Group |
Gene |
UniprotID |
Protein |
PDB |
Activity Label |
Spatial Label |
Dihedral Label |
Chelix-SaltBridge |
ActLoopNT-ActloopCT |
Ligand |
Type |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
AF-P31749-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6BUUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6BUUB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6NPZA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6NPZB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
4GV1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
0XZ |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3OCBA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XM1 |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3OCBB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XM1 |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3OW4A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SMY |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3OW4B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SMY |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3QKLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SMR |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3QKMA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SM9 |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
4EKKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
4EKKB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
4EKLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
0RF |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3CQUA |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
CQU |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3CQWA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
CQW |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3MV5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XFE |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3MVHA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
WFE |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6CCYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
EX4 |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3QKKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SMH |
Type1.5_Front |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
3O96A |
Inactive |
DFGout |
BBAminus |
none-none |
out-none |
IQO |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6HHHA |
Inactive |
DFGout |
BBAminus |
none-none |
out-out |
G4Q |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6HHJA |
Inactive |
DFGout |
BBAminus |
out-out |
out-out |
G4H |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6S9WA |
Inactive |
DFGout |
BBAminus |
out-out |
out-out |
L1Z |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
4EJNA |
Inactive |
DFGout |
BBAminus |
none-none |
out-out |
0R4 |
Type1 |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
5KCVA |
Inactive |
DFGout |
None |
none-none |
none-none |
6S1 |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
7APJA |
Inactive |
DFGout |
None |
none-none |
none-none |
No_ligand |
No_ligand |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6HHFA |
Inactive |
None |
None |
none-none |
out-none |
G4K |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6HHGA |
Inactive |
None |
None |
none-none |
out-out |
G4T |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6HHIA |
Inactive |
None |
None |
none-none |
out-out |
G4N |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
6S9XA |
Inactive |
None |
None |
none-none |
out-out |
L1W |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
7NH4A |
Inactive |
None |
None |
none-none |
out-out |
UCE |
Allosteric |
AGC |
AKT1 |
AKT1_HUMAN |
RAC-alpha serine/threonine-protein kinase |
7NH5A |
Inactive |
None |
None |
none-none |
out-out |
UC8 |
Allosteric |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
AF-P31751-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3E87A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G95 |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3E87B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G95 |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1O6KA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1O6LA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
2JDOA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
I5S |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
2JDRA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L20 |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
2UW9A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
GVP |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
2X39A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
X39 |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
2XH5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
X37 |
Type1 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3D0EA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G93 |
Type1.5_Back |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3D0EB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G93 |
Type1.5_Back |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3E88A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G96 |
Type1.5_Back |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3E88B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G96 |
Type1.5_Back |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3E8DA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G98 |
Type1.5_Back |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
3E8DB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
G98 |
Type1.5_Back |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
8Q61A |
Inactive |
DFGout |
BBAminus |
out-out |
out-none |
K06 |
Type3 |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1GZKA |
Inactive |
DFGout |
None |
in-none |
none-none |
No_ligand |
No_ligand |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1GZOA |
Inactive |
DFGout |
None |
in-none |
none-none |
No_ligand |
No_ligand |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1GZNA |
Inactive |
DFGout |
None |
in-none |
none-none |
No_ligand |
No_ligand |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1MRVA |
Inactive |
DFGout |
None |
none-none |
none-none |
No_ligand |
No_ligand |
AGC |
AKT2 |
AKT2_HUMAN |
RAC-beta serine/threonine-protein kinase |
1MRYA |
Inactive |
DFGout |
None |
none-none |
none-out |
No_ligand |
No_ligand |
AGC |
AKT3 |
AKT3_HUMAN |
RAC-gamma serine/threonine-protein kinase |
AF-Q9Y243-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
CDC42BPA |
MRCKA_HUMAN |
Serine/threonine-protein kinase MRCK alpha |
AF-Q5VT25-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
AF-Q9Y5S2-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
3QFVA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
NM7 |
Type1 |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
3QFVB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
NM7 |
Type1 |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
4UAKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP |
Type1 |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
4UALA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3FV |
Type1 |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
5OTEA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AQE |
Type1 |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
5OTFA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AQ5 |
Type1 |
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
3TKUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
M77
M77
|
Type1
Allosteric
|
AGC |
CDC42BPB |
MRCKB_HUMAN |
Serine/threonine-protein kinase MRCK beta |
3TKUB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
M77
M77
|
Type1
Allosteric
|
AGC |
CDC42BPG |
MRCKG_HUMAN |
Serine/threonine-protein kinase MRCK gamma |
AF-Q6DT37-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
CIT |
CTRO_HUMAN |
Citron Rho-interacting kinase |
AF-O14578-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
DMPK |
DMPK_HUMAN |
Myotonin-protein kinase |
AF-Q09013-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
DMPK |
DMPK_HUMAN |
Myotonin-protein kinase |
2VD5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI8 |
Type1 |
AGC |
DMPK |
DMPK_HUMAN |
Myotonin-protein kinase |
2VD5B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI8 |
Type1 |
AGC |
GRK1 |
GRK1_HUMAN |
Rhodopsin kinase GRK1 |
AF-Q15835-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
AF-P25098-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5UVCA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8PV |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5UKLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SIX |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5HE1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZS2 |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
6C2YA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
EJS |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
4MK0A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
29X |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
7K7LA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
W4D |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
7K7ZA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
W4G |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
3V5WA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8PR |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
4PNKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
KZQ |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5WG3A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AFM |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5WG4A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AFV |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5WG5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ZSO |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5UUUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
