| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CSNK1A1 | AF-P48729-K1A | P48729 | 9 | 291 | 337.0 | No_ligand | No_ligand | Active | DFGin | 6.5643 | 14.6086 | BLAminus | -131.89, 178.07 | 63.83, 65.03 | -83.92, 12.5 | 294.04, 95.5 | -60.73, -24.65 | in-in | in | 8.0209 | Saltbr-in | 2.6865 | HRD-in | -78.3, -43.51 | 64.68, 6.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8612 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.38, 135.89 | APE9-dihe-na | 97.47, -177.39 | APE8-dihe-in | -78.29, 109.51 | APE8-rot-in | 300.56 | APE67-dihe-in | -57.65, -41.12 | -48.47, -33.48 | APE12-dist-in | 12.2289 | APE11-dist-in | 12.4053 | APE10-dist-in | 6.7846 | APE9-dist-in | 3.3919 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 283.0 | 283.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | AF-P48729-K1 | CK1_CSNK1A1_HUMAN | CK1 | 1.4e-121 | 410.8 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | AF-P48729-K3A | P48729 | 9 | 291 | 337.0 | No_ligand | No_ligand | Active | DFGin | 6.6893 | 14.7295 | BLAminus | -135.46, -177.92 | 66.55, 52.14 | -77.01, 10.21 | 297.91, 102.31 | -60.85, -23.82 | in-in | in | 8.0784 | Saltbr-in | 2.7255 | HRD-in | -80.68, -43.39 | 66.41, 6.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8581 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.73, 137.95 | APE9-dihe-na | 92.53, -176.06 | APE8-dihe-in | -78.26, 109.56 | APE8-rot-in | 298.23 | APE67-dihe-in | -57.65, -40.16 | -46.1, -34.86 | APE12-dist-in | 12.1714 | APE11-dist-in | 12.2838 | APE10-dist-in | 6.7843 | APE9-dist-in | 3.2123 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 283.0 | 283.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | AF-P48729-K3 | CK1_CSNK1A1_HUMAN | CK1 | 1.4e-121 | 410.8 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 6GZDA | P48729 | 9 | 305 | 337.0 | LCI:1018 | Type1 | Active | DFGin | 6.7019 | 14.844 | BLAminus | -131.55, 177.32 | 70.46, 86.44 | -102.55, 22.91 | 293.61, 98.06 | -62.66, -35.34 | in-in | in | 8.0957 | Saltbr-in | 3.1314 | HRD-in | -82.14, -48.34 | 69.83, 12.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.984 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.35, -32.42 | APE9-dihe-na | -87.44, -150.21 | APE8-dihe-in | -91.1, 131.82 | APE8-rot-in | 300.27 | APE67-dihe-in | -60.82, -38.86 | -68.26, -34.55 | APE12-dist-in | 11.6581 | APE11-dist-in | 11.9492 | APE10-dist-in | 6.2789 | APE9-dist-in | 3.6388 | None | None | None | XRAY | 2.28 | 0.177 | 0.221 | A | 374.0 | 297.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 6gzd | CK1_CSNK1A1_HUMAN | CK1 | 6.2e-122 | 412.0 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 9OTYC | P48729 | 10 | 299 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 7.0832 | 15.3632 | BLAminus | -135.53, -172.58 | 61.81, 59.74 | -92.09, 12.17 | 285.02, 92.14 | -62.04, -34.28 | in-in | in | 7.3155 | Saltbr-in | 3.1825 | HRD-in | -76.97, -48.13 | 69.53, -5.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8473 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -124.88, -19.03 | APE9-dihe-na | -58.79, -45.33 | APE8-dihe-in | -92.79, 76.12 | APE8-rot-out | 54.48 | APE67-dihe-in | -96.47, 1.16 | -60.18, -48.56 | APE12-dist-in | 13.3013 | APE11-dist-in | 10.4642 | APE10-dist-out | 10.8617 | APE9-dist-out | 6.49 | None | None | None | EM | 3.0 | 999.0 | 999.0 | C | 294.0 | 261.0 | 24 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 9oty | CK1_CSNK1A1_HUMAN | CK1 | 1.6e-121 | 410.6 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 7WTTA | P48729 | 9 | 305 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1204 | 13.7434 | BLAminus | -128.39, -173.14 | 62.38, 68.0 | -81.66, 19.85 | 302.98, 140.15 | -65.98, -40.09 | in-in | in | 7.7056 | Saltbr-in | 3.3158 | HRD-in | -101.27, -56.01 | 70.75, -2.