Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 8HV4A | P00533 | 696 | 1020 | 1210.0 | PE5:1101,MWU:1102 | Allosteric,Type1 | Active | DFGin | 6.099 | 15.187 | BLAminus | -130.11, -171.57 | 60.63, 76.52 | -95.44, 10.11 | 292.65, 96.39 | -43.03, -44.61 | in-in | in | 8.302 | Saltbr-in | 3.322 | HRD-in | -71.74, -51.9 | 75.14, 7.17 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.828 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -96.84, 107.0 | APE9-dihe-in | -115.33, 154.25 | APE8-dihe-in | -89.19, 79.02 | APE8-rot-na | 38.66 | APE67-dihe-in | -72.78, -5.6 | -58.65, -42.93 | APE12-dist-na | 11.758 | APE11-dist-na | 10.396 | APE10-dist-na | 11.61 | APE9-dist-in | 7.39 | E865A,E866A,K867A | None | None | XRAY | 2.2 | 0.239 | 0.275 | A | 331 | 304 | 6 | 0 | 0 | 3 | [[712, 970]] | 1.0 | 8hv4 | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV6A | P00533 | 696 | 1020 | 1210.0 | PE5:1101,N86:1102 | Allosteric,Type1 | Active | DFGin | 5.904 | 15.402 | BLAminus | -126.97, -177.08 | 64.65, 81.87 | -97.77, 4.79 | 296.74, 96.36 | -40.91, -42.24 | in-in | in | 8.752 | Saltbr-in | 2.997 | HRD-in | -69.51, -52.61 | 72.53, 9.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.775 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -100.57, 119.04 | APE9-dihe-in | -126.13, 154.51 | APE8-dihe-in | -87.49, 71.86 | APE8-rot-na | 40.33 | APE67-dihe-in | -73.01, -0.15 | -52.84, -41.89 | APE12-dist-na | 11.924 | APE11-dist-na | 10.417 | APE10-dist-na | 11.442 | APE9-dist-in | 7.354 | E865A,E866A,K867A | None | None | XRAY | 2.2 | 0.249 | 0.296 | A | 331 | 307 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv6 | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV7A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N8O:1102 | Allosteric,Type1 | Active | DFGin | 5.965 | 14.783 | BLAminus | -130.55, -167.28 | 53.08, 83.5 | -92.28, 13.92 | 300.31, 94.88 | -38.75, -43.45 | in-in | in | 8.203 | Saltbr-in | 3.059 | HRD-in | -71.82, -54.11 | 72.62, 8.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.827 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.41, 111.31 | APE9-dihe-in | -116.24, 154.93 | APE8-dihe-in | -87.4, 80.61 | APE8-rot-na | 37.2 | APE67-dihe-in | -74.07, -9.58 | -59.54, -41.0 | APE12-dist-na | 11.66 | APE11-dist-na | 10.259 | APE10-dist-na | 11.546 | APE9-dist-in | 7.176 | E865A,E866A,K867A | None | None | XRAY | 2.69 | 0.222 | 0.29 | A | 331 | 301 | 10 | 0 | 0 | 6 | [[712, 970]] | 1.0 | 8hv7 | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV8A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N99:1102 | Allosteric,Type1 | Active | DFGin | 6.043 | 15.057 | BLAminus | -125.96, -170.32 | 55.74, 82.34 | -96.51, 11.07 | 293.49, 92.75 | -34.95, -51.58 | in-in | in | 8.143 | Saltbr-in | 3.326 | HRD-in | -73.99, -49.75 | 71.98, 9.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.888 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.61, 118.18 | APE9-dihe-in | -124.65, 150.54 | APE8-dihe-in | -89.53, 80.34 | APE8-rot-na | 39.28 | APE67-dihe-in | -69.5, -3.25 | -56.62, -45.74 | APE12-dist-na | 11.675 | APE11-dist-na | 10.369 | APE10-dist-na | 11.219 | APE9-dist-in | 7.28 | C797S,E865A,E866A,K867A | None | None | XRAY | 2.4 | 0.234 | 0.283 | A | 331 | 305 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv8 | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV9A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N9L:1102 | Allosteric,Type1 | Active | DFGin | 5.916 | 15.132 | BLAminus | -143.82, -178.2 | 62.01, 78.91 | -94.0, 24.14 | 301.61, 89.09 | -64.67, -16.43 | in-in | in | 8.101 | Saltbr-in | 2.657 | HRD-in | -69.38, -54.88 | 68.74, 2.