| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYA | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.7496 | 14.2737 | BLAminus | -142.14, -176.01 | 63.9, 72.69 | -96.2, 30.01 | 293.76, 86.07 | -65.9, -30.73 | in-in | in | 7.5474 | Saltbr-in | 2.8523 | HRD-in | -84.99, -48.7 | 74.29, -16.98 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8094 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.15, 32.71 | APE9-dihe-in | -103.67, 126.67 | APE8-dihe-in | -51.63, 122.63 | APE8-rot-na | 323.69 | APE67-dihe-in | -64.04, -12.74 | -56.98, -40.88 | APE12-dist-na | 14.8138 | APE11-dist-na | 10.095 | APE10-dist-na | 7.5375 | APE9-dist-in | 4.9554 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | A | 324.0 | 288.0 | 10 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pvy | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYB | P21802 | 462 | 764 | 821.0 | ACP:8002 | ATPlike | Inactive | DFGin | 6.635 | 14.0654 | BLAminus | -144.27, -177.95 | 57.14, 77.78 | -93.97, 24.89 | 293.34, 84.21 | -55.49, -34.1 | in-in | in | 7.3161 | Saltbr-in | 2.8469 | HRD-in | -81.21, -48.71 | 71.97, -12.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8523 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.68, 30.22 | APE9-dihe-in | -107.46, 135.49 | APE8-dihe-in | -57.98, 120.91 | APE8-rot-na | 329.38 | APE67-dihe-in | -64.69, -5.42 | -51.47, -46.8 | APE12-dist-na | 999.0 | APE11-dist-na | 10.6935 | APE10-dist-na | 7.435 | APE9-dist-in | 5.0657 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | B | 324.0 | 286.0 | 17 | 30 | 24 | 6 | [[481, 759]] | 1.0 | 2pvy | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYC | P21802 | 462 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.6933 | 14.018 | BLAminus | -131.41, -174.32 | 49.42, 82.58 | -94.81, 27.78 | 293.52, 79.4 | -60.72, -24.91 | in-in | in | 7.2286 | Saltbr-in | 3.5766 | HRD-in | -81.5, -47.6 | 72.07, -14.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7937 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.89, 24.55 | APE9-dihe-in | -101.87, 134.03 | APE8-dihe-in | -55.3, 120.87 | APE8-rot-na | 330.19 | APE67-dihe-in | -64.04, -6.89 | -51.83, -46.76 | APE12-dist-na | 14.3155 | APE11-dist-na | 10.3228 | APE10-dist-na | 7.4377 | APE9-dist-in | 5.0687 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | C | 324.0 | 285.0 | 18 | 30 | 25 | 5 | [[481, 759]] | 1.0 | 2pvy | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYD | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.9442 | 14.2611 | BLAminus | -139.76, -174.3 | 61.15, 74.17 | -97.41, 31.68 | 293.81, 79.18 | -66.75, -30.92 | in-in | in | 7.2983 | Saltbr-in | 3.0357 | HRD-in | -85.65, -49.02 | 75.46, -18.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8112 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.37, 33.11 | APE9-dihe-in | -102.8, 126.29 | APE8-dihe-in | -51.84, 123.89 | APE8-rot-na | 324.49 | APE67-dihe-in | -63.66, -13.12 | -61.69, -37.66 | APE12-dist-na | 14.8282 | APE11-dist-na | 10.0923 | APE10-dist-na | 7.5701 | APE9-dist-in | 4.9682 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | D | 324.0 | 283.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pvy | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYA | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.7496 | 14.2737 | BLAminus | -142.14, -176.01 | 63.9, 72.69 | -96.2, 30.01 | 293.76, 86.07 | -65.9, -30.73 | in-in | in | 7.5474 | Saltbr-in | 2.8523 | HRD-in | -84.99, -48.7 | 74.29, -16.98 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8094 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.15, 32.71 | APE9-dihe-in | -103.67, 126.67 | APE8-dihe-in | -51.63, 122.63 | APE8-rot-na | 323.69 | APE67-dihe-in | -64.04, -12.74 | -56.98, -40.88 | APE12-dist-na | 14.8138 | APE11-dist-na | 10.095 | APE10-dist-na | 7.5375 | APE9-dist-in | 4.9554 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | A | 324.0 | 288.0 | 10 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pvy | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYB | P21802 | 462 | 764 | 821.0 | ACP:8002 | ATPlike | Inactive | DFGin | 6.635 | 14.0654 | BLAminus | -144.27, -177.95 | 57.14, 77.78 | -93.97, 24.89 | 293.34, 84.21 | -55.49, -34.1 | in-in | in | 7.3161 | Saltbr-in | 2.8469 | HRD-in | -81.21, -48.71 | 71.97, -12.52 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8523 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.68, 30.22 | APE9-dihe-in | -107.46, 135.49 | APE8-dihe-in | -57.98, 120.91 | APE8-rot-na | 329.38 | APE67-dihe-in | -64.69, -5.42 | -51.47, -46.8 | APE12-dist-na | 999.0 | APE11-dist-na | 10.6935 | APE10-dist-na | 7.435 | APE9-dist-in | 5.0657 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | B | 324.0 | 286.0 | 17 | 30 | 24 | 6 | [[481, 759]] | 1.0 | 2pvy | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYC | P21802 | 462 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.6933 | 14.018 | BLAminus | -131.41, -174.32 | 49.42, 82.58 | -94.81, 27.78 | 293.52, 79.4 | -60.72, -24.91 | in-in | in | 7.2286 | Saltbr-in | 3.5766 | HRD-in | -81.5, -47.6 | 72.07, -14.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7937 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.89, 24.55 | APE9-dihe-in | -101.87, 134.03 | APE8-dihe-in | -55.3, 120.87 | APE8-rot-na | 330.19 | APE67-dihe-in | -64.04, -6.89 | -51.83, -46.76 | APE12-dist-na | 14.3155 | APE11-dist-na | 10.3228 | APE10-dist-na | 7.4377 | APE9-dist-in | 5.0687 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | C | 324.0 | 285.0 | 18 | 30 | 25 | 5 | [[481, 759]] | 1.0 | 2pvy | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PVYD | P21802 | 467 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.9442 | 14.2611 | BLAminus | -139.76, -174.3 | 61.15, 74.17 | -97.41, 31.68 | 293.81, 79.18 | -66.75, -30.92 | in-in | in | 7.2983 | Saltbr-in | 3.0357 | HRD-in | -85.65, -49.02 | 75.46, -18.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8112 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.37, 33.11 | APE9-dihe-in | -102.8, 126.29 | APE8-dihe-in | -51.84, 123.89 | APE8-rot-na | 324.49 | APE67-dihe-in | -63.66, -13.12 | -61.69, -37.66 | APE12-dist-na | 14.8282 | APE11-dist-na | 10.0923 | APE10-dist-na | 7.5701 | APE9-dist-in | 4.9682 | C491A,K659N | None | None | XRAY | 2.2 | 0.236 | 0.276 | D | 324.0 | 283.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2pvy | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.8e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|