CK1_CSNK1A1 (Casein kinase I isoform alpha)

Total number of chains: 9
Active chains: 3
Family: CK1
Uniprot: KC1A_HUMAN
Kinase Domain Residues: 17 - 283
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 9 100.0% AF-P48729-K1A

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AF-P48729-K1A 9 291 337.0 No_ligand No_ligand Active DFGin 6.564 14.609 BLAminus -131.89, 178.07 63.83, 65.03 -83.92, 12.5 294.04, 95.5 -60.73, -24.65 in-in in 8.021 Saltbr-in 2.687 HRD-in -78.3, -43.51 64.68, 6.22 in-in-in SNCiii in-in ActLoopNT-in 2.861 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.38, 135.89 APE9-dihe-na 97.47, -177.39 APE8-dihe-in -78.29, 109.51 APE8-rot-in 300.56 APE67-dihe-in -57.65, -41.12 -48.47, -33.48 APE12-dist-in 12.229 APE11-dist-in 12.405 APE10-dist-in 6.785 APE9-dist-in 3.392 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[17, 283]] 1.0 AF-P48729-K1 CK1_CSNK1A1_HUMAN CK1 1.4e-121 410.8 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
AF-P48729-K3A 9 291 337.0 No_ligand No_ligand Active DFGin 6.689 14.729 BLAminus -135.46, -177.92 66.55, 52.14 -77.01, 10.21 297.91, 102.31 -60.85, -23.82 in-in in 8.078 Saltbr-in 2.725 HRD-in -80.68, -43.39 66.41, 6.55 in-in-in SNCiii in-in ActLoopNT-in 2.858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.73, 137.95 APE9-dihe-na 92.53, -176.06 APE8-dihe-in -78.26, 109.56 APE8-rot-in 298.23 APE67-dihe-in -57.65, -40.16 -46.1, -34.86 APE12-dist-in 12.171 APE11-dist-in 12.284 APE10-dist-in 6.784 APE9-dist-in 3.212 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[17, 283]] 1.0 AF-P48729-K3 CK1_CSNK1A1_HUMAN CK1 1.4e-121 410.8 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
6GZDA 9 305 337.0 LCI:1018 Type1 Active DFGin 6.702 14.844 BLAminus -131.55, 177.32 70.46, 86.44 -102.55, 22.91 293.61, 98.06 -62.66, -35.34 in-in in 8.096 Saltbr-in 3.131 HRD-in -82.14, -48.34 69.83, 12.74 in-in-in SNCiii in-in ActLoopNT-in 2.984 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.35, -32.42 APE9-dihe-na -87.44, -150.21 APE8-dihe-in -91.1, 131.82 APE8-rot-in 300.27 APE67-dihe-in -60.82, -38.86 -68.26, -34.55 APE12-dist-in 11.658 APE11-dist-in 11.949 APE10-dist-in 6.279 APE9-dist-in 3.639 None None None XRAY 2.28 0.177 0.221 A 374 297 0 0 0 0 [[17, 283]] 1.0 6gzd CK1_CSNK1A1_HUMAN CK1 6.2e-122 412.0 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
9OTYC 10 299 337.0 No_ligand No_ligand Inactive DFGin 7.083 15.363 BLAminus -135.53, -172.58 61.81, 59.74 -92.09, 12.17 285.02, 92.14 -62.04, -34.28 in-in in 7.316 Saltbr-in 3.183 HRD-in -76.97, -48.13 69.53, -5.6 in-in-out SNCiio in-out ActLoopNT-in 2.847 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iioo APE10-dihe-na -124.88, -19.03 APE9-dihe-na -58.79, -45.33 APE8-dihe-in -92.79, 76.12 APE8-rot-out 54.48 APE67-dihe-in -96.47, 1.16 -60.18, -48.56 APE12-dist-in 13.301 APE11-dist-in 10.464 APE10-dist-out 10.862 APE9-dist-out 6.49 None None None EM 3.0 999.0 999.0 C 294 261 24 0 0 0 [[17, 283]] 1.0 9oty CK1_CSNK1A1_HUMAN CK1 1.6e-121 410.6 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
