CAMK_PIM2 (Serine/threonine-protein kinase pim-2)

Total number of chains: 6
Active chains: 3
Family: CAMK
Uniprot: PIM2_HUMAN
Kinase Domain Residues: 32 - 286
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 100.0% AF-Q9P1W9-K1A

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AF-Q9P1W9-K1A 24 294 311.0 No_ligand No_ligand Active DFGin 5.981 14.335 BLAminus -126.89, 169.76 59.25, 80.5 -87.64, 18.92 284.7, 69.92 -59.97, -36.8 in-in in 8.421 Saltbr-in 2.679 HRD-na-T -75.17, -41.63 62.22, -7.7 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -115.37, 22.21 APE9-dihe-na -84.18, -176.74 APE8-dihe-in -73.66, 121.18 APE8-rot-in 303.62 APE67-dihe-in -69.59, -15.65 -57.15, -41.47 APE12-dist-in 9.455 APE11-dist-in 8.725 APE10-dist-in 5.139 APE9-dist-in 3.821 None None None AF2 -1.0 1.0 1.0 A 271 271 0 0 0 0 [[32, 286]] 1.0 AF-Q9P1W9-K1 CAMK_PIM2_HUMAN CAMK 3.3e-61 212.8 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
AF-Q9P1W9-K3A 24 294 311.0 No_ligand No_ligand Active DFGin 5.792 13.983 BLAminus -128.64, 173.97 56.27, 78.2 -80.94, 17.18 284.85, 73.49 -59.99, -38.55 in-in in 8.261 Saltbr-in 2.667 HRD-na-T -77.09, -36.87 63.05, -18.0 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -100.04, 8.53 APE9-dihe-na -84.81, 179.89 APE8-dihe-in -75.15, 129.13 APE8-rot-in 296.96 APE67-dihe-in -68.39, -18.9 -58.68, -43.28 APE12-dist-in 9.824 APE11-dist-in 9.247 APE10-dist-in 4.122 APE9-dist-in 3.674 None None None AF2 -1.0 1.0 1.0 A 271 271 0 0 0 0 [[32, 286]] 1.0 AF-Q9P1W9-K3 CAMK_PIM2_HUMAN CAMK 3.3e-61 212.8 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
4X7QB 27 287 311.0 3YR:401 Type1 Active DFGin 6.127 14.1 BLAminus -129.33, 168.29 68.57, 75.13 -88.36, 11.07 283.21, 81.76 -55.7, -17.38 in-in in 8.187 Saltbr-in 2.586 HRD-na-T -70.88, -48.99 70.44, 7.88 in-in-in SNCiii in-in ActLoopNT-in 2.905 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.21, 66.32 APE9-dihe-na -89.41, -159.06 APE8-dihe-in -91.58, 123.37 APE8-rot-in 302.93 APE67-dihe-in -67.71, -12.45 -52.33, -48.23 APE12-dist-in 8.785 APE11-dist-in 8.505 APE10-dist-in 6.402 APE9-dist-in 4.236 None None None XRAY 2.33 0.199 0.258 B 312 243 18 0 0 0 [[32, 286]] 1.0 4x7q CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
2IWIA 32 288 311.0 HB1:1289 Type1 None DFGin 6.219 14.218 BLAminus -110.81, 164.83 68.74, 90.42 -99.66, 29.13 287.09, 66.88 -61.46, -39.74 in-none in 8.56 Saltbr-none 999.0 HRD-na-T -76.62, -35.93 58.51, 10.21 none-in-in SNCnii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.36, -16.65 APE9-dihe-na -63.74, 173.12 APE8-dihe-in -77.0, 156.24 APE8-rot-in 263.75 APE67-dihe-in -52.18, -29.37 -50.11, -60.45 APE12-dist-in 9.015 APE11-dist-in 9.245 APE10-dist-in 4.898 APE9-dist-in 5.68 None None None XRAY 2.8 0.244 0.289 A 312 244 13 0 0 0 [[32, 286]] 1.0 2iwi CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
2IWIB 22 287 311.0 HB1:1288 Type1 None DFGin 6.13 13.843 BLAminus -118.57, 161.53 68.46, 93.4 -100.16, 25.47 292.3, 69.44 -61.98, -35.07 in-none in 8.602 Saltbr-none 999.0 HRD-na-T -73.52, -38.58 59.85, 10.52 none-in-in SNCnii in-in ActLoopNT-in 2.82 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.66, -16.48 APE9-dihe-na -63.71, 174.13 APE8-dihe-in -79.54, 156.69 APE8-rot-in 292.9 APE67-dihe-in -51.11, -31.79 -54.32, -53.14 APE12-dist-in 8.851 APE11-dist-in 9.327 APE10-dist-in 4.895 APE9-dist-in 5.671 None None None XRAY 2.8 0.244 0.289 B 312 249 17 0 0 0 [[32, 286]] 1.0 2iwi CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
4X7QA 32 287 311.0 3YR:401 Type1 None DFGin 6.467 14.664 BLAminus -126.1, 165.99 65.04, 79.85 -95.42, 6.54 281.8, 81.22 -72.84, 17.13 in-in in 8.3 Saltbr-in 2.568 HRD-na-T -75.97, -46.2 69.29, -4.22 in-in-none SNCiin in-none ActLoopNT-in 3.014 ActLoopCT-none nonTYR APEdihe_aaiii APEdist_nnii APE10-dihe-na 999.0, 21.71 APE9-dihe-na -87.64, 176.68 APE8-dihe-in -77.74, 129.43 APE8-rot-in 298.56 APE67-dihe-in -70.69, -7.37 -67.84, -36.53 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 6.25 APE9-dist-in 4.16 None None None XRAY 2.33 0.199 0.258 A 312 217 39 0 0 10 [[32, 286]] 1.0 4x7q CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2

