| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | PIM1 | PIM1_HUMAN | 4GW8A | P11309 | 33 | 305 | 313.0 | 3RA:401 | Type1 | Active | DFGin | 6.2361 | 14.6142 | BLAminus | -126.36, 165.58 | 62.03, 83.71 | -89.36, 16.13 | 285.86, 76.28 | -67.97, -17.62 | in-in | in | 8.7369 | Saltbr-in | 2.7149 | HRD-naA | -74.23, -46.85 | 73.75, 9.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.85, 8.01 | APE9-dihe-na | -80.24, -160.25 | APE8-dihe-in | -87.85, 121.5 | APE8-rot-in | 304.03 | APE67-dihe-in | -71.21, -12.4 | -59.35, -38.89 | APE12-dist-in | 9.4824 | APE11-dist-in | 8.2992 | APE10-dist-in | 4.4436 | APE9-dist-in | 3.7427 | R250G | None | None | XRAY | 2.0 | 0.178 | 0.213 | A | 313.0 | 273.0 | 0 | 26 | 26 | 0 | [[38, 290]] | 1.0 | 4gw8 | CAMK_PIM1_HUMAN | CAMK | 1.5e-64 | 223.7 | 1.0 | 256.0 | 256.0 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167.0 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CMGC | CLK3 | CLK3_HUMAN | 3RAWA | P49761 | 134 | 484 | 490.0 | 3RA:1 | Type1 | Active | DFGin | 6.902 | 14.0941 | BLAminus | -124.35, 169.55 | 70.36, 85.35 | -106.01, 17.22 | 295.02, 93.37 | -60.15, -19.42 | in-in | in | 8.7233 | Saltbr-in | 2.5297 | HRD-in | -75.41, -55.66 | 80.86, -13.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8337 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.35, 172.08 | APE9-dihe-na | 79.18, 152.43 | APE8-dihe-in | -65.73, 139.23 | APE8-rot-in | 296.11 | APE67-dihe-in | -63.4, -21.96 | -51.62, -42.74 | APE12-dist-in | 13.898 | APE11-dist-in | 11.94 | APE10-dist-in | 7.4025 | APE9-dist-in | 3.0593 | None | None | None | XRAY | 2.09 | 0.182 | 0.219 | A | 381.0 | 351.0 | 0 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 3raw | CMGC_CLK3_HUMAN | CMGC | 1.5e-90 | 309.4 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 3RAWB | P49761 | 136 | 484 | 490.0 | 3RA:2 | Type1 | Inactive | DFGin | 6.9647 | 14.2368 | BLAminus | -117.05, 172.91 | 67.87, 90.75 | -108.68, 15.88 | 294.71, 94.5 | -64.13, -12.21 | in-in | in | 8.8335 | Saltbr-in | 2.6162 | HRD-in | -69.6, -50.25 | 74.29, -8.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7903 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -132.65, 172.79 | APE9-dihe-na | 79.02, 155.93 | APE8-dihe-in | -74.0, 140.2 | APE8-rot-in | 285.33 | APE67-dihe-in | -62.33, -24.2 | -48.19, -48.04 | APE12-dist-out | 14.1155 | APE11-dist-in | 11.9091 | APE10-dist-in | 7.4878 | APE9-dist-in | 3.0018 | None | None | None | XRAY | 2.09 | 0.182 | 0.219 | B | 381.0 | 349.0 | 0 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 3raw | CMGC_CLK3_HUMAN | CMGC | 1.5e-90 | 309.4 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | DYRK1A | DYR1A_HUMAN | 4AZEA | Q13627 | 132 | 481 | 763.0 | 3RA:700 | Type1 | Active | DFGin | 6.9533 | 14.6162 | BLAminus | -137.23, 169.92 | 67.49, 90.44 | -106.39, 23.89 | 283.3, 71.95 | -55.61, -37.62 | in-in | in | 9.0098 | Saltbr-in | 2.8124 | HRD-in | -70.04, -49.18 | 72.92, 15.