QRW |
Type1.5_Front |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
5UKKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8DJ |
Type1.5_Front |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
6U7CA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
Q1Y |
Type1.5_Front |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
3CIKA |
Inactive |
DFGin |
None |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
7PWDA |
Inactive |
DFGin |
None |
in-in |
in-in |
8DS |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
3KRWA |
Inactive |
DFGin |
None |
in-in |
in-in |
BA1 |
Type1 |
AGC |
GRK2 |
ARBK1_HUMAN |
Beta-adrenergic receptor kinase 1 |
3KRXA |
Inactive |
DFGin |
None |
in-in |
in-in |
BA1 |
Type1 |
AGC |
GRK3 |
ARBK2_HUMAN |
G protein-coupled receptor kinase 3 |
AF-P35626-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK4 |
GRK4_HUMAN |
G protein-coupled receptor kinase 4 |
AF-P32298-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK4 |
GRK4_HUMAN |
G protein-coupled receptor kinase 4 |
4YHJA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AN2 |
Type1 |
AGC |
GRK4 |
GRK4_HUMAN |
G protein-coupled receptor kinase 4 |
4YHJB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AN2 |
Type1 |
AGC |
GRK5 |
GRK5_HUMAN |
G protein-coupled receptor kinase 5 |
AF-P34947-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK5 |
GRK5_HUMAN |
G protein-coupled receptor kinase 5 |
4TNBA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SGV |
Type1 |
AGC |
GRK5 |
GRK5_HUMAN |
G protein-coupled receptor kinase 5 |
4TNDA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
GRK5 |
GRK5_HUMAN |
G protein-coupled receptor kinase 5 |
8UAPA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
W2T |
Type1 |
AGC |
GRK5 |
GRK5_HUMAN |
G protein-coupled receptor kinase 5 |
6PJXA |
Inactive |
DFGin |
None |
in-in |
in-in |
SGV |
Type1 |
AGC |
GRK5 |
GRK5_HUMAN |
G protein-coupled receptor kinase 5 |
8UAQA |
Inactive |
DFGin |
None |
in-in |
in-in |
W3F |
Type1 |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
AF-P43250-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
2ACXA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
2ACXB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
3NYNA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SGV |
Type1 |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
3NYNB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SGV |
Type1 |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
3NYOA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AMP |
Type1 |
AGC |
GRK6 |
GRK6_HUMAN |
G protein-coupled receptor kinase 6 |
3NYOB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AMP |
Type1 |
AGC |
GRK7 |
GRK7_HUMAN |
Rhodopsin kinase GRK7 |
AF-Q8WTQ7-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
LATS1 |
LATS1_HUMAN |
Serine/threonine-protein kinase LATS1 |
AF-O95835-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
LATS2 |
LATS2_HUMAN |
Serine/threonine-protein kinase LATS2 |
AF-Q9NRM7-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
MAST1 |
MAST1_HUMAN |
Microtubule-associated serine/threonine-protein kinase 1 |
AF-Q9Y2H9-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
MAST2 |
MAST2_HUMAN |
Microtubule-associated serine/threonine-protein kinase 2 |
AF-Q6P0Q8-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
MAST3 |
MAST3_HUMAN |
Microtubule-associated serine/threonine-protein kinase 3 |
AF-O60307-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
MAST4 |
MAST4_HUMAN |
Microtubule-associated serine/threonine-protein kinase 4 |
AF-O15021-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
MASTL |
GWL_HUMAN |
Serine/threonine-protein kinase greatwall |
AF-Q96GX5-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
MASTL |
GWL_HUMAN |
Serine/threonine-protein kinase greatwall |
5LOHA |
Inactive |
DFGin |
BLAplus |
none-none |
out-out |
STU |
Type1 |
AGC |
MASTL |
GWL_HUMAN |
Serine/threonine-protein kinase greatwall |
5LOHB |
Inactive |
None |
None |
none-none |
none-out |
STU |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXD |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXE |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXF |
None |
DFGin |
BLAminus |
in-none |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXG |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORXH |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1F8 |
Allosteric |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
8DQTA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
U35
U35
U35
|
Allosteric
Allosteric
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORZA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
2A2
BI4
|
Allosteric
Type1
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORZB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
2A2
BI4
|
Allosteric
Type1
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORZC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
2A2
BI4
|
Allosteric
Type1
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3ORZD |
Active |
DFGin |
BLAminus |
in-in |
in-in |
2A2
BI4
|
Allosteric
Type1
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3OTUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
J30
BI4
|
Allosteric
Type1.5_Front
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
AF-O15530-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1Z5MA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LI8 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2PE0A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
39Z |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2PE1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
517 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2PE2A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
464 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NUSA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
JNZ |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NUUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
JOZ |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NUYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
JPZ |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1UU9A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI3 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1H1WA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1UVRA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI8 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NUNA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
JMZ |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2XCHA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
CKG |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5HKMA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
61Y |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5HNGA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
62O |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5HO7A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
63L |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5HO8A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
63E |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1OKYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
STU |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1OKZA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
UCN |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1UU3A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LY4 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1UU7A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI2 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
1UU8A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI1 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NAYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
MP6 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NAYB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
MP6 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3RWPA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ABQ |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3RWQA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3RW |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3SC1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3S1 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3H9OA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
9BD |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2R7BA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
253 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3IONA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8H1 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3IOPA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8I1 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QCQA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q0 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QCSA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q1 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2BIYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3HRCA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3RCJA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3RC |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4RRVA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5ACKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
537 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVMA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADE |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVNA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADN |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVPA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVPB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVPC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVPD |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4CT2A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3PWYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SYP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5MRDA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
2XCKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
MH4 |
Type1 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3HRFA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
P47
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4A06A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
A06
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4AW0A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
MJF
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4AW1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
21O
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4RQKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
R1S
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4RQVA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
R2S
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
5LVOA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
78W
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4CT1A |
None |
DFGin |
BLAminus |
in-none |
in-in |
ATP
31S
|
Type1
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4XX9A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
RF4
RF4
|
Type1
Allosteric
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
4A07A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP
AZ7
AZ7
|
Type1
Allosteric
Allosteric
|
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QCXA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q2 |
Type1.5_Back |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QCYA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q3 |
Type1.5_Front |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QD0A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q4 |
Type1.5_Front |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QD3A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q5 |
Type1.5_Front |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QD4A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3Q6 |
Type1.5_Front |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3NAXA |
Inactive |
DFGout |
BBAminus |
out-out |
in-none |
MP7 |
Type2 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QC4A |
Inactive |
DFGout |
BBAminus |
out-out |
in-in |
MP7 |
Type2 |
AGC |
PDPK1 |
PDPK1_HUMAN |
3-phosphoinositide-dependent protein kinase 1 |
3QC4B |
Inactive |
DFGout |
None |
out-out |
in-in |
MP7 |
Type2 |
AGC |
PKN1 |
PKN1_HUMAN |
Serine/threonine-protein kinase N1 |
4OTDA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PKN1 |
PKN1_HUMAN |
Serine/threonine-protein kinase N1 |
4OTGA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
2V9 |
Type1 |
AGC |
PKN1 |
PKN1_HUMAN |
Serine/threonine-protein kinase N1 |
AF-Q16512-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PKN1 |
PKN1_HUMAN |
Serine/threonine-protein kinase N1 |
4OTHA |
Inactive |
DFGin |
BLAplus |
in-in |
out-none |
DRN |
Type1 |
AGC |
PKN1 |
PKN1_HUMAN |
Serine/threonine-protein kinase N1 |
4OTIA |
Inactive |
DFGin |
BLAplus |
in-in |
none-none |
MI1 |
Type1 |
AGC |
PKN2 |
PKN2_HUMAN |
Serine/threonine-protein kinase N2 |
AF-Q16513-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PKN2 |
PKN2_HUMAN |
Serine/threonine-protein kinase N2 |
4CRSA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
AGS |
Type1 |
AGC |
PKN3 |
PKN3_HUMAN |
Serine/threonine-protein kinase N3 |
AF-Q6P5Z2-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4AE6A |
Inactive |
DFGin |
ABAminus |
out-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4AE6B |
Inactive |
DFGin |
ABAminus |
out-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4AE9A |
Inactive |
DFGin |
ABAminus |
out-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4AE9B |
Inactive |
DFGin |
ABAminus |
out-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
7Y1GB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
I5G |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3AMBA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
VX6 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8X5LA |
Inactive |
DFGin |
ABAminus |
in-out |
out-out |
RKD |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8X5LB |
Inactive |
DFGin |
ABAminus |
out-out |
out-out |
RKD |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5IZJA |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
6J9 |
Allosteric |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5IZJB |
Inactive |
DFGin |
BLAminus |
out-out |
in-in |
6J9 |
Allosteric |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5J5XA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
6J9 |
Allosteric |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
AF-P17612-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6BYSA |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6BYSC |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6BYSE |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6BYSG |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6NO7A |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6NO7C |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3AGMA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5IZFA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3MVJB |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3NX8A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6WJFA |
Inactive |
DFGin |
BLAminus |
out-out |
out-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6WJFB |
Inactive |
DFGin |
BLAminus |
out-out |
out-out |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6WJGA |
Inactive |
DFGin |
BLAminus |
out-out |
out-in |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6WJGB |
Inactive |
DFGin |
BLAminus |
out-out |
out-out |
No_ligand |
No_ligand |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4WB8A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4WB5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6NO7E |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6NO7G |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3AGLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A03 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3AGLB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
A03 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3L9LA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L9L |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3L9LB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L9L |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3OOGA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
YTP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3OVVA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
1SB |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3OWPA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
2SB |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3OXTA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3SB |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3P0MA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4SB |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3POOA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
S69 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3VQHA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
IQB |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4UJ1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
NVX |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4UJ2A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
NVV |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4UJ9A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
S3N |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4UJAA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4L7 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4UJBA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8BQ |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5BX6A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
495 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5BX7A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4W1 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5UZKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
504 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6QJ7A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
J4B |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
7Y1GA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
I5G |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6C0UA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
EE4 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3MVJA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XFE |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3MVJE |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XFE |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3L9MA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L9M |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3L9MB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L9M |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3L9NA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
L9N |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4WB7A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4WB7B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6BYRA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6BYRC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8FE2A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XTI |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8FE2B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XTI |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8FE5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XTT |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8FE5B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XTT |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8FECA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XU0 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