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.2597 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -73.94, -42.92 | APE9-dihe-na | -87.72, -162.75 | APE8-dihe-in | -87.85, 147.74 | APE8-rot-out | 176.57 | APE67-dihe-in | -67.85, -28.34 | -88.15, -5.46 | APE12-dist-in | 11.8151 | APE11-dist-in | 11.8986 | APE10-dist-in | 6.0092 | APE9-dist-in | 3.7141 | None | None | None | EM | 3.1 | 999.0 | 999.0 | a | 337.0 | 297.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 7wtt | CK1_CSNK1A1_HUMAN | CK1 | 4.4e-122 | 412.5 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 5FQDC | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 7.1899 | 14.608 | BLAminus | -125.14, -175.38 | 65.4, 78.63 | -95.45, 17.62 | 293.94, 97.24 | -64.3, -25.66 | in-in | in | 7.5278 | Saltbr-in | 2.9374 | HRD-in | -75.92, -48.67 | 70.64, 10.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8902 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -109.2, 125.17 | APE9-dihe-na | 98.79, -173.66 | APE8-dihe-in | -78.36, 139.15 | APE8-rot-out | 66.08 | APE67-dihe-in | -62.19, -40.83 | -65.42, -28.56 | APE12-dist-in | 12.8171 | APE11-dist-in | 11.8826 | APE10-dist-in | 6.3685 | APE9-dist-in | 3.8027 | None | None | None | XRAY | 2.45 | 0.182 | 0.21 | C | 341.0 | 294.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 5fqd | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 5FQDF | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 7.2613 | 14.6165 | BLAminus | -126.36, -172.4 | 58.11, 85.84 | -99.98, 16.26 | 293.59, 98.23 | -62.63, -25.38 | in-in | in | 7.5454 | Saltbr-in | 2.9315 | HRD-in | -76.28, -48.08 | 72.0, 10.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9347 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -108.84, 125.52 | APE9-dihe-na | 98.6, -172.43 | APE8-dihe-in | -78.79, 134.52 | APE8-rot-out | 72.63 | APE67-dihe-in | -46.09, -48.64 | -60.33, -42.7 | APE12-dist-in | 13.0884 | APE11-dist-in | 11.9092 | APE10-dist-in | 6.405 | APE9-dist-in | 3.7857 | None | None | None | XRAY | 2.45 | 0.182 | 0.21 | F | 341.0 | 294.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 5fqd | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 8G66C | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 6.6839 | 14.6911 | BLAminus | -132.63, -176.05 | 63.82, 67.83 | -87.54, 23.41 | 293.98, 101.77 | -61.01, -29.47 | in-in | in | 7.6968 | Saltbr-in | 2.6681 | HRD-in | -73.13, -43.43 | 60.31, 11.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8489 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iini | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -172.78 | APE8-dihe-in | -126.42, 94.07 | APE8-rot-out | 29.36 | APE67-dihe-in | -55.97, -42.77 | -45.09, -31.87 | APE12-dist-in | 12.304 | APE11-dist-in | 11.9371 | APE10-dist-none | 999.0 | APE9-dist-in | 5.3993 | None | None | None | XRAY | 3.45 | 0.215 | 0.272 | C | 341.0 | 289.0 | 5 | 35 | 34 | 1 | [[17, 283]] | 1.0 | 8g66 | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | 8G66F | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | None | DFGin | 6.691 | 14.7063 | BLAminus | -136.03, -174.06 | 61.85, 69.19 | -78.04, 10.68 | 292.24, 95.4 | -51.34, -23.46 | in-in | in | 7.6821 | Saltbr-in | 3.3772 | HRD-in | -83.58, -49.33 | 62.86, 12.64 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9827 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_iiii | APE10-dihe-na | -102.78, 114.36 | APE9-dihe-na | 120.82, 175.64 | APE8-dihe-in | -62.9, 131.79 | APE8-rot-none | 999.0 | APE67-dihe-in | -50.33, -44.66 | -60.52, -40.89 | APE12-dist-in | 12.9582 | APE11-dist-in | 11.9332 | APE10-dist-in | 6.4038 | APE9-dist-in | 3.8307 | None | None | None | XRAY | 3.45 | 0.215 | 0.272 | F | 341.0 | 294.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 8g66 | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CSNK1A1 | KC1A_HUMAN | AF-P48729-K1A | P48729 | 9 | 291 | 337.0 | No_ligand | No_ligand | Active | DFGin | 6.5643 | 14.6086 | BLAminus | -131.89, 178.07 | 63.83, 65.03 | -83.92, 12.5 | 294.04, 95.5 | -60.73, -24.65 | in-in | in | 8.0209 | Saltbr-in | 2.6865 | HRD-in | -78.3, -43.51 | 64.68, 6.