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8739 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.19, 169.65 | APE9-dihe-na | 74.45, 134.72 | APE8-dihe-in | -60.37, 136.79 | APE8-rot-in | 289.06 | APE67-dihe-in | -57.82, -32.3 | -48.27, -49.81 | APE12-dist-in | 12.2654 | APE11-dist-in | 10.5618 | APE10-dist-in | 6.6352 | APE9-dist-in | 3.2564 | None | SEP301,PTR321 | SEP301,PTR321 | XRAY | 3.15 | 0.219 | 0.248 | A | 382.0 | 350.0 | 0 | 25 | 25 | 0 | [[159, 479]] | 1.0 | 4aze | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1.0 | 301.0 | 301.0 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287.0 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 4AZEB | Q13627 | 135 | 481 | 763.0 | 3RA:700 | Type1 | Active | DFGin | 6.9238 | 14.6128 | BLAminus | -138.16, 169.5 | 68.4, 90.42 | -106.1, 24.2 | 283.49, 72.02 | -57.21, -35.99 | in-in | in | 9.0221 | Saltbr-in | 2.9003 | HRD-in | -69.57, -48.1 | 73.99, 12.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8331 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.81, 169.0 | APE9-dihe-na | 74.6, 134.75 | APE8-dihe-in | -60.95, 138.61 | APE8-rot-in | 290.43 | APE67-dihe-in | -56.44, -36.37 | -49.68, -48.78 | APE12-dist-in | 12.2764 | APE11-dist-in | 10.5588 | APE10-dist-in | 6.6312 | APE9-dist-in | 3.2256 | None | SEP301,PTR321 | SEP301,PTR321 | XRAY | 3.15 | 0.219 | 0.248 | B | 382.0 | 347.0 | 0 | 25 | 25 | 0 | [[159, 479]] | 1.0 | 4aze | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1.0 | 301.0 | 301.0 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287.0 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 4AZEC | Q13627 | 132 | 481 | 763.0 | 3RA:700 | Type1 | Active | DFGin | 6.9331 | 14.6073 | BLAminus | -136.67, 171.08 | 67.02, 92.32 | -107.7, 25.06 | 283.25, 71.9 | -57.45, -37.58 | in-in | in | 9.0017 | Saltbr-in | 2.8354 | HRD-in | -68.51, -50.21 | 73.5, 15.7 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8424 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.49, 169.71 | APE9-dihe-na | 73.57, 134.86 | APE8-dihe-in | -60.52, 139.24 | APE8-rot-in | 289.26 | APE67-dihe-in | -57.24, -34.82 | -50.4, -48.08 | APE12-dist-in | 12.3165 | APE11-dist-in | 10.5695 | APE10-dist-in | 6.591 | APE9-dist-in | 3.2797 | None | SEP301,PTR321 | SEP301,PTR321 | XRAY | 3.15 | 0.219 | 0.248 | C | 382.0 | 350.0 | 0 | 25 | 25 | 0 | [[159, 479]] | 1.0 | 4aze | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1.0 | 301.0 | 301.0 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287.0 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK2 | DYRK2_HUMAN | 4AZFA | Q92630 | 146 | 536 | 601.0 | 3RA:60600 | Type1 | Inactive | DFGin | 6.9946 | 15.3904 | BLAminus | -118.77, 179.61 | 61.33, 77.52 | -93.54, 30.44 | 283.47, 77.53 | -76.64, -12.42 | in-in | in | 9.0817 | Saltbr-in | 2.7335 | HRD-in | -73.11, -47.79 | 80.4, -7.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9212 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -141.82, 174.61 | APE9-dihe-na | 70.03, 158.03 | APE8-dihe-in | -81.89, 134.84 | APE8-rot-out | 174.41 | APE67-dihe-in | -64.03, -20.73 | -38.64, -55.03 | APE12-dist-in | 10.2473 | APE11-dist-in | 11.6168 | APE10-dist-in | 7.1161 | APE9-dist-in | 3.2122 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.55 | 0.2 | 0.255 | A | 417.0 | 389.0 | 2 | 25 | 25 | 0 | [[222, 535]] | 1.0 | 4azf | CMGC_DYRK2_HUMAN | CMGC | 1.3e-98 | 336.0 | 1.0 | 301.0 | 301.0 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348.0 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | PIM1 | PIM1_HUMAN | 4GW8A | P11309 | 33 | 305 | 313.0 | 3RA:401 | Type1 | Active | DFGin | 6.2361 | 14.6142 | BLAminus | -126.36, 165.58 | 62.03, 83.71 | -89.36, 16.13 | 285.86, 76.28 | -67.97, -17.62 | in-in | in | 8.7369 | Saltbr-in | 2.7149 | HRD-naA | -74.23, -46.85 | 73.75, 9.