| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PSQA | P21802 | 468 | 765 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.875 | 13.7212 | BLAminus | -128.93, -172.72 | 52.18, 79.93 | -92.08, 23.28 | 298.98, 73.8 | -58.43, -25.99 | in-in | in | 7.4798 | Saltbr-in | 3.1998 | HRD-in | -73.69, -49.43 | 74.12, -12.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9464 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.29, 16.98 | APE9-dihe-in | -98.81, 130.21 | APE8-dihe-in | -53.9, 115.54 | APE8-rot-na | 323.02 | APE67-dihe-in | -67.54, -7.82 | -55.22, -37.78 | APE12-dist-na | 10.1238 | APE11-dist-na | 10.6949 | APE10-dist-na | 7.2102 | APE9-dist-in | 5.0417 | None | None | None | XRAY | 2.4 | 0.211 | 0.258 | A | 370.0 | 287.0 | 11 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2psq | TYR_FGFR2_HUMAN | TYR | 4.5e-104 | 353.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PSQB | P21802 | 467 | 766 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.661 | 13.8383 | BLAminus | -134.84, -175.34 | 56.99, 78.24 | -93.68, 24.63 | 295.92, 77.95 | -61.79, -34.13 | in-in | in | 7.4112 | Saltbr-in | 2.6888 | HRD-in | -74.4, -46.06 | 70.25, -13.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8711 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.1, 12.51 | APE9-dihe-in | -92.24, 130.01 | APE8-dihe-in | -52.44, 120.68 | APE8-rot-na | 324.14 | APE67-dihe-in | -73.23, -4.23 | -55.2, -38.33 | APE12-dist-na | 9.9488 | APE11-dist-na | 10.675 | APE10-dist-na | 7.2062 | APE9-dist-in | 5.0225 | None | None | None | XRAY | 2.4 | 0.211 | 0.258 | B | 370.0 | 286.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2psq | TYR_FGFR2_HUMAN | TYR | 4.5e-104 | 353.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PSQA | P21802 | 468 | 765 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.875 | 13.7212 | BLAminus | -128.93, -172.72 | 52.18, 79.93 | -92.08, 23.28 | 298.98, 73.8 | -58.43, -25.99 | in-in | in | 7.4798 | Saltbr-in | 3.1998 | HRD-in | -73.69, -49.43 | 74.12, -12.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9464 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.29, 16.98 | APE9-dihe-in | -98.81, 130.21 | APE8-dihe-in | -53.9, 115.54 | APE8-rot-na | 323.02 | APE67-dihe-in | -67.54, -7.82 | -55.22, -37.78 | APE12-dist-na | 10.1238 | APE11-dist-na | 10.6949 | APE10-dist-na | 7.2102 | APE9-dist-in | 5.0417 | None | None | None | XRAY | 2.4 | 0.211 | 0.258 | A | 370.0 | 287.0 | 11 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2psq | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 4.5e-104 | 353.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PSQB | P21802 | 467 | 766 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.661 | 13.8383 | BLAminus | -134.84, -175.34 | 56.99, 78.24 | -93.68, 24.63 | 295.92, 77.95 | -61.79, -34.13 | in-in | in | 7.4112 | Saltbr-in | 2.6888 | HRD-in | -74.4, -46.06 | 70.25, -13.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8711 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.1, 12.51 | APE9-dihe-in | -92.24, 130.01 | APE8-dihe-in | -52.44, 120.68 | APE8-rot-na | 324.14 | APE67-dihe-in | -73.23, -4.23 | -55.2, -38.33 | APE12-dist-na | 9.9488 | APE11-dist-na | 10.675 | APE10-dist-na | 7.2062 | APE9-dist-in | 5.0225 | None | None | None | XRAY | 2.4 | 0.211 | 0.258 | B | 370.0 | 286.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2psq | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 4.5e-104 | 353.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|