| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| MAPK3 | AF-P27361-K1A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5927 | 14.8959 | BLAminus | -130.53, -179.67 | 55.56, 73.68 | -81.57, 15.4 | 283.43, 73.42 | -60.15, -27.17 | in-in | in | 9.0976 | Saltbr-in | 2.6988 | HRD-in | -71.43, -46.13 | 64.54, 6.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8631 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -74.91, 170.97 | APE9-dihe-na | 59.86, 147.58 | APE8-dihe-in | -63.62, 134.74 | APE8-rot-in | 298.27 | APE67-dihe-in | -68.94, -17.88 | -46.37, -48.07 | APE12-dist-in | 12.835 | APE11-dist-in | 11.3255 | APE10-dist-in | 6.8179 | APE9-dist-in | 3.0367 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K1 | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | AF-P27361-K3A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5353 | 14.6344 | BLAminus | -133.14, -176.56 | 56.67, 65.23 | -76.5, 14.43 | 283.46, 73.65 | -63.2, -17.33 | in-in | in | 9.0366 | Saltbr-in | 2.6885 | HRD-in | -77.08, -46.07 | 62.9, 16.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8517 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -69.1, 168.93 | APE9-dihe-na | 59.76, 143.47 | APE8-dihe-in | -62.52, 135.83 | APE8-rot-in | 298.7 | APE67-dihe-in | -69.69, -17.66 | -48.0, -47.1 | APE12-dist-in | 12.4845 | APE11-dist-in | 11.0788 | APE10-dist-in | 6.6158 | APE9-dist-in | 3.0598 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K3 | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | 6GESB | P27361 | 25 | 374 | 379.0 | 6H3:401 | Type1 | Inactive | DFGin | 6.894 | 15.4972 | BLAminus | -138.79, 174.04 | 68.33, 84.06 | -104.81, 19.96 | 280.63, 68.61 | -61.52, -24.52 | in-in | in | 9.3661 | Saltbr-in | 2.9312 | HRD-in | -74.27, -56.06 | 78.37, 3.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7841 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -97.48, -39.89 | APE9-dihe-na | -63.16, 160.66 | APE8-dihe-in | -55.88, 126.17 | APE8-rot-in | 317.05 | APE67-dihe-in | -63.74, -19.63 | -50.02, -51.48 | APE12-dist-out | 14.3289 | APE11-dist-in | 10.9522 | APE10-dist-in | 6.917 | APE9-dist-in | 4.4242 | None | None | None | XRAY | 2.07 | 0.172 | 0.213 | B | 380.0 | 350.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 6ges | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | 2ZOQA | P27361 | 24 | 375 | 379.0 | 5ID:382 | Type1 | Inactive | DFGin | 6.8223 | 14.8763 | BLAminus | -110.57, 174.03 | 16.61, 106.79 | -100.79, 23.94 | 292.4, 62.55 | -56.98, -29.52 | in-in | in | 9.2231 | Saltbr-in | 2.8581 | HRD-in | -74.22, -49.1 | 69.67, -4.29 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7148 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -88.46, -39.85 | APE9-dihe-na | -45.11, 153.81 | APE8-dihe-in | -55.88, 121.07 | APE8-rot-in | 311.89 | APE67-dihe-in | -58.47, -14.87 | -49.12, -49.9 | APE12-dist-out | 14.3791 | APE11-dist-in | 9.7967 | APE10-dist-in | 6.8647 | APE9-dist-in | 4.6144 | None | PTR204 | PTR204 | XRAY | 2.39 | 0.249 | 0.267 | A | 382.0 | 352.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 2zoq | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | 2ZOQB | P27361 | 24 | 375 | 379.0 | 5ID:382 | Type1 | Inactive | DFGin | 7.0812 | 14.6957 | BLAminus | -126.97, -169.7 | 58.49, 71.36 | -96.75, 32.61 | 283.64, 67.73 | -68.29, -24.37 | in-out | in | 9.6478 | Saltbr-out | 3.7469 | HRD-in | -67.75, -54.76 | 76.39, 2.97 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.7866 | ActLoopCT-out | nonTYR | APEdihe_aaoio | APEdist_iiii | APE10-dihe-na | -62.22, -135.12 | APE9-dihe-na | -49.82, -170.24 | APE8-dihe-out | -38.65, -56.7 | APE8-rot-in | 299.06 | APE67-dihe-out | -72.56, -16.77 | 136.84, -44.19 | APE12-dist-in | 13.6669 | APE11-dist-in | 11.4134 | APE10-dist-in | 7.869 | APE9-dist-in | 4.0763 | None | PTR204 | PTR204 | XRAY | 2.39 | 0.249 | 0.267 | B | 382.0 | 352.