| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| FES | AF-P07332-K3A | P07332 | 553 | 822 | 822.0 | No_ligand | No_ligand | Active | DFGin | 6.4175 | 14.6414 | BLAminus | -142.38, -175.33 | 53.57, 59.12 | -75.25, 15.18 | 286.52, 76.48 | -62.08, -27.31 | in-in | in | 7.592 | Saltbr-in | 2.6622 | HRD-in | -73.15, -46.35 | 69.14, -10.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8174 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.91, 80.44 | APE9-dihe-in | -112.25, 130.79 | APE8-dihe-in | -64.97, 100.04 | APE8-rot-na | 33.22 | APE67-dihe-in | -66.83, -15.49 | -47.81, -36.89 | APE12-dist-na | 7.8052 | APE11-dist-na | 11.9896 | APE10-dist-na | 9.2217 | APE9-dist-in | 5.4303 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 270.0 | 270.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | AF-P07332-K3 | TYR_FES_HUMAN | TYR | 2.1e-94 | 321.6 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | 3CBLA | P07332 | 448 | 821 | 822.0 | STU:60901,STU:60902,STU:60903 | Type1,Allosteric,Allosteric | Active | DFGin | 6.9919 | 14.3472 | BLAminus | -129.39, -161.99 | 36.63, 77.42 | -90.17, 19.41 | 283.19, 78.42 | -59.92, -34.07 | in-in | in | 7.0184 | Saltbr-in | 2.618 | HRD-in | -73.99, -51.91 | 78.82, -2.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7424 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -89.35, 116.24 | APE9-dihe-in | -118.34, 122.46 | APE8-dihe-in | -80.03, 88.22 | APE8-rot-na | 26.81 | APE67-dihe-in | -66.64, -12.19 | -59.28, -46.73 | APE12-dist-na | 13.8621 | APE11-dist-na | 9.6806 | APE10-dist-na | 8.625 | APE9-dist-in | 6.8668 | None | None | None | XRAY | 1.75 | 0.183 | 0.227 | A | 377.0 | 354.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 3cbl | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | 3CD3A | P07332 | 448 | 821 | 822.0 | STU:60901,STU:60902,STU:60903 | Type1,Allosteric,Allosteric | Active | DFGin | 7.0423 | 14.319 | BLAminus | -131.29, -161.96 | 36.95, 76.94 | -87.41, 20.64 | 283.25, 80.52 | -64.77, -30.01 | in-in | in | 6.9546 | Saltbr-in | 2.4508 | HRD-in | -75.66, -48.21 | 74.09, -7.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8131 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -102.76, 114.63 | APE9-dihe-in | -118.9, 123.98 | APE8-dihe-in | -79.16, 82.58 | APE8-rot-na | 23.88 | APE67-dihe-in | -66.61, -9.96 | -49.19, -54.65 | APE12-dist-na | 14.1032 | APE11-dist-na | 10.0433 | APE10-dist-na | 8.9304 | APE9-dist-in | 7.039 | None | PTR713 | PTR713 | XRAY | 1.98 | 0.188 | 0.247 | A | 377.0 | 351.0 | 4 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 3cd3 | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | AF-P07332-K1A | P07332 | 553 | 822 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.616 | 14.3011 | BLAminus | -138.77, -177.26 | 56.29, 65.33 | -79.53, 14.85 | 285.5, 79.64 | -63.21, -28.28 | in-in | in | 7.673 | Saltbr-in | 2.6555 | HRD-in | -69.27, -45.67 | 70.04, -15.15 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8285 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -138.25, 20.49 | APE9-dihe-in | -85.26, 122.58 | APE8-dihe-in | -74.28, 80.8 | APE8-rot-na | 32.03 | APE67-dihe-in | -71.29, -15.98 | -48.6, -40.01 | APE12-dist-na | 14.3882 | APE11-dist-na | 13.6242 | APE10-dist-na | 9.089 | APE9-dist-in | 7.0454 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 270.0 | 270.