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8612 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.38, 135.89 | APE9-dihe-na | 97.47, -177.39 | APE8-dihe-in | -78.29, 109.51 | APE8-rot-in | 300.56 | APE67-dihe-in | -57.65, -41.12 | -48.47, -33.48 | APE12-dist-in | 12.2289 | APE11-dist-in | 12.4053 | APE10-dist-in | 6.7846 | APE9-dist-in | 3.3919 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 283.0 | 283.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | AF-P48729-K1 | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 1.4e-121 | 410.8 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | AF-P48729-K3A | P48729 | 9 | 291 | 337.0 | No_ligand | No_ligand | Active | DFGin | 6.6893 | 14.7295 | BLAminus | -135.46, -177.92 | 66.55, 52.14 | -77.01, 10.21 | 297.91, 102.31 | -60.85, -23.82 | in-in | in | 8.0784 | Saltbr-in | 2.7255 | HRD-in | -80.68, -43.39 | 66.41, 6.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8581 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.73, 137.95 | APE9-dihe-na | 92.53, -176.06 | APE8-dihe-in | -78.26, 109.56 | APE8-rot-in | 298.23 | APE67-dihe-in | -57.65, -40.16 | -46.1, -34.86 | APE12-dist-in | 12.1714 | APE11-dist-in | 12.2838 | APE10-dist-in | 6.7843 | APE9-dist-in | 3.2123 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 283.0 | 283.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | AF-P48729-K3 | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 1.4e-121 | 410.8 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 6GZDA | P48729 | 9 | 305 | 337.0 | LCI:1018 | Type1 | Active | DFGin | 6.7019 | 14.844 | BLAminus | -131.55, 177.32 | 70.46, 86.44 | -102.55, 22.91 | 293.61, 98.06 | -62.66, -35.34 | in-in | in | 8.0957 | Saltbr-in | 3.1314 | HRD-in | -82.14, -48.34 | 69.83, 12.74 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.984 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.35, -32.42 | APE9-dihe-na | -87.44, -150.21 | APE8-dihe-in | -91.1, 131.82 | APE8-rot-in | 300.27 | APE67-dihe-in | -60.82, -38.86 | -68.26, -34.55 | APE12-dist-in | 11.6581 | APE11-dist-in | 11.9492 | APE10-dist-in | 6.2789 | APE9-dist-in | 3.6388 | None | None | None | XRAY | 2.28 | 0.177 | 0.221 | A | 374.0 | 297.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 6gzd | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 6.2e-122 | 412.0 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 9OTYC | P48729 | 10 | 299 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 7.0832 | 15.3632 | BLAminus | -135.53, -172.58 | 61.81, 59.74 | -92.09, 12.17 | 285.02, 92.14 | -62.04, -34.28 | in-in | in | 7.3155 | Saltbr-in | 3.1825 | HRD-in | -76.97, -48.13 | 69.53, -5.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8473 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iioo | APE10-dihe-na | -124.88, -19.03 | APE9-dihe-na | -58.79, -45.33 | APE8-dihe-in | -92.79, 76.12 | APE8-rot-out | 54.48 | APE67-dihe-in | -96.47, 1.16 | -60.18, -48.56 | APE12-dist-in | 13.3013 | APE11-dist-in | 10.4642 | APE10-dist-out | 10.8617 | APE9-dist-out | 6.49 | None | None | None | EM | 3.0 | 999.0 | 999.0 | C | 294.0 | 261.0 | 24 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 9oty | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 1.6e-121 | 410.6 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 7WTTA | P48729 | 9 | 305 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1204 | 13.7434 | BLAminus | -128.39, -173.14 | 62.38, 68.0 | -81.66, 19.85 | 302.98, 140.15 | -65.98, -40.09 | in-in | in | 7.7056 | Saltbr-in | 3.3158 | HRD-in | -101.27, -56.01 | 70.75, -2.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.2597 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -73.94, -42.92 | APE9-dihe-na | -87.72, -162.75 | APE8-dihe-in | -87.85, 147.74 | APE8-rot-out | 176.57 | APE67-dihe-in | -67.85, -28.34 | -88.15, -5.46 | APE12-dist-in | 11.8151 | APE11-dist-in | 11.8986 | APE10-dist-in | 6.0092 | APE9-dist-in | 3.7141 | None | None | None | EM | 3.1 | 999.0 | 999.0 | a | 337.0 | 297.