CAMK_PIM2 (Serine/threonine-protein kinase pim-2)

Total number of chains: 6
Active chains: 3
Family: CAMK
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 100.0% AF-Q9P1W9-K1A

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PIM2_HUMAN AF-Q9P1W9-K1A Q9P1W9 24 294 311.0 No_ligand No_ligand Active DFGin 5.981 14.335 BLAminus -126.89, 169.76 59.25, 80.5 -87.64, 18.92 284.7, 69.92 -59.97, -36.8 in-in in 8.421 Saltbr-in 2.679 HRD-na-T -75.17, -41.63 62.22, -7.7 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -115.37, 22.21 APE9-dihe-na -84.18, -176.74 APE8-dihe-in -73.66, 121.18 APE8-rot-in 303.62 APE67-dihe-in -69.59, -15.65 -57.15, -41.47 APE12-dist-in 9.455 APE11-dist-in 8.725 APE10-dist-in 5.139 APE9-dist-in 3.821 None None None AF2 -1.0 1.0 1.0 A 271 271 0 0 0 0 [[32, 286]] 1.0 AF-Q9P1W9-K1 Homo sapiens CAMK_PIM2_HUMAN CAMK 3.3e-61 212.8 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
PIM2_HUMAN AF-Q9P1W9-K3A Q9P1W9 24 294 311.0 No_ligand No_ligand Active DFGin 5.792 13.983 BLAminus -128.64, 173.97 56.27, 78.2 -80.94, 17.18 284.85, 73.49 -59.99, -38.55 in-in in 8.261 Saltbr-in 2.667 HRD-na-T -77.09, -36.87 63.05, -18.0 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -100.04, 8.53 APE9-dihe-na -84.81, 179.89 APE8-dihe-in -75.15, 129.13 APE8-rot-in 296.96 APE67-dihe-in -68.39, -18.9 -58.68, -43.28 APE12-dist-in 9.824 APE11-dist-in 9.247 APE10-dist-in 4.122 APE9-dist-in 3.674 None None None AF2 -1.0 1.0 1.0 A 271 271 0 0 0 0 [[32, 286]] 1.0 AF-Q9P1W9-K3 Homo sapiens CAMK_PIM2_HUMAN CAMK 3.3e-61 212.8 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
PIM2_HUMAN 4X7QB Q9P1W9 27 287 311.0 3YR:401 Type1 Active DFGin 6.127 14.1 BLAminus -129.33, 168.29 68.57, 75.13 -88.36, 11.07 283.21, 81.76 -55.7, -17.38 in-in in 8.187 Saltbr-in 2.586 HRD-na-T -70.88, -48.99 70.44, 7.88 in-in-in SNCiii in-in ActLoopNT-in 2.905 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.21, 66.32 APE9-dihe-na -89.41, -159.06 APE8-dihe-in -91.58, 123.37 APE8-rot-in 302.93 APE67-dihe-in -67.71, -12.45 -52.33, -48.23 APE12-dist-in 8.785 APE11-dist-in 8.505 APE10-dist-in 6.402 APE9-dist-in 4.236 None None None XRAY 2.33 0.199 0.258 B 312 243 18 0 0 0 [[32, 286]] 1.0 4x7q Homo sapiens CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
