| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 1MQBA | P29317 | 605 | 887 | 976.0 | ANP:1000 | ATPlike | Inactive | DFGin | 5.7122 | 14.9239 | BLAminus | -127.53, -172.03 | 57.53, 74.63 | -109.94, 122.74 | 306.64, 100.38 | 176.53, 104.78 | in-out | in | 8.4647 | Saltbr-out | 5.6749 | HRD-in | -62.1, -45.48 | 77.42, -17.66 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -37.06 | APE9-dihe-in | -88.14, 119.95 | APE8-dihe-in | -73.81, 144.85 | APE8-rot-na | 33.04 | APE67-dihe-in | -82.72, 0.0 | -54.3, -43.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 9.5534 | APE9-dist-in | 5.5976 | None | None | None | XRAY | 2.3 | 0.237 | 0.288 | A | 333.0 | 263.0 | 20 | 31 | 14 | 17 | [[613, 873]] | 1.0 | 1mqb | TYR_EPHA2_HUMAN | TYR | 7.4e-108 | 365.7 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 1MQBB | P29317 | 602 | 883 | 976.0 | ANP:1001 | ATPlike | None | DFGin | 5.6905 | 14.8889 | BLAminus | -139.65, -173.77 | 51.28, 81.33 | -92.67, 10.65 | 292.99, 95.58 | -41.77, -44.65 | in-in | in | 8.2733 | Saltbr-in | 2.6399 | HRD-in | -72.65, -50.06 | 79.19, -16.04 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9923 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -50.3 | APE9-dihe-in | -134.32, 148.66 | APE8-dihe-in | -83.15, 83.63 | APE8-rot-na | 31.61 | APE67-dihe-in | -80.07, -2.61 | -53.54, -47.95 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.3278 | APE9-dist-in | 6.6333 | None | None | None | XRAY | 2.3 | 0.237 | 0.288 | B | 333.0 | 265.0 | 17 | 31 | 18 | 13 | [[613, 873]] | 1.0 | 1mqb | TYR_EPHA2_HUMAN | TYR | 7.4e-108 | 365.7 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 1MQBA | P29317 | 605 | 887 | 976.0 | ANP:1000 | ATPlike | Inactive | DFGin | 5.7122 | 14.9239 | BLAminus | -127.53, -172.03 | 57.53, 74.63 | -109.94, 122.74 | 306.64, 100.38 | 176.53, 104.78 | in-out | in | 8.4647 | Saltbr-out | 5.6749 | HRD-in | -62.1, -45.48 | 77.42, -17.66 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -37.06 | APE9-dihe-in | -88.14, 119.95 | APE8-dihe-in | -73.81, 144.85 | APE8-rot-na | 33.04 | APE67-dihe-in | -82.72, 0.0 | -54.3, -43.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 9.5534 | APE9-dist-in | 5.5976 | None | None | None | XRAY | 2.3 | 0.237 | 0.288 | A | 333.0 | 263.0 | 20 | 31 | 14 | 17 | [[613, 873]] | 1.0 | 1mqb | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 7.4e-108 | 365.7 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 1MQBB | P29317 | 602 | 883 | 976.0 | ANP:1001 | ATPlike | None | DFGin | 5.6905 | 14.8889 | BLAminus | -139.65, -173.77 | 51.28, 81.33 | -92.67, 10.65 | 292.99, 95.58 | -41.77, -44.65 | in-in | in | 8.2733 | Saltbr-in | 2.6399 | HRD-in | -72.65, -50.06 | 79.19, -16.04 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9923 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -50.3 | APE9-dihe-in | -134.32, 148.66 | APE8-dihe-in | -83.15, 83.63 | APE8-rot-na | 31.61 | APE67-dihe-in | -80.07, -2.61 | -53.54, -47.95 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.3278 | APE9-dist-in | 6.6333 | None | None | None | XRAY | 2.3 | 0.237 | 0.288 | B | 333.0 | 265.0 | 17 | 31 | 18 | 13 | [[613, 873]] | 1.0 | 1mqb | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 7.4e-108 | 365.7 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|