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 7wtt | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 4.4e-122 | 412.5 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 5FQDC | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 7.1899 | 14.608 | BLAminus | -125.14, -175.38 | 65.4, 78.63 | -95.45, 17.62 | 293.94, 97.24 | -64.3, -25.66 | in-in | in | 7.5278 | Saltbr-in | 2.9374 | HRD-in | -75.92, -48.67 | 70.64, 10.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8902 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -109.2, 125.17 | APE9-dihe-na | 98.79, -173.66 | APE8-dihe-in | -78.36, 139.15 | APE8-rot-out | 66.08 | APE67-dihe-in | -62.19, -40.83 | -65.42, -28.56 | APE12-dist-in | 12.8171 | APE11-dist-in | 11.8826 | APE10-dist-in | 6.3685 | APE9-dist-in | 3.8027 | None | None | None | XRAY | 2.45 | 0.182 | 0.21 | C | 341.0 | 294.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 5fqd | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 5FQDF | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 7.2613 | 14.6165 | BLAminus | -126.36, -172.4 | 58.11, 85.84 | -99.98, 16.26 | 293.59, 98.23 | -62.63, -25.38 | in-in | in | 7.5454 | Saltbr-in | 2.9315 | HRD-in | -76.28, -48.08 | 72.0, 10.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9347 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -108.84, 125.52 | APE9-dihe-na | 98.6, -172.43 | APE8-dihe-in | -78.79, 134.52 | APE8-rot-out | 72.63 | APE67-dihe-in | -46.09, -48.64 | -60.33, -42.7 | APE12-dist-in | 13.0884 | APE11-dist-in | 11.9092 | APE10-dist-in | 6.405 | APE9-dist-in | 3.7857 | None | None | None | XRAY | 2.45 | 0.182 | 0.21 | F | 341.0 | 294.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 5fqd | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 8G66C | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | Inactive | DFGin | 6.6839 | 14.6911 | BLAminus | -132.63, -176.05 | 63.82, 67.83 | -87.54, 23.41 | 293.98, 101.77 | -61.01, -29.47 | in-in | in | 7.6968 | Saltbr-in | 2.6681 | HRD-in | -73.13, -43.43 | 60.31, 11.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8489 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iini | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -172.78 | APE8-dihe-in | -126.42, 94.07 | APE8-rot-out | 29.36 | APE67-dihe-in | -55.97, -42.77 | -45.09, -31.87 | APE12-dist-in | 12.304 | APE11-dist-in | 11.9371 | APE10-dist-none | 999.0 | APE9-dist-in | 5.3993 | None | None | None | XRAY | 3.45 | 0.215 | 0.272 | C | 341.0 | 289.0 | 5 | 35 | 34 | 1 | [[17, 283]] | 1.0 | 8g66 | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| CSNK1A1 | KC1A_HUMAN | 8G66F | P48729 | 10 | 303 | 337.0 | No_ligand | No_ligand | None | DFGin | 6.691 | 14.7063 | BLAminus | -136.03, -174.06 | 61.85, 69.19 | -78.04, 10.68 | 292.24, 95.4 | -51.34, -23.46 | in-in | in | 7.6821 | Saltbr-in | 3.3772 | HRD-in | -83.58, -49.33 | 62.86, 12.64 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9827 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_iiii | APE10-dihe-na | -102.78, 114.36 | APE9-dihe-na | 120.82, 175.64 | APE8-dihe-in | -62.9, 131.79 | APE8-rot-none | 999.0 | APE67-dihe-in | -50.33, -44.66 | -60.52, -40.89 | APE12-dist-in | 12.9582 | APE11-dist-in | 11.9332 | APE10-dist-in | 6.4038 | APE9-dist-in | 3.8307 | None | None | None | XRAY | 3.45 | 0.215 | 0.272 | F | 341.0 | 294.0 | 0 | 35 | 35 | 0 | [[17, 283]] | 1.0 | 8g66 | Homo sapiens | CK1_CSNK1A1_HUMAN | CK1 | 2.7e-121 | 409.9 | 1.0 | 261.0 | 261.0 | 156 | 157 | 158 | 160 | 162 | 46 | 60 | 64 | 133 | 135 | 134 | 136.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 91 | Casein kinase I isoform alpha |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|