391 | 14.2798 | BLAminus | -131.94, -168.62 | 54.17, 75.02 | -93.02, 25.01 | 292.99, 76.23 | -61.28, -25.59 | in-in | in | 7.6919 | Saltbr-in | 3.0703 | HRD-in | -69.87, -47.96 | 69.48, -8.93 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9161 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.23, 16.85 | APE9-dihe-in | -95.43, 136.0 | APE8-dihe-in | -55.13, 121.27 | APE8-rot-na | 324.13 | APE67-dihe-in | -66.61, -7.86 | -55.94, -44.16 | APE12-dist-na | 10.0887 | APE11-dist-na | 10.8542 | APE10-dist-na | 7.4849 | APE9-dist-in | 4.9122 | C491A,N549H | None | None | XRAY | 2.4 | 0.21 | 0.238 | B | 324.0 | 286.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pwl | TYR_FGFR2_HUMAN | TYR | 3.1e-104 | 353.8 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PWLA | P21802 | 467 | 764 | 821.0 | ACP:300 | ATPlike | Inactive | DFGin | 6.4511 | 14.1775 | BLAminus | -131.61, -167.38 | 56.51, 73.64 | -92.98, 26.06 | 293.6, 74.93 | -63.45, -20.7 | in-in | in | 7.5864 | Saltbr-in | 2.8562 | HRD-in | -77.4, -49.09 | 71.28, -7.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8847 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.03, 20.75 | APE9-dihe-in | -94.74, 135.38 | APE8-dihe-in | -58.69, 123.68 | APE8-rot-na | 326.81 | APE67-dihe-in | -69.99, -5.92 | -52.74, -45.54 | APE12-dist-na | 10.002 | APE11-dist-na | 10.6782 | APE10-dist-na | 7.4317 | APE9-dist-in | 4.749 | C491A,N549H | None | None | XRAY | 2.4 | 0.21 | 0.238 | A | 324.0 | 284.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pwl | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 3.1e-104 | 353.8 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PWLB | P21802 | 468 | 765 | 821.0 | ACP:300 | ATPlike | Inactive | DFGin | 6.4391 | 14.2798 | BLAminus | -131.94, -168.62 | 54.17, 75.02 | -93.02, 25.01 | 292.99, 76.23 | -61.28, -25.59 | in-in | in | 7.6919 | Saltbr-in | 3.0703 | HRD-in | -69.87, -47.96 | 69.48, -8.93 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9161 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.23, 16.85 | APE9-dihe-in | -95.43, 136.0 | APE8-dihe-in | -55.13, 121.27 | APE8-rot-na | 324.13 | APE67-dihe-in | -66.61, -7.86 | -55.94, -44.16 | APE12-dist-na | 10.0887 | APE11-dist-na | 10.8542 | APE10-dist-na | 7.4849 | APE9-dist-in | 4.9122 | C491A,N549H | None | None | XRAY | 2.4 | 0.21 | 0.238 | B | 324.0 | 286.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pwl | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 3.1e-104 | 353.8 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|