8FECB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XU0 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
2GU8A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
796 |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4WB6A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
4WB6B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
5N23A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
35R |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
3AMAA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
SKE |
Type1 |
AGC |
PRKACA |
KAPCA_HUMAN |
cAMP-dependent protein kinase catalytic subunit alpha |
6FRXA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
E3Z |
Type1 |
AGC |
PRKACB |
KAPCB_HUMAN |
cAMP-dependent protein kinase catalytic subunit beta |
AF-P22694-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKACG |
KAPCG_HUMAN |
cAMP-dependent protein kinase catalytic subunit gamma |
AF-P22612-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
AF-P17252-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
4RA4A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3KZ |
Type1 |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
3IW4A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LW4 |
Type1 |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
3IW4B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LW4 |
Type1 |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
3IW4C |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LW4 |
Type1 |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
8U37A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
V5U |
Type1 |
AGC |
PRKCA |
KPCA_HUMAN |
Protein kinase C alpha type |
8UAKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
W39 |
Type1 |
AGC |
PRKCB |
KPCB_HUMAN |
Protein kinase C beta type |
AF-P05771-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCB |
KPCB_HUMAN |
Protein kinase C beta type |
2I0EA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
PDS |
Type1 |
AGC |
PRKCB |
KPCB_HUMAN |
Protein kinase C beta type |
2I0EB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
PDS |
Type1 |
AGC |
PRKCD |
KPCD_HUMAN |
Protein kinase C delta type |
AF-Q05655-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCE |
KPCE_HUMAN |
Protein kinase C epsilon type |
AF-Q02156-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCG |
KPCG_HUMAN |
Protein kinase C gamma type |
AF-P05129-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCH |
KPCL_HUMAN |
Protein kinase C eta type |
AF-P24723-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCH |
KPCL_HUMAN |
Protein kinase C eta type |
8FP1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
XXF |
Type1 |
AGC |
PRKCH |
KPCL_HUMAN |
Protein kinase C eta type |
8FP3A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
Y3I |
Type1 |
AGC |
PRKCH |
KPCL_HUMAN |
Protein kinase C eta type |
3TXOA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
07U |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
6ILZA |
Inactive |
DFGin |
ABAminus |
in-none |
in-in |
AFU |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
AF-P41743-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3A8XA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3A8XB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3A8WA |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
ATP |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3A8WB |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
ATP |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
6ILZC |
None |
DFGin |
BLAminus |
in-none |
in-in |
AFU |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
6ILZE |
None |
DFGin |
BLAminus |
in-none |
in-in |
AFU |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
6ILZG |
None |
DFGin |
BLAminus |
in-none |
in-in |
AFU |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3ZH8A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
C58 |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3ZH8B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
C58 |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
3ZH8C |
Active |
DFGin |
BLAminus |
in-in |
in-in |
C58 |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
5LIHA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
5LIHB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
5LI9A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ACP |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
5LI1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKCI |
KPCI_HUMAN |
Protein kinase C iota type |
1ZRZA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
BI1 |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
AF-Q04759-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
4Q9ZA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
PZW |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
4Q9ZB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
PZW |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
4RA5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3L0 |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
4RA5B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3L0 |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
2JEDA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LG8 |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
2JEDB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
LG8 |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
5F9EA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
5VS |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
5F9EB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
5VS |
Type1 |
AGC |
PRKCQ |
KPCT_HUMAN |
Protein kinase C theta type |
1XJDA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
STU |
Type1 |
AGC |
PRKCZ |
KPCZ_HUMAN |
Protein kinase C zeta type |
AF-Q05513-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4UA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
EX6 |
Allosteric |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4UB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
EX6 |
Allosteric |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4WA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
EZJ |
Allosteric |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4WB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
EZJ |
Allosteric |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4TA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
PCG
ATP
|
Allosteric
Type1
|
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4TB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
PCG
ATP
|
Allosteric
Type1
|
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4VA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
EXZ |
Allosteric |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7T4VB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
EXZ |
Allosteric |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
AF-Q13976-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6BDLA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
No_ligand |
No_ligand |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6BDLB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6BG2A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6BG2B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6BG2C |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6BG2D |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7LV3A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
7LV3B |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
PRKG1 |
KGP1_HUMAN |
cGMP-dependent protein kinase 1 |
6C0TA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
EE4 |
Type1.5_Front |
AGC |
PRKG2 |
KGP2_HUMAN |
cGMP-dependent protein kinase 2 |
AF-Q13237-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
PRKX |
PRKX_HUMAN |
cAMP-dependent protein kinase catalytic subunit PRKX |
AF-P51817-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NDMA |
Inactive |
DFGin |
ABAminus |
in-out |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NCZA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3NC |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NCZB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3NC |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NCZC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3NC |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NCZD |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3NC |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NDMB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3ND |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NDMC |
Inactive |
DFGin |
ABAminus |
in-in |
in-none |
3ND |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3NDMD |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3ND |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNFA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B4V |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNFB |
Inactive |
DFGin |
ABAminus |
in-in |
in-none |
B4V |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNFC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B4V |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNFD |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B4V |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNGA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B4Y |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNGB |
Inactive |
DFGin |
ABAminus |
in-in |
in-none |