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 2zoq | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | 6GESA | P27361 | 25 | 374 | 379.0 | 6H3:401,EWH:402 | Type1,Allosteric | Inactive | DFGin | 6.9525 | 15.557 | BLAminus | -139.32, 176.86 | 65.58, 87.64 | -106.07, 21.81 | 281.49, 72.32 | -67.67, -20.97 | in-in | in | 9.4645 | Saltbr-in | 2.8664 | HRD-in | -74.62, -54.83 | 79.01, 3.71 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7498 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -96.37, -37.93 | APE9-dihe-na | -66.29, 158.31 | APE8-dihe-in | -54.71, 127.96 | APE8-rot-in | 319.22 | APE67-dihe-in | -62.74, -20.38 | -53.12, -50.26 | APE12-dist-out | 14.2267 | APE11-dist-in | 11.0263 | APE10-dist-in | 6.9344 | APE9-dist-in | 4.4094 | None | None | None | XRAY | 2.07 | 0.172 | 0.213 | A | 380.0 | 350.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 6ges | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | 4QTBA | P27361 | 24 | 374 | 379.0 | 38Z:418 | Type1.5_Front | Inactive | DFGin | 6.9632 | 16.1915 | BLAminus | -128.63, 172.06 | 72.12, 87.31 | -104.64, 23.58 | 286.23, 74.76 | -64.07, -28.14 | in-in | in | 9.6383 | Saltbr-in | 2.6538 | HRD-in | -72.11, -54.76 | 73.09, 8.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7675 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -93.95, -29.12 | APE9-dihe-na | -67.78, 160.1 | APE8-dihe-in | -53.91, 125.98 | APE8-rot-in | 310.28 | APE67-dihe-in | -65.26, -17.27 | -52.54, -50.1 | APE12-dist-out | 14.1554 | APE11-dist-in | 10.8041 | APE10-dist-in | 6.8428 | APE9-dist-in | 4.4119 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | A | 380.0 | 351.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | 4QTBB | P27361 | 27 | 374 | 379.0 | 38Z:412 | Type1.5_Front | Inactive | DFGin | 6.9886 | 16.0949 | BLAminus | -131.38, 169.9 | 76.01, 86.99 | -105.18, 21.27 | 288.36, 77.86 | -59.51, -32.2 | in-in | in | 9.5939 | Saltbr-in | 2.7088 | HRD-in | -72.51, -53.5 | 77.51, 5.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8241 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -90.9, -27.9 | APE9-dihe-na | -67.55, 157.04 | APE8-dihe-in | -54.84, 126.95 | APE8-rot-in | 308.82 | APE67-dihe-in | -67.72, -16.58 | -53.94, -47.75 | APE12-dist-out | 14.1875 | APE11-dist-in | 10.8583 | APE10-dist-in | 7.0815 | APE9-dist-in | 4.4109 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | B | 380.0 | 348.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| MAPK3 | MK03_HUMAN | AF-P27361-K1A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5927 | 14.8959 | BLAminus | -130.53, -179.67 | 55.56, 73.68 | -81.57, 15.4 | 283.43, 73.42 | -60.15, -27.17 | in-in | in | 9.0976 | Saltbr-in | 2.6988 | HRD-in | -71.43, -46.13 | 64.54, 6.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8631 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -74.91, 170.97 | APE9-dihe-na | 59.86, 147.58 | APE8-dihe-in | -63.62, 134.74 | APE8-rot-in | 298.27 | APE67-dihe-in | -68.94, -17.88 | -46.37, -48.07 | APE12-dist-in | 12.835 | APE11-dist-in | 11.3255 | APE10-dist-in | 6.8179 | APE9-dist-in | 3.0367 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K1 | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | AF-P27361-K3A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5353 | 14.6344 | BLAminus | -133.14, -176.56 | 56.67, 65.23 | -76.5, 14.43 | 283.46, 73.65 | -63.2, -17.33 | in-in | in | 9.0366 | Saltbr-in | 2.6885 | HRD-in | -77.08, -46.07 | 62.9, 16.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8517 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -69.1, 168.93 | APE9-dihe-na | 59.76, 143.47 | APE8-dihe-in | -62.52, 135.83 | APE8-rot-in | 298.7 | APE67-dihe-in | -69.69, -17.66 | -48.0, -47.1 | APE12-dist-in | 12.4845 | APE11-dist-in | 11.0788 | APE10-dist-in | 6.6158 | APE9-dist-in | 3.0598 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K3 | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | 6GESB | P27361 | 25 | 374 | 379.0 | 6H3:401 | Type1 | Inactive | DFGin | 6.894 | 15.4972 | BLAminus | -138.79, 174.04 | 68.33, 84.06 | -104.81, 19.96 | 280.63, 68.61 | -61.52, -24.52 | in-in | in | 9.3661 | Saltbr-in | 2.9312 | HRD-in | -74.27, -56.06 | 78.37, 3.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7841 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -97.48, -39.89 | APE9-dihe-na | -63.16, 160.66 | APE8-dihe-in | -55.88, 126.17 | APE8-rot-in | 317.05 | APE67-dihe-in | -63.74, -19.63 | -50.02, -51.48 | APE12-dist-out | 14.3289 | APE11-dist-in | 10.9522 | APE10-dist-in | 6.917 | APE9-dist-in | 4.4242 | None | None | None | XRAY | 2.07 | 0.172 | 0.213 | B | 380.0 | 350.