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | AF-P07332-K1 | TYR_FES_HUMAN | TYR | 2.1e-94 | 321.6 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | 6JMFA | P07332 | 450 | 821 | 822.0 | 9FC:903 | Type1 | Inactive | DFGin | 6.8162 | 14.679 | BLAminus | -130.91, -175.84 | 55.98, 73.35 | -96.13, 15.68 | 280.32, 79.2 | -57.92, -39.7 | in-in | in | 7.2168 | Saltbr-in | 2.6088 | HRD-in | -75.98, -48.96 | 77.02, -9.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7506 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 43.82, 40.62 | APE9-dihe-in | -61.47, 134.95 | APE8-dihe-in | -78.56, 75.16 | APE8-rot-na | 29.63 | APE67-dihe-in | -71.18, -14.66 | -50.39, -45.71 | APE12-dist-na | 8.4646 | APE11-dist-na | 11.6272 | APE10-dist-na | 11.1699 | APE9-dist-in | 7.231 | None | None | None | XRAY | 2.0 | 0.199 | 0.241 | A | 375.0 | 372.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 6jmf | TYR_FES_HUMAN | TYR | 6.4e-94 | 320.1 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | 3BKBA | P07332 | 449 | 821 | 822.0 | STU:826 | Type1 | Inactive | DFGin | 6.8661 | 14.4239 | BLAminus | -130.98, -162.57 | 38.75, 71.71 | -85.89, 14.89 | 281.41, 76.5 | -59.73, -36.44 | in-in | in | 6.7723 | Saltbr-in | 2.6204 | HRD-in | -78.26, -50.49 | 76.66, -9.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8204 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 47.37, 40.72 | APE9-dihe-in | -62.75, 132.26 | APE8-dihe-in | -76.49, 72.71 | APE8-rot-na | 30.4 | APE67-dihe-in | -70.68, -13.35 | -50.64, -47.62 | APE12-dist-na | 8.3405 | APE11-dist-na | 11.9812 | APE10-dist-na | 11.2254 | APE9-dist-in | 7.3541 | None | None | None | XRAY | 1.78 | 0.15 | 0.189 | A | 377.0 | 373.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 3bkb | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | 8XKPA | P07332 | 450 | 821 | 822.0 | A1LWS:903 | Type1 | Inactive | DFGin | 6.8893 | 14.6648 | BLAminus | -139.85, -171.28 | 56.78, 67.35 | -92.19, 14.82 | 278.0, 78.57 | -61.1, -30.38 | in-in | in | 7.5442 | Saltbr-in | 2.7546 | HRD-in | -72.91, -47.87 | 76.57, -5.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8412 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 51.79, 39.24 | APE9-dihe-in | -68.18, 139.98 | APE8-dihe-in | -82.66, 80.06 | APE8-rot-na | 34.15 | APE67-dihe-in | -67.92, -19.84 | -55.62, -43.43 | APE12-dist-na | 8.3857 | APE11-dist-na | 11.696 | APE10-dist-na | 10.9597 | APE9-dist-in | 7.1073 | None | None | None | XRAY | 2.05 | 0.192 | 0.234 | A | 375.0 | 372.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 8xkp | TYR_FES_HUMAN | TYR | 8.6e-94 | 319.7 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | 4E93A | P07332 | 448 | 822 | 822.0 | GUI:60901 | Type1 | None | DFGin | 7.2393 | 15.2064 | BLAminus | -147.07, -173.8 | 68.79, 70.92 | -92.31, 15.15 | 286.08, 92.67 | -61.32, -36.23 | in-in | in | 8.1557 | Saltbr-in | 2.8146 | HRD-in | -75.42, -47.46 | 72.8, -15.51 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8988 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -46.55 | APE8-dihe-in | -81.8, 74.32 | APE8-rot-na | 28.54 | APE67-dihe-in | -65.5, -10.65 | -48.91, -48.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.5764 | None | None | None | XRAY | 1.84 | 0.189 | 0.238 | A | 377.0 | 359.0 | 14 | 30 | 16 | 14 | [[561, 816]] | 1.0 | 4e93 | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| FES | FES_HUMAN | AF-P07332-K3A | P07332 | 553 | 822 | 822.0 | No_ligand | No_ligand | Active | DFGin | 6.4175 | 14.6414 | BLAminus | -142.38, -175.33 | 53.57, 59.12 | -75.25, 15.18 | 286.52, 76.48 | -62.08, -27.31 | in-in | in | 7.592 | Saltbr-in | 2.6622 | HRD-in | -73.15, -46.35 | 69.14, -10.