Ligand: R78

Total number of chains: 7
Active chains: 1
Total number of genes: 3
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 7 100.0% 2RKUA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CAMK CAMKK2 KKCC2_HUMAN 6BQQA Q96RR4 161 448 588.0 R78:60501 Type1 Active DFGin 6.5868 15.2478 BLAminus -117.25, 175.16 63.58, 81.13 -94.81, 22.39 287.89, 75.14 -58.43, -30.74 out-in out 10.0035 Saltbr-in 3.0722 HRD-in -71.13, -51.2 74.86, 1.34 in-in-in SNCiii in-in ActLoopNT-in 2.8393 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.24, 165.59 APE9-dihe-na 119.03, -163.74 APE8-dihe-in -97.53, 123.98 APE8-rot-in 297.33 APE67-dihe-in -61.07, -18.54 -48.02, -46.96 APE12-dist-in 8.8723 APE11-dist-in 11.3745 APE10-dist-in 5.4537 APE9-dist-in 3.4896 None None None XRAY 1.8 0.192 0.228 A 291.0 269.0 19 28 28 0 [[165, 446]] 1.0 6bqq CAMK_CAMKK2_HUMAN CAMK 1.2e-73 253.6 1.0 256.0 256.0 329 330 331 333 335 194 236 240 309 311 310 312.0 372 357 352 351 350 349 348 347 346 268 Calcium/calmodulin-dependent protein kinase kinase 2
CAMK PLK1 PLK1_HUMAN 9R8CA P53350 38 326 603.0 R78:1001 Type1 Inactive DFGin 5.5848 14.99 BLAminus -126.1, -176.63 65.4, 78.62 -95.8, 30.2 285.88, 88.19 -70.16, -23.86 in-in in 9.0969 Saltbr-in 2.8706 HRD-in -73.52, -53.38 78.38, -0.66 in-in-out SNCiio in-out ActLoopNT-in 2.9616 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.03, 32.02 APE9-dihe-na 163.26, -177.26 APE8-dihe-in -109.84, 116.09 APE8-rot-in 291.16 APE67-dihe-out -62.02, -59.2 -61.3, 153.09 APE12-dist-in 10.4112 APE11-dist-out 6.2561 APE10-dist-in 5.7623 APE9-dist-out 8.6225 None None None XRAY 2.243 0.191 0.236 A 315.0 289.0 0 28 28 0 [[53, 305]] 1.0 9r8c CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 9R8CB P53350 38 323 603.0 R78:1001 Type1 Inactive DFGin 5.5457 14.9956 BLAminus -130.55, -176.06 59.62, 83.99 -94.79, 30.62 285.83, 86.69 -68.45, -26.03 in-in in 9.1508 Saltbr-in 2.7676 HRD-in -75.84, -53.52 77.99, 2.7 in-in-out SNCiio in-out ActLoopNT-in 2.9529 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.08, 50.7 APE9-dihe-na 152.38, 176.7 APE8-dihe-in -113.61, 115.98 APE8-rot-in 316.69 APE67-dihe-out -67.47, -56.35 -62.32, 152.06 APE12-dist-in 9.9595 APE11-dist-out 7.059 APE10-dist-in 6.6227 APE9-dist-out 8.5077 None None None XRAY 2.243 0.191 0.236 B 315.0 286.0 0 28 28 0 [[53, 305]] 1.0 9r8c CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 2RKUA P53350 37 330 603.0 R78:500 Type1 Inactive DFGin 5.6778 15.0171 BLAminus -134.22, -169.5 54.06, 79.11 -86.67, 25.63 283.82, 88.21 -64.51, -26.07 in-in in 9.7168 Saltbr-in 3.0799 HRD-in -74.95, -48.26 75.93, -2.57 in-in-out SNCiio in-out ActLoopNT-in 2.9425 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -90.21, 90.69 APE9-dihe-na 162.46, 178.28 APE8-dihe-in -124.7, 88.6 APE8-rot-in 309.54 APE67-dihe-out -73.41, -64.04 -71.02, 160.05 APE12-dist-in 10.9294 APE11-dist-out 7.2828 APE10-dist-in 7.9206 APE9-dist-out 8.1342 T210V None None XRAY 1.95 0.192 0.241 A 294.0 294.0 0 28 28 0 [[53, 305]] 1.0 2rku CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 9R1XA P53350 39 334 603.0 R78:401 Type1 Inactive DFGin 5.4509 14.7459 BLAminus -129.34, -169.27 61.33, 81.84 -99.46, 30.78 291.65, 94.79 -60.61, -43.02 in-in in 9.6846 Saltbr-in 2.7211 HRD-in -71.39, -48.31 73.02, 3.83 in-in-out SNCiio in-out ActLoopNT-in 2.9715 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.63, 46.88 APE9-dihe-na 161.22, 163.69 APE8-dihe-in -103.28, 108.1 APE8-rot-in 301.35 APE67-dihe-out -58.97, -56.16 -54.1, 148.74 APE12-dist-in 10.3877 APE11-dist-out 6.5599 APE10-dist-in 6.7414 APE9-dist-out 8.5087 K225D,K226A None None XRAY 2.84 0.222 0.277 A 325.0 296.0 0 28 28 0 [[53, 305]] 1.0 9r1x CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 9R1XB P53350 39 326 603.0 R78:401 Type1 Inactive DFGin 5.4448 14.7258 BLAminus -129.89, -169.09 62.76, 81.42 -99.44, 28.81 292.45, 94.66 -58.03, -43.63 in-in in 9.6661 Saltbr-in 2.714 HRD-in -71.6, -47.96 72.32, 5.61 in-in-out SNCiio in-out ActLoopNT-in 2.9664 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -82.43, 34.44 APE9-dihe-na 160.48, 165.73 APE8-dihe-in -102.91, 108.17 APE8-rot-in 301.26 APE67-dihe-out -58.46, -55.69 -54.97, 148.64 APE12-dist-in 10.4044 APE11-dist-out 6.5324 APE10-dist-in 5.999 APE9-dist-out 8.4468 K225D,K226A None None XRAY 2.84 0.222 0.277 B 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1x CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK2 PLK2_HUMAN 4I5MA Q9NYY3 71 354 685.0 R78:60401 Type1 Inactive DFGin 6.1179 14.6063 BLAminus -135.0, -176.4 62.06, 78.64 -90.58, 19.32 306.45, 87.75 -51.33, -30.59 in-in in 9.2706 Saltbr-in 2.7444 HRD-in -74.53, -53.1 71.46, 0.19 in-in-out SNCiio in-out ActLoopNT-in 2.6631 ActLoopCT-out nonTYR APEdihe_aanoo APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 115.38 APE8-rot-out 169.65 APE67-dihe-out -76.41, -43.82 -77.31, 170.4 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 C83S,V87T,A119S,A216S,C259A,C291S,L335T None None XRAY 1.801 0.324 0.392 A 308.0 273.0 11 28 17 11 [[82, 334]] 1.0 4i5m CAMK_PLK2_HUMAN CAMK 2.6e-82 281.9 1.0 256.0 256.0 222 223 224 226 228 111 130 134 202 204 203 205.0 262 250 245 244 243 242 241 240 239 160 Serine/threonine-protein kinase PLK2