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.85, 8.01 | APE9-dihe-na | -80.24, -160.25 | APE8-dihe-in | -87.85, 121.5 | APE8-rot-in | 304.03 | APE67-dihe-in | -71.21, -12.4 | -59.35, -38.89 | APE12-dist-in | 9.4824 | APE11-dist-in | 8.2992 | APE10-dist-in | 4.4436 | APE9-dist-in | 3.7427 | R250G | None | None | XRAY | 2.0 | 0.178 | 0.213 | A | 313.0 | 273.0 | 0 | 26 | 26 | 0 | [[38, 290]] | 1.0 | 4gw8 | Homo sapiens | CAMK_PIM1_HUMAN | CAMK | 1.5e-64 | 223.7 | 1.0 | 256.0 | 256.0 | 185 | 186 | 187 | 189 | 191 | 67 | 89 | 93 | 164 | 166 | 165 | 167.0 | 224 | 211 | 206 | 205 | 204 | 203 | 202 | 201 | 200 | 121 | Serine/threonine-protein kinase pim-1 |
| CMGC | CLK3 | CLK3_HUMAN | 3RAWA | P49761 | 134 | 484 | 490.0 | 3RA:1 | Type1 | Active | DFGin | 6.902 | 14.0941 | BLAminus | -124.35, 169.55 | 70.36, 85.35 | -106.01, 17.22 | 295.02, 93.37 | -60.15, -19.42 | in-in | in | 8.7233 | Saltbr-in | 2.5297 | HRD-in | -75.41, -55.66 | 80.86, -13.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8337 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.35, 172.08 | APE9-dihe-na | 79.18, 152.43 | APE8-dihe-in | -65.73, 139.23 | APE8-rot-in | 296.11 | APE67-dihe-in | -63.4, -21.96 | -51.62, -42.74 | APE12-dist-in | 13.898 | APE11-dist-in | 11.94 | APE10-dist-in | 7.4025 | APE9-dist-in | 3.0593 | None | None | None | XRAY | 2.09 | 0.182 | 0.219 | A | 381.0 | 351.0 | 0 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 3raw | Homo sapiens | CMGC_CLK3_HUMAN | CMGC | 1.5e-90 | 309.4 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 3RAWB | P49761 | 136 | 484 | 490.0 | 3RA:2 | Type1 | Inactive | DFGin | 6.9647 | 14.2368 | BLAminus | -117.05, 172.91 | 67.87, 90.75 | -108.68, 15.88 | 294.71, 94.5 | -64.13, -12.21 | in-in | in | 8.8335 | Saltbr-in | 2.6162 | HRD-in | -69.6, -50.25 | 74.29, -8.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7903 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -132.65, 172.79 | APE9-dihe-na | 79.02, 155.93 | APE8-dihe-in | -74.0, 140.2 | APE8-rot-in | 285.33 | APE67-dihe-in | -62.33, -24.2 | -48.19, -48.04 | APE12-dist-out | 14.1155 | APE11-dist-in | 11.9091 | APE10-dist-in | 7.4878 | APE9-dist-in | 3.0018 | None | None | None | XRAY | 2.09 | 0.182 | 0.219 | B | 381.0 | 349.0 | 0 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 3raw | Homo sapiens | CMGC_CLK3_HUMAN | CMGC | 1.5e-90 | 309.4 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | DYRK1A | DYR1A_HUMAN | 4AZEA | Q13627 | 132 | 481 | 763.0 | 3RA:700 | Type1 | Active | DFGin | 6.9533 | 14.6162 | BLAminus | -137.23, 169.92 | 67.49, 90.44 | -106.39, 23.89 | 283.3, 71.95 | -55.61, -37.62 | in-in | in | 9.0098 | Saltbr-in | 2.8124 | HRD-in | -70.04, -49.18 | 72.92, 15.