B4Y |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNGC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B4Y |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNGD |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B4Y |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNHA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B5G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNHB |
Inactive |
DFGin |
ABAminus |
in-in |
in-none |
B5G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNHC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B5G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNHD |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
B5G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
6E9WA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
J0P |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
6E9WB |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
J0P |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
AF-Q13464-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S26D |
None |
DFGin |
BLAminus |
in-in |
in-none |
No_ligand |
No_ligand |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S26A |
None |
DFGin |
BLAminus |
in-in |
in-none |
86K |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S26B |
None |
DFGin |
BLAminus |
in-in |
none-none |
86K |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2V55A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2V55C |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TV7A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
07Q |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TV7B |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
07Q |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TV7C |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
07Q |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TV7D |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
07Q |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3V8SA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
0HD |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3V8SB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
0HD |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3V8SC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
0HD |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3V8SD |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
0HD |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4W7PA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3J7 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4W7PB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3J7 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4W7PC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3J7 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4W7PD |
Active |
DFGin |
BLAminus |
in-in |
in-in |
3J7 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7JOUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
VFS |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2ESMA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
M77 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2ESMB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
M77 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2ETKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
HFS |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2ETKB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
HFS |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2ETRA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
Y27 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
2ETRB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
Y27 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3D9VA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
H52 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3D9VB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
H52 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4YVCA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4KH |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4YVCB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
4KH |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4YVEA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4KK |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
4YVEB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
4KK |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5BMLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
4TW |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5BMLB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
4TW |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5KKSA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
6U1 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5KKTA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
6U2 |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5UZJA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
8UV |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5UZJB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
8UV |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TWJA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
07R |
Type1.5_Back |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5HVUA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
65R |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5HVUB |
None |
DFGin |
BLAminus |
in-in |
in-none |
65R |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5KKSB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
6U1 |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5KKTB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
6U2 |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNEA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
B4J |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNEB |
None |
DFGin |
BLAminus |
in-in |
in-none |
B4J |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNEC |
Active |
DFGin |
BLAminus |
in-in |
in-in |
B4J |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
5WNED |
Active |
DFGin |
BLAminus |
in-in |
in-in |
B4J |
Type1.5_Front |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S26C |
Inactive |
DFGin |
BLBminus |
in-in |
none-none |
86K |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TWJC |
Inactive |
DFGin |
None |
in-out |
out-out |
07R |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TWJB |
Inactive |
DFGinter |
None |
in-in |
out-in |
No_ligand |
No_ligand |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
3TWJD |
Inactive |
DFGinter |
None |
in-in |
out-in |
No_ligand |
No_ligand |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S25A |
Inactive |
DFGout |
None |
in-in |
none-out |
86G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S25B |
Inactive |
DFGout |
None |
in-in |
none-out |
86G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S25C |
Inactive |
DFGout |
None |
in-in |
none-none |
86G |
Type1 |
AGC |
ROCK1 |
ROCK1_HUMAN |
Rho-associated protein kinase 1 |
7S25D |
Inactive |
None |
None |
in-in |
none-none |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5MC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5MD |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7QA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7QB |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7QC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7QD |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7RA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
81G |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7RC |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
81G |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5PA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
O1V |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5PB |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
O1V |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5PC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
O1V |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5PD |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
O1V |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
4WOTA |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
3SG |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
4WOTB |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3SG |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
4WOTC |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
3SG |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
4WOTD |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
3SG |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
4L6QA |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
1WU |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
4L6QB |
Inactive |
DFGin |
ABAminus |
in-out |
in-in |
1WU |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
AF-O75116-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7RB |
Active |
DFGin |
BLAminus |
in-in |
in-in |
81G |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5MA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
O1S |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6P5MB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
O1S |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVA |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVB |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVC |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVD |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVE |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVF |
Active |
DFGin |
BLAminus |
in-in |
in-in |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVG |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JOVH |
Active |
DFGin |
BLAminus |
in-in |
in-in |
VFS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTA |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTB |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTC |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTD |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTE |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTF |
Active |
DFGin |
BLAminus |
in-in |
in-in |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTG |
None |
DFGin |
BLAminus |
in-in |
in-none |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7JNTH |
Active |
DFGin |
BLAminus |
in-in |
in-in |
VFA |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NB |
None |
DFGin |
BLAminus |
in-in |
in-none |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NC |
None |
DFGin |
BLAminus |
in-in |
in-none |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6ND |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NE |
None |
DFGin |
BLAminus |
in-in |
in-none |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NF |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NG |
None |
DFGin |
BLAminus |
in-in |
in-none |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
7P6NH |
None |
DFGin |
BLAminus |
in-in |
in-none |
5YS |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6ED6A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
J0P |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
6ED6B |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
J0P |
Type1.5_Front |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
5U7RD |
Inactive |
DFGin |
None |
in-in |
in-out |
81G |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
8GDSA |
Inactive |
DFGout |
BBAminus |
out-out |
in-out |
Z8O |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
8GDSB |
Inactive |
DFGout |
BBAminus |
out-none |
in-out |
Z8O |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
8GDSC |
Inactive |
DFGout |
BBAminus |
out-none |
in-out |
Z8O |
Type1 |
AGC |
ROCK2 |
ROCK2_HUMAN |
Rho-associated protein kinase 2 |
8GDSD |
Inactive |
DFGout |
BBAminus |
out-none |
in-in |
Z8O |
Type1.5_Front |
AGC |
RPS6KA1 |
KS6A1_HUMAN |
Ribosomal protein S6 kinase alpha-1 |
AF-Q15418-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KA1 |
KS6A1_HUMAN |
Ribosomal protein S6 kinase alpha-1 |
8XOVA |
Inactive |
DFGin |
BLAplus |
out-out |
out-out |
ANP |
Type1 |
AGC |
RPS6KA1 |
KS6A1_HUMAN |
Ribosomal protein S6 kinase alpha-1 |
2Z7QA |
Inactive |
DFGin |
BLBplus |
none-none |
out-out |
ACP |
Type1 |
AGC |
RPS6KA1 |
KS6A1_HUMAN |
Ribosomal protein S6 kinase alpha-1 |
2Z7RA |
Inactive |
DFGin |
BLBplus |
none-none |
out-out |
STU |
Type1 |
AGC |
RPS6KA1 |
KS6A1_HUMAN |
Ribosomal protein S6 kinase alpha-1 |
2Z7SA |
Inactive |
DFGin |
BLBplus |
none-none |
out-out |
P01 |
Type1 |
AGC |
RPS6KA2 |
KS6A2_HUMAN |
Ribosomal protein S6 kinase alpha-2 |
AF-Q15349-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
4NW5A |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
2NR |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
4NW6A |
Inactive |
DFGin |
ABAminus |
in-in |
in-in |
2NS |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
AF-P51812-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
7OPOA |
Inactive |
DFGin |
None |
none-none |
out-none |
ANP |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
7OPOE |
Inactive |
DFGin |
None |
none-none |
out-none |
ANP |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
7OPOI |
Inactive |
DFGin |
None |
none-none |
out-none |
ANP |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
7OPOK |
Inactive |
DFGin |
None |
none-none |
out-none |
ANP |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
7OPOC |
Inactive |
DFGinter |
None |
none-none |
out-out |
ANP |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
7OPOG |
Inactive |
DFGinter |
None |
out-out |
out-none |
ANP |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8EQ5A |
Inactive |
DFGout |
None |
none-none |
out-out |
QCT |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYA |
Inactive |
DFGout |
None |
out-out |
out-out |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYB |
Inactive |
DFGout |
None |
out-out |
out-out |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYC |
Inactive |
DFGout |
None |
none-none |
out-out |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYD |
Inactive |
DFGout |
None |
none-none |
out-out |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYE |
Inactive |
DFGout |
None |
none-none |
out-in |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYF |
Inactive |
DFGout |
None |
none-none |
out-out |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYG |
Inactive |
DFGout |
None |
in-out |
out-in |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYH |
Inactive |
DFGout |
None |
out-out |
out-in |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYI |
Inactive |
DFGout |
None |
none-none |
out-out |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
8XFYJ |
Inactive |
DFGout |
None |
none-none |
out-in |
A1LU8 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
4NUSA |
Inactive |
DFGout |
None |
in-out |
out-in |
2NK |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
5D9LA |
Inactive |
DFGout |
None |
in-out |
out-out |
583 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
5D9KA |
Inactive |
DFGout |
None |
in-out |
out-in |
584 |
Type1 |
AGC |
RPS6KA3 |
KS6A3_HUMAN |
Ribosomal protein S6 kinase alpha-3 |
5D9KB |
Inactive |
DFGout |
None |
in-none |
out-in |
584 |
Type1 |
AGC |
RPS6KA4 |
KS6A4_HUMAN |
Ribosomal protein S6 kinase alpha-4 |
AF-O75676-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KA5 |
KS6A5_HUMAN |
Ribosomal protein S6 kinase alpha-5 |
AF-O75582-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KA5 |
KS6A5_HUMAN |
Ribosomal protein S6 kinase alpha-5 |
1VZOA |
Inactive |
DFGinter |
None |
out-out |
out-out |
No_ligand |
No_ligand |
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
AF-Q9UK32-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
6G77A |
Inactive |
DFGin |
None |
none-none |
out-in |
ANP
ANP
|
Allosteric
Type1
|
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
6G77B |
Inactive |
DFGin |
None |
none-none |
out-in |
ANP
ANP
|
Allosteric
Type1
|
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
6G76B |
Inactive |
DFGinter |
None |
none-none |
out-none |
ANP |
Type1 |
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
6G78A |
Inactive |
DFGinter |
None |
none-none |
out-out |
ANP |
Type1 |
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
6G78B |
Inactive |
DFGinter |
None |
none-none |
out-out |
ANP |
Type1 |
AGC |
RPS6KA6 |
KS6A6_HUMAN |
Ribosomal protein S6 kinase alpha-6 |
6G76A |
Inactive |
DFGinter |
None |
none-none |
out-in |
ANP
ANP
|
Type1
Allosteric
|
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4RLPA |
Inactive |
DFGin |
ABAminus |
none-none |
in-out |
72B |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L3JA |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L3LA |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
7N91A |
Inactive |
DFGin |
ABAminus |
in-in |
none-out |
1RJ |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
7N91B |
Inactive |
DFGin |
ABAminus |
in-in |
none-none |
1RJ |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
7N93A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
1SK |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
7N93B |
Inactive |
DFGin |
ABAminus |
in-in |
none-out |
1SK |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3A62A |
Inactive |
DFGin |
ABAminus |
in-in |
none-out |
STU |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3WE4A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3WF5A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
FZ8 |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3WF6A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
FZ9 |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L45A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L42A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L46A |
Inactive |
DFGin |
ABAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
AF-P23443-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3WF8A |
Inactive |
DFGin |
BLAminus |
in-in |
out-out |
F76 |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3WF9A |
Inactive |
DFGin |
BLAminus |
in-in |
out-out |
FS7 |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L43A |
Inactive |
DFGin |
BLAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4L44A |
Inactive |
DFGin |
BLAminus |
in-in |
out-out |
5FI |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4RLOA |
Inactive |
DFGin |
None |
in-in |
in-out |
3T3 |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3A60A |
Inactive |
DFGin |
None |
in-out |
out-none |
STU |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3A61A |
Inactive |
DFGin |
None |
in-in |
none-out |
STU |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3WF7A |
Inactive |
DFGin |
None |
out-out |
out-out |
FS9 |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
4RLOB |
Inactive |
None |
None |
none-none |
out-none |
STU |
Type1 |
AGC |
RPS6KB1 |
KS6B1_HUMAN |
Ribosomal protein S6 kinase beta-1 |
3A60B |
Inactive |
None |
None |
none-none |
in-out |
STU |
Type1 |
AGC |
RPS6KB2 |
KS6B2_HUMAN |
Ribosomal protein S6 kinase beta-2 |
AF-Q9UBS0-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
RSKR |
KS6R_HUMAN |
Ribosomal protein S6 kinase-related protein |
AF-Q96LW2-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
SGK1 |
SGK1_HUMAN |
Serine/threonine-protein kinase Sgk1 |
AF-O00141-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
SGK1 |
SGK1_HUMAN |
Serine/threonine-protein kinase Sgk1 |
2R5TA |
Inactive |
DFGinter |
None |
none-none |
out-out |
ANP |
Type1 |
AGC |
SGK1 |
SGK1_HUMAN |
Serine/threonine-protein kinase Sgk1 |
3HDMA |
Inactive |
DFGinter |
None |
none-none |
out-out |
MMG |
Type1 |
AGC |
SGK1 |
SGK1_HUMAN |
Serine/threonine-protein kinase Sgk1 |
3HDNA |
Inactive |
DFGinter |
None |
none-none |
out-out |