Ligand: R78

Total number of chains: 7
Active chains: 1
Total number of genes: 3
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 7 100.0% 2RKUA

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CAMK CAMKK2 KKCC2_HUMAN 6BQQA Q96RR4 161 448 588.0 R78:60501 Type1 Active DFGin 6.5868 15.2478 BLAminus -117.25, 175.16 63.58, 81.13 -94.81, 22.39 287.89, 75.14 -58.43, -30.74 out-in out 10.0035 Saltbr-in 3.0722 HRD-in -71.13, -51.2 74.86, 1.34 in-in-in SNCiii in-in ActLoopNT-in 2.8393 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.24, 165.59 APE9-dihe-na 119.03, -163.74 APE8-dihe-in -97.53, 123.98 APE8-rot-in 297.33 APE67-dihe-in -61.07, -18.54 -48.02, -46.96 APE12-dist-in 8.8723 APE11-dist-in 11.3745 APE10-dist-in 5.4537 APE9-dist-in 3.4896 None None None XRAY 1.8 0.192 0.228 A 291.0 269.0 19 28 28 0 [[165, 446]] 1.0 6bqq Homo sapiens CAMK_CAMKK2_HUMAN CAMK 1.2e-73 253.6 1.0 256.0 256.0 329 330 331 333 335 194 236 240 309 311 310 312.0 372 357 352 351 350 349 348 347 346 268 Calcium/calmodulin-dependent protein kinase kinase 2
CAMK PLK1 PLK1_HUMAN 9R8CA P53350 38 326 603.0 R78:1001 Type1 Inactive DFGin 5.5848 14.99 BLAminus -126.1, -176.63 65.4, 78.62 -95.8, 30.2 285.88, 88.19 -70.16, -23.86 in-in in 9.0969 Saltbr-in 2.8706 HRD-in -73.52, -53.38 78.38, -0.66 in-in-out SNCiio in-out ActLoopNT-in 2.9616 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.03, 32.02 APE9-dihe-na 163.26, -177.26 APE8-dihe-in -109.84, 116.09 APE8-rot-in 291.16 APE67-dihe-out -62.02, -59.2 -61.3, 153.09 APE12-dist-in 10.4112 APE11-dist-out 6.2561 APE10-dist-in 5.7623 APE9-dist-out 8.6225 None None None XRAY 2.243 0.191 0.236 A 315.0 289.0 0 28 28 0 [[53, 305]] 1.0 9r8c Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 9R8CB P53350 38 323 603.0 R78:1001 Type1 Inactive DFGin 5.5457 14.9956 BLAminus -130.55, -176.06 59.62, 83.99 -94.79, 30.62 285.83, 86.69 -68.45, -26.03 in-in in 9.1508 Saltbr-in 2.7676 HRD-in -75.84, -53.52 77.99, 2.7 in-in-out SNCiio in-out ActLoopNT-in 2.9529 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.08, 50.7 APE9-dihe-na 152.38, 176.7 APE8-dihe-in -113.61, 115.98 APE8-rot-in 316.69 APE67-dihe-out -67.47, -56.35 -62.32, 152.06 APE12-dist-in 9.9595 APE11-dist-out 7.059 APE10-dist-in 6.6227 APE9-dist-out 8.5077 None None None XRAY 2.243 0.191 0.236 B 315.0 286.0 0 28 28 0 [[53, 305]] 1.0 9r8c Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 2RKUA P53350 37 330 603.0 R78:500 Type1 Inactive DFGin 5.6778 15.0171 BLAminus -134.22, -169.5 54.06, 79.11 -86.67, 25.63 283.82, 88.21 -64.51, -26.07 in-in in 9.7168 Saltbr-in 3.0799 HRD-in -74.95, -48.26 75.93, -2.57 in-in-out SNCiio in-out ActLoopNT-in 2.9425 