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8739 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.19, 169.65 | APE9-dihe-na | 74.45, 134.72 | APE8-dihe-in | -60.37, 136.79 | APE8-rot-in | 289.06 | APE67-dihe-in | -57.82, -32.3 | -48.27, -49.81 | APE12-dist-in | 12.2654 | APE11-dist-in | 10.5618 | APE10-dist-in | 6.6352 | APE9-dist-in | 3.2564 | None | SEP301,PTR321 | SEP301,PTR321 | XRAY | 3.15 | 0.219 | 0.248 | A | 382.0 | 350.0 | 0 | 25 | 25 | 0 | [[159, 479]] | 1.0 | 4aze | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1.0 | 301.0 | 301.0 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287.0 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 4AZEB | Q13627 | 135 | 481 | 763.0 | 3RA:700 | Type1 | Active | DFGin | 6.9238 | 14.6128 | BLAminus | -138.16, 169.5 | 68.4, 90.42 | -106.1, 24.2 | 283.49, 72.02 | -57.21, -35.99 | in-in | in | 9.0221 | Saltbr-in | 2.9003 | HRD-in | -69.57, -48.1 | 73.99, 12.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8331 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.81, 169.0 | APE9-dihe-na | 74.6, 134.75 | APE8-dihe-in | -60.95, 138.61 | APE8-rot-in | 290.43 | APE67-dihe-in | -56.44, -36.37 | -49.68, -48.78 | APE12-dist-in | 12.2764 | APE11-dist-in | 10.5588 | APE10-dist-in | 6.6312 | APE9-dist-in | 3.2256 | None | SEP301,PTR321 | SEP301,PTR321 | XRAY | 3.15 | 0.219 | 0.248 | B | 382.0 | 347.0 | 0 | 25 | 25 | 0 | [[159, 479]] | 1.0 | 4aze | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1.0 | 301.0 | 301.0 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287.0 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 4AZEC | Q13627 | 132 | 481 | 763.0 | 3RA:700 | Type1 | Active | DFGin | 6.9331 | 14.6073 | BLAminus | -136.67, 171.08 | 67.02, 92.32 | -107.7, 25.06 | 283.25, 71.9 | -57.45, -37.58 | in-in | in | 9.0017 | Saltbr-in | 2.8354 | HRD-in | -68.51, -50.21 | 73.5, 15.7 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8424 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.49, 169.71 | APE9-dihe-na | 73.57, 134.86 | APE8-dihe-in | -60.52, 139.24 | APE8-rot-in | 289.26 | APE67-dihe-in | -57.24, -34.82 | -50.4, -48.08 | APE12-dist-in | 12.3165 | APE11-dist-in | 10.5695 | APE10-dist-in | 6.591 | APE9-dist-in | 3.2797 | None | SEP301,PTR321 | SEP301,PTR321 | XRAY | 3.15 | 0.219 | 0.248 | C | 382.0 | 350.0 | 0 | 25 | 25 | 0 | [[159, 479]] | 1.0 | 4aze | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1.0 | 301.0 | 301.0 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287.0 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK2 | DYRK2_HUMAN | 4AZFA | Q92630 | 146 | 536 | 601.0 | 3RA:60600 | Type1 | Inactive | DFGin | 6.9946 | 15.3904 | BLAminus | -118.77, 179.61 | 61.33, 77.52 | -93.54, 30.44 | 283.47, 77.53 | -76.64, -12.42 | in-in | in | 9.0817 | Saltbr-in | 2.7335 | HRD-in | -73.11, -47.79 | 80.4, -7.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9212 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -141.82, 174.61 | APE9-dihe-na | 70.03, 158.03 | APE8-dihe-in | -81.89, 134.84 | APE8-rot-out | 174.41 | APE67-dihe-in | -64.03, -20.73 | -38.64, -55.03 | APE12-dist-in | 10.2473 | APE11-dist-in | 11.6168 | APE10-dist-in | 7.1161 | APE9-dist-in | 3.2122 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.55 | 0.2 | 0.255 | A | 417.0 | 389.0 | 2 | 25 | 25 | 0 | [[222, 535]] | 1.0 | 4azf | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.3e-98 | 336.0 | 1.0 | 301.0 | 301.0 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348.0 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|