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8174 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.91, 80.44 | APE9-dihe-in | -112.25, 130.79 | APE8-dihe-in | -64.97, 100.04 | APE8-rot-na | 33.22 | APE67-dihe-in | -66.83, -15.49 | -47.81, -36.89 | APE12-dist-na | 7.8052 | APE11-dist-na | 11.9896 | APE10-dist-na | 9.2217 | APE9-dist-in | 5.4303 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 270.0 | 270.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | AF-P07332-K3 | Homo sapiens | TYR_FES_HUMAN | TYR | 2.1e-94 | 321.6 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | 3CBLA | P07332 | 448 | 821 | 822.0 | STU:60901,STU:60902,STU:60903 | Type1,Allosteric,Allosteric | Active | DFGin | 6.9919 | 14.3472 | BLAminus | -129.39, -161.99 | 36.63, 77.42 | -90.17, 19.41 | 283.19, 78.42 | -59.92, -34.07 | in-in | in | 7.0184 | Saltbr-in | 2.618 | HRD-in | -73.99, -51.91 | 78.82, -2.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7424 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -89.35, 116.24 | APE9-dihe-in | -118.34, 122.46 | APE8-dihe-in | -80.03, 88.22 | APE8-rot-na | 26.81 | APE67-dihe-in | -66.64, -12.19 | -59.28, -46.73 | APE12-dist-na | 13.8621 | APE11-dist-na | 9.6806 | APE10-dist-na | 8.625 | APE9-dist-in | 6.8668 | None | None | None | XRAY | 1.75 | 0.183 | 0.227 | A | 377.0 | 354.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 3cbl | Homo sapiens | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | 3CD3A | P07332 | 448 | 821 | 822.0 | STU:60901,STU:60902,STU:60903 | Type1,Allosteric,Allosteric | Active | DFGin | 7.0423 | 14.319 | BLAminus | -131.29, -161.96 | 36.95, 76.94 | -87.41, 20.64 | 283.25, 80.52 | -64.77, -30.01 | in-in | in | 6.9546 | Saltbr-in | 2.4508 | HRD-in | -75.66, -48.21 | 74.09, -7.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8131 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -102.76, 114.63 | APE9-dihe-in | -118.9, 123.98 | APE8-dihe-in | -79.16, 82.58 | APE8-rot-na | 23.88 | APE67-dihe-in | -66.61, -9.96 | -49.19, -54.65 | APE12-dist-na | 14.1032 | APE11-dist-na | 10.0433 | APE10-dist-na | 8.9304 | APE9-dist-in | 7.039 | None | PTR713 | PTR713 | XRAY | 1.98 | 0.188 | 0.247 | A | 377.0 | 351.0 | 4 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 3cd3 | Homo sapiens | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | AF-P07332-K1A | P07332 | 553 | 822 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.616 | 14.3011 | BLAminus | -138.77, -177.26 | 56.29, 65.33 | -79.53, 14.85 | 285.5, 79.64 | -63.21, -28.28 | in-in | in | 7.673 | Saltbr-in | 2.6555 | HRD-in | -69.27, -45.67 | 70.04, -15.15 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8285 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -138.25, 20.49 | APE9-dihe-in | -85.26, 122.58 | APE8-dihe-in | -74.28, 80.8 | APE8-rot-na | 32.03 | APE67-dihe-in | -71.29, -15.98 | -48.6, -40.01 | APE12-dist-na | 14.3882 | APE11-dist-na | 13.6242 | APE10-dist-na | 9.089 | APE9-dist-in | 7.0454 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 270.0 | 270.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | AF-P07332-K1 | Homo sapiens | TYR_FES_HUMAN | TYR | 2.1e-94 | 321.6 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | 6JMFA | P07332 | 450 | 821 | 822.0 | 9FC:903 | Type1 | Inactive | DFGin | 6.8162 | 14.679 | BLAminus | -130.91, -175.84 | 55.98, 73.35 | -96.13, 15.68 | 280.32, 79.2 | -57.92, -39.7 | in-in | in | 7.2168 | Saltbr-in | 2.6088 | HRD-in | -75.98, -48.96 | 77.02, -9.