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -90.21, 90.69 APE9-dihe-na 162.46, 178.28 APE8-dihe-in -124.7, 88.6 APE8-rot-in 309.54 APE67-dihe-out -73.41, -64.04 -71.02, 160.05 APE12-dist-in 10.9294 APE11-dist-out 7.2828 APE10-dist-in 7.9206 APE9-dist-out 8.1342 T210V None None XRAY 1.95 0.192 0.241 A 294.0 294.0 0 28 28 0 [[53, 305]] 1.0 2rku Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 9R1XA P53350 39 334 603.0 R78:401 Type1 Inactive DFGin 5.4509 14.7459 BLAminus -129.34, -169.27 61.33, 81.84 -99.46, 30.78 291.65, 94.79 -60.61, -43.02 in-in in 9.6846 Saltbr-in 2.7211 HRD-in -71.39, -48.31 73.02, 3.83 in-in-out SNCiio in-out ActLoopNT-in 2.9715 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.63, 46.88 APE9-dihe-na 161.22, 163.69 APE8-dihe-in -103.28, 108.1 APE8-rot-in 301.35 APE67-dihe-out -58.97, -56.16 -54.1, 148.74 APE12-dist-in 10.3877 APE11-dist-out 6.5599 APE10-dist-in 6.7414 APE9-dist-out 8.5087 K225D,K226A None None XRAY 2.84 0.222 0.277 A 325.0 296.0 0 28 28 0 [[53, 305]] 1.0 9r1x Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK1 PLK1_HUMAN 9R1XB P53350 39 326 603.0 R78:401 Type1 Inactive DFGin 5.4448 14.7258 BLAminus -129.89, -169.09 62.76, 81.42 -99.44, 28.81 292.45, 94.66 -58.03, -43.63 in-in in 9.6661 Saltbr-in 2.714 HRD-in -71.6, -47.96 72.32, 5.61 in-in-out SNCiio in-out ActLoopNT-in 2.9664 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -82.43, 34.44 APE9-dihe-na 160.48, 165.73 APE8-dihe-in -102.91, 108.17 APE8-rot-in 301.26 APE67-dihe-out -58.46, -55.69 -54.97, 148.64 APE12-dist-in 10.4044 APE11-dist-out 6.5324 APE10-dist-in 5.999 APE9-dist-out 8.4468 K225D,K226A None None XRAY 2.84 0.222 0.277 B 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1x Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
CAMK PLK2 PLK2_HUMAN 4I5MA Q9NYY3 71 354 685.0 R78:60401 Type1 Inactive DFGin 6.1179 14.6063 BLAminus -135.0, -176.4 62.06, 78.64 -90.58, 19.32 306.45, 87.75 -51.33, -30.59 in-in in 9.2706 Saltbr-in 2.7444 HRD-in -74.53, -53.1 71.46, 0.19 in-in-out SNCiio in-out ActLoopNT-in 2.6631 ActLoopCT-out nonTYR APEdihe_aanoo APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 115.38 APE8-rot-out 169.65 APE67-dihe-out -76.41, -43.82 -77.31, 170.4 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 C83S,V87T,A119S,A216S,C259A,C291S,L335T None None XRAY 1.801 0.324 0.392 A 308.0 273.0 11 28 17 11 [[82, 334]] 1.0 4i5m Homo sapiens CAMK_PLK2_HUMAN CAMK 2.6e-82 281.9 1.0 256.0 256.0 222 223 224 226 228 111 130 134 202 204 203 205.0 262 250 245 244 243 242 241 240 239 160 Serine/threonine-protein kinase PLK2

Ligand: R78

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name