| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 1PKGA | P10721 | 567 | 927 | 976.0 | ADP:1480 | ATPlike | Inactive | DFGin | 6.4807 | 14.1365 | BLAminus | -130.56, -161.98 | 47.26, 79.76 | -98.59, 34.29 | 290.92, 88.36 | -71.71, -28.0 | in-out | in | 8.1383 | Saltbr-out | 3.8827 | HRD-in | -70.61, -44.29 | 71.47, -6.33 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.9813 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 81.05, 87.98 | APE9-dihe-in | -123.34, 167.37 | APE8-dihe-in | -84.87, 64.98 | APE8-rot-na | 27.08 | APE67-dihe-in | -64.22, -13.25 | -46.84, -45.75 | APE12-dist-na | 14.8174 | APE11-dist-na | 9.099 | APE10-dist-na | 11.173 | APE9-dist-in | 6.8945 | None | PTR568,PTR570 | PTR568,PTR570 | XRAY | 2.9 | 0.229 | 0.311 | A | 329.0 | 292.0 | 11 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 1pkg | TYR_KIT_HUMAN | TYR | 4.5e-102 | 346.9 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 1PKGB | P10721 | 566 | 929 | 976.0 | ADP:1486 | ATPlike | None | DFGin | 6.5368 | 13.8185 | BLAminus | -133.94, -165.75 | 57.9, 93.59 | -119.64, 36.22 | 290.23, 87.19 | -80.39, -20.36 | in-in | in | 6.9344 | Saltbr-in | 2.9154 | HRD-in | -72.14, -51.55 | 69.69, 17.19 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8877 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 110.55 | APE9-dihe-in | -141.29, 162.93 | APE8-dihe-in | -80.26, 78.25 | APE8-rot-na | 29.66 | APE67-dihe-in | -62.74, -24.13 | -40.98, -43.63 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.7652 | APE9-dist-in | 6.4939 | None | PTR568,PTR570 | PTR568,PTR570 | XRAY | 2.9 | 0.229 | 0.311 | B | 329.0 | 279.0 | 27 | 30 | 17 | 13 | [[589, 926]] | 1.0 | 1pkg | TYR_KIT_HUMAN | TYR | 4.5e-102 | 346.9 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 1PKGA | P10721 | 567 | 927 | 976.0 | ADP:1480 | ATPlike | Inactive | DFGin | 6.4807 | 14.1365 | BLAminus | -130.56, -161.98 | 47.26, 79.76 | -98.59, 34.29 | 290.92, 88.36 | -71.71, -28.0 | in-out | in | 8.1383 | Saltbr-out | 3.8827 | HRD-in | -70.61, -44.29 | 71.47, -6.33 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.9813 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 81.05, 87.98 | APE9-dihe-in | -123.34, 167.37 | APE8-dihe-in | -84.87, 64.98 | APE8-rot-na | 27.08 | APE67-dihe-in | -64.22, -13.25 | -46.84, -45.75 | APE12-dist-na | 14.8174 | APE11-dist-na | 9.099 | APE10-dist-na | 11.173 | APE9-dist-in | 6.8945 | None | PTR568,PTR570 | PTR568,PTR570 | XRAY | 2.9 | 0.229 | 0.311 | A | 329.0 | 292.0 | 11 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 1pkg | Homo sapiens | TYR_KIT_HUMAN | TYR | 4.5e-102 | 346.9 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 1PKGB | P10721 | 566 | 929 | 976.0 | ADP:1486 | ATPlike | None | DFGin | 6.5368 | 13.8185 | BLAminus | -133.94, -165.75 | 57.9, 93.59 | -119.64, 36.22 | 290.23, 87.19 | -80.39, -20.36 | in-in | in | 6.9344 | Saltbr-in | 2.9154 | HRD-in | -72.14, -51.55 | 69.69, 17.19 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8877 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 110.55 | APE9-dihe-in | -141.29, 162.93 | APE8-dihe-in | -80.26, 78.25 | APE8-rot-na | 29.66 | APE67-dihe-in | -62.74, -24.13 | -40.98, -43.63 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.7652 | APE9-dist-in | 6.4939 | None | PTR568,PTR570 | PTR568,PTR570 | XRAY | 2.9 | 0.229 | 0.311 | B | 329.0 | 279.0 | 27 | 30 | 17 | 13 | [[589, 926]] | 1.0 | 1pkg | Homo sapiens | TYR_KIT_HUMAN | TYR | 4.5e-102 | 346.9 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|