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 6ges | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | 2ZOQA | P27361 | 24 | 375 | 379.0 | 5ID:382 | Type1 | Inactive | DFGin | 6.8223 | 14.8763 | BLAminus | -110.57, 174.03 | 16.61, 106.79 | -100.79, 23.94 | 292.4, 62.55 | -56.98, -29.52 | in-in | in | 9.2231 | Saltbr-in | 2.8581 | HRD-in | -74.22, -49.1 | 69.67, -4.29 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7148 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -88.46, -39.85 | APE9-dihe-na | -45.11, 153.81 | APE8-dihe-in | -55.88, 121.07 | APE8-rot-in | 311.89 | APE67-dihe-in | -58.47, -14.87 | -49.12, -49.9 | APE12-dist-out | 14.3791 | APE11-dist-in | 9.7967 | APE10-dist-in | 6.8647 | APE9-dist-in | 4.6144 | None | PTR204 | PTR204 | XRAY | 2.39 | 0.249 | 0.267 | A | 382.0 | 352.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 2zoq | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | 2ZOQB | P27361 | 24 | 375 | 379.0 | 5ID:382 | Type1 | Inactive | DFGin | 7.0812 | 14.6957 | BLAminus | -126.97, -169.7 | 58.49, 71.36 | -96.75, 32.61 | 283.64, 67.73 | -68.29, -24.37 | in-out | in | 9.6478 | Saltbr-out | 3.7469 | HRD-in | -67.75, -54.76 | 76.39, 2.97 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.7866 | ActLoopCT-out | nonTYR | APEdihe_aaoio | APEdist_iiii | APE10-dihe-na | -62.22, -135.12 | APE9-dihe-na | -49.82, -170.24 | APE8-dihe-out | -38.65, -56.7 | APE8-rot-in | 299.06 | APE67-dihe-out | -72.56, -16.77 | 136.84, -44.19 | APE12-dist-in | 13.6669 | APE11-dist-in | 11.4134 | APE10-dist-in | 7.869 | APE9-dist-in | 4.0763 | None | PTR204 | PTR204 | XRAY | 2.39 | 0.249 | 0.267 | B | 382.0 | 352.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 2zoq | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | 6GESA | P27361 | 25 | 374 | 379.0 | 6H3:401,EWH:402 | Type1,Allosteric | Inactive | DFGin | 6.9525 | 15.557 | BLAminus | -139.32, 176.86 | 65.58, 87.64 | -106.07, 21.81 | 281.49, 72.32 | -67.67, -20.97 | in-in | in | 9.4645 | Saltbr-in | 2.8664 | HRD-in | -74.62, -54.83 | 79.01, 3.71 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7498 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -96.37, -37.93 | APE9-dihe-na | -66.29, 158.31 | APE8-dihe-in | -54.71, 127.96 | APE8-rot-in | 319.22 | APE67-dihe-in | -62.74, -20.38 | -53.12, -50.26 | APE12-dist-out | 14.2267 | APE11-dist-in | 11.0263 | APE10-dist-in | 6.9344 | APE9-dist-in | 4.4094 | None | None | None | XRAY | 2.07 | 0.172 | 0.213 | A | 380.0 | 350.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 6ges | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | 4QTBA | P27361 | 24 | 374 | 379.0 | 38Z:418 | Type1.5_Front | Inactive | DFGin | 6.9632 | 16.1915 | BLAminus | -128.63, 172.06 | 72.12, 87.31 | -104.64, 23.58 | 286.23, 74.76 | -64.07, -28.14 | in-in | in | 9.6383 | Saltbr-in | 2.6538 | HRD-in | -72.11, -54.76 | 73.09, 8.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7675 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -93.95, -29.12 | APE9-dihe-na | -67.78, 160.1 | APE8-dihe-in | -53.91, 125.98 | APE8-rot-in | 310.28 | APE67-dihe-in | -65.26, -17.27 | -52.54, -50.1 | APE12-dist-out | 14.1554 | APE11-dist-in | 10.8041 | APE10-dist-in | 6.8428 | APE9-dist-in | 4.4119 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | A | 380.0 | 351.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| MAPK3 | MK03_HUMAN | 4QTBB | P27361 | 27 | 374 | 379.0 | 38Z:412 | Type1.5_Front | Inactive | DFGin | 6.9886 | 16.0949 | BLAminus | -131.38, 169.9 | 76.01, 86.99 | -105.18, 21.27 | 288.36, 77.86 | -59.51, -32.2 | in-in | in | 9.5939 | Saltbr-in | 2.7088 | HRD-in | -72.51, -53.5 | 77.51, 5.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8241 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -90.9, -27.9 | APE9-dihe-na | -67.55, 157.04 | APE8-dihe-in | -54.84, 126.95 | APE8-rot-in | 308.82 | APE67-dihe-in | -67.72, -16.58 | -53.94, -47.75 | APE12-dist-out | 14.1875 | APE11-dist-in | 10.8583 | APE10-dist-in | 7.0815 | APE9-dist-in | 4.4109 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | B | 380.0 | 348.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|