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.77 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.98, 135.96 | APE9-dihe-in | -139.68, 157.73 | APE8-dihe-in | -88.14, 76.12 | APE8-rot-na | 37.34 | APE67-dihe-in | -77.83, -6.94 | -60.36, -47.24 | APE12-dist-na | 12.179 | APE11-dist-na | 10.885 | APE10-dist-na | 11.275 | APE9-dist-in | 7.023 | E865A,E866A,K867A | None | None | XRAY | 2.5 | 0.254 | 0.274 | A | 331 | 306 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv9 | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV1A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N6N:1102 | Allosteric,Type1 | Active | DFGin | 5.813 | 15.137 | BLAminus | -141.64, -174.89 | 64.07, 81.43 | -91.77, 15.88 | 294.7, 99.28 | -49.71, -35.13 | in-in | in | 8.633 | Saltbr-in | 3.064 | HRD-in | -77.13, -49.05 | 68.6, 6.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.976 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.53, 105.98 | APE9-dihe-in | -114.36, 147.65 | APE8-dihe-in | -82.64, 80.16 | APE8-rot-na | 37.74 | APE67-dihe-in | -74.01, -6.57 | -60.27, -40.96 | APE12-dist-na | 11.899 | APE11-dist-na | 10.789 | APE10-dist-na | 11.152 | APE9-dist-in | 7.211 | E865A,E866A,K867A | None | None | XRAY | 2.4 | 0.191 | 0.219 | A | 331 | 309 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv1 | TYR_EGFR_HUMAN | TYR | 4.6e-86 | 294.4 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV3A | P00533 | 696 | 1020 | 1210.0 | PE5:1101,MWU:1103 | Allosteric,Type1 | Active | DFGin | 6.179 | 15.626 | BLAminus | -127.58, -179.0 | 62.59, 85.31 | -101.31, 9.93 | 297.08, 83.02 | -46.24, -27.8 | in-in | in | 8.645 | Saltbr-in | 3.166 | HRD-in | -72.86, -48.63 | 69.9, 8.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.918 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.05, 111.65 | APE9-dihe-in | -122.27, 146.52 | APE8-dihe-in | -88.12, 79.7 | APE8-rot-na | 39.71 | APE67-dihe-in | -75.54, -1.37 | -55.44, -43.37 | APE12-dist-na | 12.055 | APE11-dist-na | 10.393 | APE10-dist-na | 11.129 | APE9-dist-in | 7.354 | E865A,E866A,K867A | None | None | XRAY | 2.4 | 0.214 | 0.25 | A | 331 | 307 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv3 | TYR_EGFR_HUMAN | TYR | 4.6e-86 | 294.4 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV5A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N7C:1102 | Allosteric,Type1 | Active | DFGin | 5.973 | 15.251 | BLAminus | -130.95, 178.54 | 67.19, 85.27 | -98.38, 23.1 | 296.48, 89.98 | -54.53, -35.87 | in-in | in | 8.727 | Saltbr-in | 3.383 | HRD-in | -76.07, -52.83 | 75.02, 1.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.921 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.39, 115.59 | APE9-dihe-in | -118.26, 144.05 | APE8-dihe-in | -81.44, 79.55 | APE8-rot-na | 38.48 | APE67-dihe-in | -70.6, -7.98 | -54.36, -43.35 | APE12-dist-na | 11.884 | APE11-dist-na | 10.562 | APE10-dist-na | 10.953 | APE9-dist-in | 7.218 | E865A,E866A,K867A | None | None | XRAY | 2.2 | 0.188 | 0.224 | A | 331 | 306 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv5 | TYR_EGFR_HUMAN | TYR | 4.6e-86 | 294.4 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 8HV4A | P00533 | 696 | 1020 | 1210.0 | PE5:1101,MWU:1102 | Allosteric,Type1 | Active | DFGin | 6.099 | 15.187 | BLAminus | -130.11, -171.57 | 60.63, 76.52 | -95.44, 10.11 | 292.65, 96.39 | -43.03, -44.61 | in-in | in | 8.302 | Saltbr-in | 3.322 | HRD-in | -71.74, -51.9 | 75.14, 7.17 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.828 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -96.84, 107.0 | APE9-dihe-in | -115.33, 154.25 | APE8-dihe-in | -89.19, 79.02 | APE8-rot-na | 38.66 | APE67-dihe-in | -72.78, -5.6 | -58.65, -42.93 | APE12-dist-na | 11.758 | APE11-dist-na | 10.396 | APE10-dist-na | 11.61 | APE9-dist-in | 7.39 | E865A,E866A,K867A | None | None | XRAY | 2.2 | 0.239 | 0.275 | A | 331 | 304 | 6 | 0 | 0 | 3 | [[712, 970]] | 1.0 | 8hv4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV6A | P00533 | 696 | 1020 | 1210.0 | PE5:1101,N86:1102 | Allosteric,Type1 | Active | DFGin | 5.904 | 15.402 | BLAminus | -126.97, -177.08 | 64.65, 81.87 | -97.77, 4.79 | 296.74, 96.36 | -40.91, -42.24 | in-in | in | 8.752 | Saltbr-in | 2.997 | HRD-in | -69.51, -52.61 | 72.53, 9.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.775 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -100.57, 119.04 | APE9-dihe-in | -126.13, 154.51 | APE8-dihe-in | -87.49, 71.86 | APE8-rot-na | 40.33 | APE67-dihe-in | -73.01, -0.15 | -52.84, -41.89 | APE12-dist-na | 11.924 | APE11-dist-na | 10.417 | APE10-dist-na | 11.442 | APE9-dist-in | 7.354 | E865A,E866A,K867A | None | None | XRAY | 2.2 | 0.249 | 0.296 | A | 331 | 307 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv6 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV7A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N8O:1102 | Allosteric,Type1 | Active | DFGin | 5.965 | 14.783 | BLAminus | -130.55, -167.28 | 53.08, 83.5 | -92.28, 13.92 | 300.31, 94.88 | -38.75, -43.45 | in-in | in | 8.203 | Saltbr-in | 3.059 | HRD-in | -71.82, -54.11 | 72.62, 8.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.827 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.41, 111.31 | APE9-dihe-in | -116.24, 154.93 | APE8-dihe-in | -87.4, 80.61 | APE8-rot-na | 37.2 | APE67-dihe-in | -74.07, -9.58 | -59.54, -41.0 | APE12-dist-na | 11.66 | APE11-dist-na | 10.259 | APE10-dist-na | 11.546 | APE9-dist-in | 7.176 | E865A,E866A,K867A | None | None | XRAY | 2.69 | 0.222 | 0.29 | A | 331 | 301 | 10 | 0 | 0 | 6 | [[712, 970]] | 1.0 | 8hv7 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV8A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N99:1102 | Allosteric,Type1 | Active | DFGin | 6.043 | 15.057 | BLAminus | -125.96, -170.32 | 55.74, 82.34 | -96.51, 11.07 | 293.49, 92.75 | -34.95, -51.58 | in-in | in | 8.143 | Saltbr-in | 3.326 | HRD-in | -73.99, -49.75 | 71.98, 9.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.888 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.61, 118.18 | APE9-dihe-in | -124.65, 150.54 | APE8-dihe-in | -89.53, 80.34 | APE8-rot-na | 39.28 | APE67-dihe-in | -69.5, -3.25 | -56.62, -45.74 | APE12-dist-na | 11.675 | APE11-dist-na | 10.369 | APE10-dist-na | 11.219 | APE9-dist-in | 7.28 | C797S,E865A,E866A,K867A | None | None | XRAY | 2.4 | 0.234 | 0.283 | A | 331 | 305 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv8 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV9A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N9L:1102 | Allosteric,Type1 | Active | DFGin | 5.916 | 15.132 | BLAminus | -143.82, -178.2 | 62.01, 78.91 | -94.0, 24.14 | 301.61, 89.09 | -64.67, -16.43 | in-in | in | 8.101 | Saltbr-in | 2.657 | HRD-in | -69.38, -54.88 | 68.74, 2.