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7506 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 43.82, 40.62 | APE9-dihe-in | -61.47, 134.95 | APE8-dihe-in | -78.56, 75.16 | APE8-rot-na | 29.63 | APE67-dihe-in | -71.18, -14.66 | -50.39, -45.71 | APE12-dist-na | 8.4646 | APE11-dist-na | 11.6272 | APE10-dist-na | 11.1699 | APE9-dist-in | 7.231 | None | None | None | XRAY | 2.0 | 0.199 | 0.241 | A | 375.0 | 372.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 6jmf | Homo sapiens | TYR_FES_HUMAN | TYR | 6.4e-94 | 320.1 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | 3BKBA | P07332 | 449 | 821 | 822.0 | STU:826 | Type1 | Inactive | DFGin | 6.8661 | 14.4239 | BLAminus | -130.98, -162.57 | 38.75, 71.71 | -85.89, 14.89 | 281.41, 76.5 | -59.73, -36.44 | in-in | in | 6.7723 | Saltbr-in | 2.6204 | HRD-in | -78.26, -50.49 | 76.66, -9.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8204 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 47.37, 40.72 | APE9-dihe-in | -62.75, 132.26 | APE8-dihe-in | -76.49, 72.71 | APE8-rot-na | 30.4 | APE67-dihe-in | -70.68, -13.35 | -50.64, -47.62 | APE12-dist-na | 8.3405 | APE11-dist-na | 11.9812 | APE10-dist-na | 11.2254 | APE9-dist-in | 7.3541 | None | None | None | XRAY | 1.78 | 0.15 | 0.189 | A | 377.0 | 373.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 3bkb | Homo sapiens | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | 8XKPA | P07332 | 450 | 821 | 822.0 | A1LWS:903 | Type1 | Inactive | DFGin | 6.8893 | 14.6648 | BLAminus | -139.85, -171.28 | 56.78, 67.35 | -92.19, 14.82 | 278.0, 78.57 | -61.1, -30.38 | in-in | in | 7.5442 | Saltbr-in | 2.7546 | HRD-in | -72.91, -47.87 | 76.57, -5.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8412 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 51.79, 39.24 | APE9-dihe-in | -68.18, 139.98 | APE8-dihe-in | -82.66, 80.06 | APE8-rot-na | 34.15 | APE67-dihe-in | -67.92, -19.84 | -55.62, -43.43 | APE12-dist-na | 8.3857 | APE11-dist-na | 11.696 | APE10-dist-na | 10.9597 | APE9-dist-in | 7.1073 | None | None | None | XRAY | 2.05 | 0.192 | 0.234 | A | 375.0 | 372.0 | 0 | 30 | 30 | 0 | [[561, 816]] | 1.0 | 8xkp | Homo sapiens | TYR_FES_HUMAN | TYR | 8.6e-94 | 319.7 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| FES | FES_HUMAN | 4E93A | P07332 | 448 | 822 | 822.0 | GUI:60901 | Type1 | None | DFGin | 7.2393 | 15.2064 | BLAminus | -147.07, -173.8 | 68.79, 70.92 | -92.31, 15.15 | 286.08, 92.67 | -61.32, -36.23 | in-in | in | 8.1557 | Saltbr-in | 2.8146 | HRD-in | -75.42, -47.46 | 72.8, -15.51 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8988 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -46.55 | APE8-dihe-in | -81.8, 74.32 | APE8-rot-na | 28.54 | APE67-dihe-in | -65.5, -10.65 | -48.91, -48.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.5764 | None | None | None | XRAY | 1.84 | 0.189 | 0.238 | A | 377.0 | 359.0 | 14 | 30 | 16 | 14 | [[561, 816]] | 1.0 | 4e93 | Homo sapiens | TYR_FES_HUMAN | TYR | 6.6e-94 | 320.0 | 1.0 | 260.0 | 260.0 | 700 | 701 | 702 | 704 | 706 | 590 | 607 | 611 | 680 | 682 | 681 | 683.0 | 742 | 730 | 725 | 724 | 723 | 722 | 721 | 720 | 719 | 637 | Tyrosine-protein kinase Fes/Fps |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|