GMG |
Type1 |
AGC |
SGK1 |
SGK1_HUMAN |
Serine/threonine-protein kinase Sgk1 |
7PUEA |
Inactive |
DFGout |
None |
none-none |
out-out |
86H |
Type1 |
AGC |
SGK2 |
SGK2_HUMAN |
Serine/threonine-protein kinase Sgk2 |
AF-Q9HBY8-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
SGK3 |
SGK3_HUMAN |
Serine/threonine-protein kinase Sgk3 |
AF-Q96BR1-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
AF-Q8WU08-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
4FR4A |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
4FR4B |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
4FR4C |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
4FR4D |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
4FR4E |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
AGC |
STK32A |
ST32A_HUMAN |
Serine/threonine-protein kinase 32A |
4FR4F |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
STU |
Type1 |
AGC |
STK32B |
ST32B_HUMAN |
Serine/threonine-protein kinase 32B |
AF-Q9NY57-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
STK32C |
ST32C_HUMAN |
Serine/threonine-protein kinase 32C |
AF-Q86UX6-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
STK38 |
STK38_HUMAN |
Serine/threonine-protein kinase 38 |
AF-Q15208-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
AGC |
STK38 |
STK38_HUMAN |
Serine/threonine-protein kinase 38 |
6BXIA |
Inactive |
DFGin |
None |
out-out |
out-out |
ANP |
Type1 |
AGC |
STK38 |
STK38_HUMAN |
Serine/threonine-protein kinase 38 |
6BXIB |
Inactive |
DFGin |
None |
out-out |
out-out |
ANP |
Type1 |
AGC |
STK38L |
ST38L_HUMAN |
Serine/threonine-protein kinase 38-like |
AF-Q9Y2H1-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DPVA |
Inactive |
DFGin |
ABAminus |
out-in |
in-out |
5DN
SKE
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DR6A |
Inactive |
DFGin |
ABAminus |
out-in |
in-out |
5E1
SKE
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2WTWA |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
ZZL |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3E5AA |
Inactive |
DFGin |
ABAminus |
out-out |
in-in |
VX6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2NP8A |
Inactive |
DFGin |
ABAminus |
out-out |
out-none |
CC3 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4C3PD |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4BYIA |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
FH3 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ONEA |
Inactive |
DFGin |
ABAminus |
out-out |
out-out |
9YQ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DT0A |
Inactive |
DFGin |
ABAminus |
in-in |
in-out |
SKE |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UODA |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
0C3 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UP2A |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
0C8 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4DEAA |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
NHI |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5AAFA |
Inactive |
DFGin |
ABAminus |
in-out |
in-out |
NL4 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5AAGA |
Inactive |
DFGin |
ABAminus |
out-none |
in-out |
6F2 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8GUWA |
Inactive |
DFGin |
ABAminus |
out-out |
in-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8GUWB |
Inactive |
DFGin |
ABAminus |
out-out |
none-none |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8GUWC |
Inactive |
DFGin |
ABAminus |
out-out |
none-none |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6GRAA |
Inactive |
DFGin |
ABAminus |
out-out |
none-none |
F8Z |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DN3A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5DN
ATP
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1EA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
T0X
ATP
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DT4A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5DN
ATP
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1MA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
T4X
ADP
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8SSPA |
Inactive |
DFGin |
BLAminus |
out-out |
in-in |
PDO
627
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DOSA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5DN
ATP
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DR2A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
5E1
ATP
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1DA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
T2F
ADP
T5L
|
Allosteric
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1GA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
T3I
ADP
T5L
|
Allosteric
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1HA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
T3U
ADP
T5L
|
Allosteric
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1KA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
T4O
ADP
T5L
|
Allosteric
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
AF-O14965-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6CPEA |
None |
DFGin |
BLAminus |
in-in |
in-none |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4J8NA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4J8NB |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4J8NC |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4J8ND |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4BN1A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3HA6A |
Inactive |
DFGin |
BLAminus |
in-out |
in-in |
2JZ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
1MQ4A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3MYGA |
None |
DFGin |
BLAminus |
in-in |
in-none |
EML |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3VAPA |
None |
DFGin |
BLAminus |
in-in |
none-out |
0FY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DNRA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ATP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DT3A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ATP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2W1CA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
L0C |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2W1DA |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
L0D |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2W1EA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
L0E |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2W1FA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
L0F |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2W1GA |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
L0G |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ZANA |
None |
DFGin |
BLAminus |
out-none |
in-out |
9A6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
1OL5A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
1OL7A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4O0SA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
ADN |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5G15A |
Inactive |
DFGin |
BLAminus |
out-out |
in-in |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2XNGA |
None |
DFGin |
BLAminus |
in-out |
in-none |
A0H |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4JAJA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
XU1 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2DWBA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ANP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2X6DA |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
X6D |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2X6EA |
None |
DFGin |
BLAminus |
in-out |
in-none |
YM4 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4ZS0A |
None |
DFGin |
BLAminus |
out-out |
in-none |
4QV |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6I2UA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
COA |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6CPFA |
None |
DFGin |
BLAminus |
out-none |
in-out |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPGA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ANP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DRDA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ATP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2XRUA |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
400 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UO4A |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
0C0 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UO5A |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
0BX |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UP7A |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
0C9 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4DEBA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
NHJ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4DEDA |
Inactive |
DFGin |
BLAminus |
in-out |
in-out |
NHU |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4DEEA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPIA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ANP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4JBOA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
WPH |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3NRMA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
NRM |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3R21A |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
D36 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5LXMA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4CEGA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5AADA |
None |
DFGin |
BLAminus |
in-in |
in-none |
5GX |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5G1XA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2XNEA |
None |
DFGin |
BLAminus |
out-out |