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.77 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.98, 135.96 | APE9-dihe-in | -139.68, 157.73 | APE8-dihe-in | -88.14, 76.12 | APE8-rot-na | 37.34 | APE67-dihe-in | -77.83, -6.94 | -60.36, -47.24 | APE12-dist-na | 12.179 | APE11-dist-na | 10.885 | APE10-dist-na | 11.275 | APE9-dist-in | 7.023 | E865A,E866A,K867A | None | None | XRAY | 2.5 | 0.254 | 0.274 | A | 331 | 306 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv9 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 3.5e-86 | 294.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV1A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N6N:1102 | Allosteric,Type1 | Active | DFGin | 5.813 | 15.137 | BLAminus | -141.64, -174.89 | 64.07, 81.43 | -91.77, 15.88 | 294.7, 99.28 | -49.71, -35.13 | in-in | in | 8.633 | Saltbr-in | 3.064 | HRD-in | -77.13, -49.05 | 68.6, 6.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.976 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.53, 105.98 | APE9-dihe-in | -114.36, 147.65 | APE8-dihe-in | -82.64, 80.16 | APE8-rot-na | 37.74 | APE67-dihe-in | -74.01, -6.57 | -60.27, -40.96 | APE12-dist-na | 11.899 | APE11-dist-na | 10.789 | APE10-dist-na | 11.152 | APE9-dist-in | 7.211 | E865A,E866A,K867A | None | None | XRAY | 2.4 | 0.191 | 0.219 | A | 331 | 309 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv1 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 4.6e-86 | 294.4 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV3A | P00533 | 696 | 1020 | 1210.0 | PE5:1101,MWU:1103 | Allosteric,Type1 | Active | DFGin | 6.179 | 15.626 | BLAminus | -127.58, -179.0 | 62.59, 85.31 | -101.31, 9.93 | 297.08, 83.02 | -46.24, -27.8 | in-in | in | 8.645 | Saltbr-in | 3.166 | HRD-in | -72.86, -48.63 | 69.9, 8.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.918 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.05, 111.65 | APE9-dihe-in | -122.27, 146.52 | APE8-dihe-in | -88.12, 79.7 | APE8-rot-na | 39.71 | APE67-dihe-in | -75.54, -1.37 | -55.44, -43.37 | APE12-dist-na | 12.055 | APE11-dist-na | 10.393 | APE10-dist-na | 11.129 | APE9-dist-in | 7.354 | E865A,E866A,K867A | None | None | XRAY | 2.4 | 0.214 | 0.25 | A | 331 | 307 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv3 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 4.6e-86 | 294.4 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8HV5A | P00533 | 696 | 1019 | 1210.0 | PE5:1101,N7C:1102 | Allosteric,Type1 | Active | DFGin | 5.973 | 15.251 | BLAminus | -130.95, 178.54 | 67.19, 85.27 | -98.38, 23.1 | 296.48, 89.98 | -54.53, -35.87 | in-in | in | 8.727 | Saltbr-in | 3.383 | HRD-in | -76.07, -52.83 | 75.02, 1.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.921 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.39, 115.59 | APE9-dihe-in | -118.26, 144.05 | APE8-dihe-in | -81.44, 79.55 | APE8-rot-na | 38.48 | APE67-dihe-in | -70.6, -7.98 | -54.36, -43.35 | APE12-dist-na | 11.884 | APE11-dist-na | 10.562 | APE10-dist-na | 10.953 | APE9-dist-in | 7.218 | E865A,E866A,K867A | None | None | XRAY | 2.2 | 0.188 | 0.224 | A | 331 | 306 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8hv5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 4.6e-86 | 294.4 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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