7WTTA 9 305 337.0 No_ligand No_ligand Inactive DFGin 5.12 13.743 BLAminus -128.39, -173.14 62.38, 68.0 -81.66, 19.85 302.98, 140.15 -65.98, -40.09 in-in in 7.706 Saltbr-in 3.316 HRD-in -101.27, -56.01 70.75, -2.06 in-in-out SNCiio in-out ActLoopNT-in 3.26 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -73.94, -42.92 APE9-dihe-na -87.72, -162.75 APE8-dihe-in -87.85, 147.74 APE8-rot-out 176.57 APE67-dihe-in -67.85, -28.34 -88.15, -5.46 APE12-dist-in 11.815 APE11-dist-in 11.899 APE10-dist-in 6.009 APE9-dist-in 3.714 None None None EM 3.1 999.0 999.0 a 337 297 0 0 0 0 [[17, 283]] 1.0 7wtt CK1_CSNK1A1_HUMAN CK1 4.4e-122 412.5 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
5FQDC 10 303 337.0 No_ligand No_ligand Inactive DFGin 7.19 14.608 BLAminus -125.14, -175.38 65.4, 78.63 -95.45, 17.62 293.94, 97.24 -64.3, -25.66 in-in in 7.528 Saltbr-in 2.937 HRD-in -75.92, -48.67 70.64, 10.95 in-in-out SNCiio in-out ActLoopNT-in 2.89 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -109.2, 125.17 APE9-dihe-na 98.79, -173.66 APE8-dihe-in -78.36, 139.15 APE8-rot-out 66.08 APE67-dihe-in -62.19, -40.83 -65.42, -28.56 APE12-dist-in 12.817 APE11-dist-in 11.883 APE10-dist-in 6.369 APE9-dist-in 3.803 None None None XRAY 2.45 0.182 0.21 C 341 294 0 0 0 0 [[17, 283]] 1.0 5fqd CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
5FQDF 10 303 337.0 No_ligand No_ligand Inactive DFGin 7.261 14.617 BLAminus -126.36, -172.4 58.11, 85.84 -99.98, 16.26 293.59, 98.23 -62.63, -25.38 in-in in 7.545 Saltbr-in 2.932 HRD-in -76.28, -48.08 72.0, 10.39 in-in-out SNCiio in-out ActLoopNT-in 2.935 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -108.84, 125.52 APE9-dihe-na 98.6, -172.43 APE8-dihe-in -78.79, 134.52 APE8-rot-out 72.63 APE67-dihe-in -46.09, -48.64 -60.33, -42.7 APE12-dist-in 13.088 APE11-dist-in 11.909 APE10-dist-in 6.405 APE9-dist-in 3.786 None None None XRAY 2.45 0.182 0.21 F 341 294 0 0 0 0 [[17, 283]] 1.0 5fqd CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
8G66C 10 303 337.0 No_ligand No_ligand Inactive DFGin 6.684 14.691 BLAminus -132.63, -176.05 63.82, 67.83 -87.54, 23.41 293.98, 101.77 -61.01, -29.47 in-in in 7.697 Saltbr-in 2.668 HRD-in -73.13, -43.43 60.31, 11.81 in-in-out SNCiio in-out ActLoopNT-in 2.849 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iini APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -172.78 APE8-dihe-in -126.42, 94.07 APE8-rot-out 29.36 APE67-dihe-in -55.97, -42.77 -45.09, -31.87 APE12-dist-in 12.304 APE11-dist-in 11.937 APE10-dist-none 999.0 APE9-dist-in 5.399 None None None XRAY 3.45 0.215 0.272 C 341 289 5 0 0 1 [[17, 283]] 1.0 8g66 CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
8G66F 10 303 337.0 No_ligand No_ligand None DFGin 6.691 14.706 BLAminus -136.03, -174.06 61.85, 69.19 -78.04, 10.68 292.24, 95.4 -51.34, -23.46 in-in in 7.682 Saltbr-in 3.377 HRD-in -83.58, -49.33 62.86, 12.64 in-in-none SNCiin in-none ActLoopNT-in 2.983 ActLoopCT-none nonTYR APEdihe_aaini APEdist_iiii APE10-dihe-na -102.78, 114.36 APE9-dihe-na 120.82, 175.64 APE8-dihe-in -62.9, 131.79 APE8-rot-none 999.0 APE67-dihe-in -50.33, -44.66 -60.52, -40.89 APE12-dist-in 12.958 APE11-dist-in 11.933 APE10-dist-in 6.404 APE9-dist-in 3.831 None None None XRAY 3.45 0.215 0.272 F 341 294 0 0 0 0 [[17, 283]] 1.0 8g66 CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha

CK1_CSNK1A1 (Casein kinase I isoform alpha)

Total number of chains: 9
Active chains: 3
Family: CK1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 9 100.0% AF-P48729-K1A

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
KC1A_HUMAN AF-P48729-K1A P48729 9 291 337.0 No_ligand No_ligand Active DFGin 6.564 14.609 BLAminus -131.89, 178.07 63.83, 65.03 -83.92, 12.5 294.04, 95.5 -60.73, -24.65 in-in in 8.021 Saltbr-in 2.687 HRD-in -78.3, -43.51 64.68, 6.22 in-in-in SNCiii in-in ActLoopNT-in 2.861 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -112.38, 135.89 APE9-dihe-na 97.47, -177.39 APE8-dihe-in -78.29, 109.51 APE8-rot-in 300.56 APE67-dihe-in -57.65, -41.12 -48.47, -33.48 APE12-dist-in 12.229 APE11-dist-in 12.405 APE10-dist-in 6.785 APE9-dist-in 3.392 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[17, 283]] 1.0 AF-P48729-K1 Homo sapiens CK1_CSNK1A1_HUMAN CK1 1.4e-121 410.8 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN AF-P48729-K3A P48729 9 291 337.0 No_ligand No_ligand Active DFGin 6.689 14.729 BLAminus -135.46, -177.92 66.55, 52.14 -77.01, 10.21 297.91, 102.31 -60.85, -23.82 in-in in 8.078 Saltbr-in 2.725 HRD-in -80.68, -43.39 66.41, 6.55 in-in-in SNCiii in-in ActLoopNT-in 2.858 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.73, 137.95 APE9-dihe-na 92.53, -176.06 APE8-dihe-in -78.26, 109.56 APE8-rot-in 298.23 APE67-dihe-in -57.65, -40.16 -46.1, -34.86 APE12-dist-in 12.171 APE11-dist-in 12.284 APE10-dist-in 6.784 APE9-dist-in 3.212 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[17, 283]] 1.0 AF-P48729-K3 Homo sapiens CK1_CSNK1A1_HUMAN CK1 1.4e-121 410.8 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 6GZDA P48729 9 305 337.0 LCI:1018 Type1 Active DFGin 6.702 14.844 BLAminus -131.55, 177.32 70.46, 86.44 -102.55, 22.91 293.61, 98.06 -62.66, -35.34 in-in in 8.096 Saltbr-in 3.131 HRD-in -82.14, -48.34 69.83, 12.74 in-in-in SNCiii in-in ActLoopNT-in 2.984 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.35, -32.42 APE9-dihe-na -87.44, -150.21 APE8-dihe-in -91.1, 131.82 APE8-rot-in 300.27 APE67-dihe-in -60.82, -38.86 -68.26, -34.55 APE12-dist-in 11.658 APE11-dist-in 11.949 APE10-dist-in 6.279 APE9-dist-in 3.639 None None None XRAY 2.28 0.177 0.221 A 374 297 0 0 0 0 [[17, 283]] 1.0 6gzd Homo sapiens CK1_CSNK1A1_HUMAN CK1 6.2e-122 412.0 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 9OTYC P48729 10 299 337.0 No_ligand No_ligand Inactive DFGin 7.083 15.363 BLAminus -135.53, -172.58 61.81, 59.74 -92.09, 12.17 285.02, 92.14 -62.04, -34.28 in-in in 7.316 Saltbr-in 3.183 HRD-in -76.97, -48.13 69.53, -5.6 in-in-out SNCiio in-out ActLoopNT-in 2.847 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iioo APE10-dihe-na -124.88, -19.03 APE9-dihe-na -58.79, -45.33 APE8-dihe-in -92.79, 76.12 APE8-rot-out 54.48 APE67-dihe-in -96.47, 1.16 -60.18, -48.56 APE12-dist-in 13.301 APE11-dist-in 10.464 APE10-dist-out 10.862 APE9-dist-out 6.49 None None None EM 3.0 999.0 999.0 C 294 261 24 0 0 0 [[17, 283]] 1.0 9oty Homo sapiens CK1_CSNK1A1_HUMAN CK1 1.6e-121 410.6 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 7WTTA P48729 9 305 337.0 No_ligand No_ligand Inactive DFGin 5.12 13.743 BLAminus -128.39, -173.14 62.38, 68.0 -81.66, 19.85 302.98, 140.15 -65.98, -40.09 in-in in 7.706 Saltbr-in 3.316 HRD-in -101.27, -56.01 70.75, -2.06 in-in-out SNCiio in-out ActLoopNT-in 3.26 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -73.94, -42.92 APE9-dihe-na -87.72, -162.75 APE8-dihe-in -87.85, 147.74 APE8-rot-out 176.57 APE67-dihe-in -67.85, -28.34 -88.15, -5.46 APE12-dist-in 11.815 APE11-dist-in 11.899 APE10-dist-in 6.009 APE9-dist-in 3.714 None None None EM 3.1 999.0 999.0 a 337 297 0 0 0 0 [[17, 283]] 1.0 7wtt Homo sapiens CK1_CSNK1A1_HUMAN CK1 4.4e-122 412.5 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 5FQDC P48729 10 303 337.0 No_ligand No_ligand Inactive DFGin 7.19 14.608 BLAminus -125.14, -175.38 65.4, 78.63 -95.45, 17.62 293.94, 97.24 -64.3, -25.66 in-in in 7.528 Saltbr-in 2.937 HRD-in -75.92, -48.67 70.64, 10.95 in-in-out SNCiio in-out ActLoopNT-in 2.89 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -109.2, 125.17 APE9-dihe-na 98.79, -173.66 APE8-dihe-in -78.36, 139.15 APE8-rot-out 66.08 APE67-dihe-in -62.19, -40.83 -65.42, -28.56 APE12-dist-in 12.817 APE11-dist-in 11.883 APE10-dist-in 6.369 APE9-dist-in 3.803 None None None XRAY 2.45 0.182 0.21 C 341 294 0 0 0 0 [[17, 283]] 1.0 5fqd Homo sapiens CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 5FQDF P48729 10 303 337.0 No_ligand No_ligand Inactive DFGin 7.261 14.617 BLAminus -126.36, -172.4 58.11, 85.84 -99.98, 16.26 293.59, 98.23 -62.63, -25.38 in-in in 7.545 Saltbr-in 2.932 HRD-in -76.28, -48.08 72.0, 10.39 in-in-out SNCiio in-out ActLoopNT-in 2.935 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -108.84, 125.52 APE9-dihe-na 98.6, -172.43 APE8-dihe-in -78.79, 134.52 APE8-rot-out 72.63 APE67-dihe-in -46.09, -48.64 -60.33, -42.7 APE12-dist-in 13.088 APE11-dist-in 11.909 APE10-dist-in 6.405 APE9-dist-in 3.786 None None None XRAY 2.45 0.182 0.21 F 341 294 0 0 0 0 [[17, 283]] 1.0 5fqd Homo sapiens CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 8G66C P48729 10 303 337.0 No_ligand No_ligand Inactive DFGin 6.684 14.691 BLAminus -132.63, -176.05 63.82, 67.83 -87.54, 23.41 293.98, 101.77 -61.01, -29.47 in-in in 7.697 Saltbr-in 2.668 HRD-in -73.13, -43.43 60.31, 11.81 in-in-out SNCiio in-out ActLoopNT-in 2.849 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iini APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -172.78 APE8-dihe-in -126.42, 94.07 APE8-rot-out 29.36 APE67-dihe-in -55.97, -42.77 -45.09, -31.87 APE12-dist-in 12.304 APE11-dist-in 11.937 APE10-dist-none 999.0 APE9-dist-in 5.399 None None None XRAY 3.45 0.215 0.272 C 341 289 5 0 0 1 [[17, 283]] 1.0 8g66 Homo sapiens CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha
KC1A_HUMAN 8G66F P48729 10 303 337.0 No_ligand No_ligand None DFGin 6.691 14.706 BLAminus -136.03, -174.06 61.85, 69.19 -78.04, 10.68 292.24, 95.4 -51.34, -23.46 in-in in 7.682 Saltbr-in 3.377 HRD-in -83.58, -49.33 62.86, 12.64 in-in-none SNCiin in-none ActLoopNT-in 2.983 ActLoopCT-none nonTYR APEdihe_aaini APEdist_iiii APE10-dihe-na -102.78, 114.36 APE9-dihe-na 120.82, 175.64 APE8-dihe-in -62.9, 131.79 APE8-rot-none 999.0 APE67-dihe-in -50.33, -44.66 -60.52, -40.89 APE12-dist-in 12.958 APE11-dist-in 11.933 APE10-dist-in 6.404 APE9-dist-in 3.831 None None None XRAY 3.45 0.215 0.272 F 341 294 0 0 0 0 [[17, 283]] 1.0 8g66 Homo sapiens CK1_CSNK1A1_HUMAN CK1 2.7e-121 409.9 1 261 261 156 157 158 160 162 46 60 64 133 135 134 136 203 191 186 185 184 183 182 181 180 91 Casein kinase I isoform alpha

CK1_CSNK1A1 (Casein kinase I isoform alpha)

Total number of chains: 0
Active chains: 0
Family: CK1
Spatial label Dihedral label Number of Chains Percent Representative

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name