PIM2_HUMAN 2IWIA Q9P1W9 32 288 311.0 HB1:1289 Type1 None DFGin 6.219 14.218 BLAminus -110.81, 164.83 68.74, 90.42 -99.66, 29.13 287.09, 66.88 -61.46, -39.74 in-none in 8.56 Saltbr-none 999.0 HRD-na-T -76.62, -35.93 58.51, 10.21 none-in-in SNCnii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.36, -16.65 APE9-dihe-na -63.74, 173.12 APE8-dihe-in -77.0, 156.24 APE8-rot-in 263.75 APE67-dihe-in -52.18, -29.37 -50.11, -60.45 APE12-dist-in 9.015 APE11-dist-in 9.245 APE10-dist-in 4.898 APE9-dist-in 5.68 None None None XRAY 2.8 0.244 0.289 A 312 244 13 0 0 0 [[32, 286]] 1.0 2iwi Homo sapiens CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
PIM2_HUMAN 2IWIB Q9P1W9 22 287 311.0 HB1:1288 Type1 None DFGin 6.13 13.843 BLAminus -118.57, 161.53 68.46, 93.4 -100.16, 25.47 292.3, 69.44 -61.98, -35.07 in-none in 8.602 Saltbr-none 999.0 HRD-na-T -73.52, -38.58 59.85, 10.52 none-in-in SNCnii in-in ActLoopNT-in 2.82 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.66, -16.48 APE9-dihe-na -63.71, 174.13 APE8-dihe-in -79.54, 156.69 APE8-rot-in 292.9 APE67-dihe-in -51.11, -31.79 -54.32, -53.14 APE12-dist-in 8.851 APE11-dist-in 9.327 APE10-dist-in 4.895 APE9-dist-in 5.671 None None None XRAY 2.8 0.244 0.289 B 312 249 17 0 0 0 [[32, 286]] 1.0 2iwi Homo sapiens CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2
PIM2_HUMAN 4X7QA Q9P1W9 32 287 311.0 3YR:401 Type1 None DFGin 6.467 14.664 BLAminus -126.1, 165.99 65.04, 79.85 -95.42, 6.54 281.8, 81.22 -72.84, 17.13 in-in in 8.3 Saltbr-in 2.568 HRD-na-T -75.97, -46.2 69.29, -4.22 in-in-none SNCiin in-none ActLoopNT-in 3.014 ActLoopCT-none nonTYR APEdihe_aaiii APEdist_nnii APE10-dihe-na 999.0, 21.71 APE9-dihe-na -87.64, 176.68 APE8-dihe-in -77.74, 129.43 APE8-rot-in 298.56 APE67-dihe-in -70.69, -7.37 -67.84, -36.53 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 6.25 APE9-dist-in 4.16 None None None XRAY 2.33 0.199 0.258 A 312 217 39 0 0 10 [[32, 286]] 1.0 4x7q Homo sapiens CAMK_PIM2_HUMAN CAMK 5.5e-61 212.0 1 256 256 181 182 183 185 187 61 83 87 160 162 161 163 220 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase pim-2

CAMK_PIM2 (Serine/threonine-protein kinase pim-2)

Total number of chains: 0
Active chains: 0
Family: CAMK
Spatial label Dihedral label Number of Chains Percent Representative

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name