in-none |
ASH |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
1OL6A |
None |
DFGin |
BLAminus |
in-out |
in-none |
ATP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPLA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
ANP
R7D
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPLB |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
ANP
R7D
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPMA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
AMP
R74
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPMB |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
AMP
R74
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5DR9A |
Inactive |
DFGin |
BLAminus |
out-out |
out-out |
SKE
5E2
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORLA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A4W
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORNA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A5E
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OROA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A5H
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORPA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A5K
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORRA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A5Q
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORSA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A5W
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORTA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A5Z
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORVA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A65
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORWA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A6E
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORXA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A6H
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORYA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
AY4
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ORZA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A6W
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS0A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A6Z
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS1A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A7H
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS2A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A7K
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS3A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A7N
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS4A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A8H
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS6A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A7Q
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OSEA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A98
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OSFA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A9E
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OSDA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A9B
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OS5A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
A8K
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6R49A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
JSB
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6R4AA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
JRT
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6R4BA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
JSN
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6R4CA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
JRQ
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6R4DA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
JRW
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
7ZTLA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ADP
BCN
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8OF5A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
MPO
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C14A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
T5L
T0L
|
Type1
Allosteric
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C15A |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
T4C
T5L
|
Type1
Allosteric
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1FA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
T5L
T2O
|
Type1
Allosteric
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8C1IA |
Inactive |
DFGin |
BLAminus |
in-in |
in-out |
ADP
T1L
T5L
|
Type1
Allosteric
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3M11A |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
AKI |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4JBPA |
Inactive |
DFGin |
BLAminus |
out-out |
in-out |
YPH |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4J8MA |
Inactive |
DFGin |
BLAplus |
out-out |
out-out |
CJ5 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8JF4A |
Inactive |
DFGin |
None |
out-none |
none-out |
C0N |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8JMXA |
Inactive |
DFGin |
None |
out-none |
none-out |
E47 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4C3PA |
Inactive |
DFGin |
None |
out-out |
in-out |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
7AYIA |
Inactive |
DFGin |
None |
out-out |
none-none |
S9K |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2J4ZB |
Inactive |
DFGin |
None |
out-out |
out-out |
626 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4O0WA |
Inactive |
DFGin |
None |
out-out |
in-out |
ADN |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2C6DA |
Inactive |
DFGin |
None |
out-out |
out-out |
ANP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H0ZA |
Inactive |
DFGin |
None |
out-out |
none-none |
45B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4DHFA |
Inactive |
DFGin |
None |
in-in |
in-out |
0K6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4DHFB |
Inactive |
DFGin |
None |
in-in |
in-out |
0K6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4PRJA |
Inactive |
DFGin |
None |
in-in |
in-out |
2VU |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5AAEA |
Inactive |
DFGin |
None |
out-none |
in-out |
7HD |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4O0UA |
Inactive |
DFGin |
None |
out-out |
in-out |
ADN |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5ODTA |
Inactive |
DFGin |
None |
out-out |
out-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OBJA |
Inactive |
DFGin |
None |
out-out |
in-out |
ATP
9QK
|
Type1
Allosteric
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4UZDA |
Inactive |
DFGin |
None |
out-out |
none-out |
QMN |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4UZDB |
Inactive |
DFGin |
None |
out-out |
none-out |
QMN |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4UYNA |
Inactive |
DFGin |
None |
out-out |
none-none |
Y3M |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6XKAA |
Inactive |
DFGinter |
None |
out-out |
out-out |
No_ligand |
No_ligand |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2WTVA |
Inactive |
DFGinter |
None |
out-out |
out-out |
ZZL |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2WTVB |
Inactive |
DFGinter |
None |
out-out |
out-out |
ZZL |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2WTVC |
Inactive |
DFGinter |
None |
out-out |
out-out |
ZZL |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2WTVD |
Inactive |
DFGinter |
None |
out-out |
out-out |
ZZL |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5EW9A |
Inactive |
DFGinter |
None |
out-out |
out-out |
5VC |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6C2RA |
Inactive |
DFGinter |
None |
out-none |
out-none |
EG7 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6C2TA |
Inactive |
DFGinter |
None |
out-out |
out-out |
EGJ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W16A |
Inactive |
DFGinter |
None |
out-out |
out-out |
P9J |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2J50A |
Inactive |
DFGinter |
None |
out-out |
out-out |
627 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2J50B |
Inactive |
DFGinter |
None |
out-out |
out-out |
627 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4C3RA |
Inactive |
DFGinter |
None |
out-out |
out-out |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4ZTRA |
Inactive |
DFGinter |
None |
out-out |
none-out |
4RJ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6Z4YA |
Inactive |
DFGinter |
None |
out-out |
out-out |
Q7Q |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6C83B |
Inactive |
DFGinter |
None |
out-out |
none-out |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6CPGA |
Inactive |
DFGinter |
None |
out-out |
none-out |
35R |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6CPGD |
Inactive |
DFGinter |
None |
out-out |
none-out |
35R |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8SSOA |
Inactive |
DFGinter |
None |
out-out |
out-out |
627 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
8SSOD |
Inactive |
DFGinter |
None |
out-out |
out-none |
627 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
1MUOA |
Inactive |
DFGinter |
None |
out-out |
none-out |
ADN |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2J4ZA |
Inactive |
DFGinter |
None |
out-out |
out-out |
626 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UNZA |
Inactive |
DFGinter |
None |
out-out |
out-out |
0BZ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UNZB |
Inactive |
DFGinter |
None |
out-out |
out-out |
0BZ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UO6A |
Inactive |
DFGinter |
None |
out-out |
out-out |
0BY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UO6B |
Inactive |
DFGinter |
None |
out-out |
out-out |
0BY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOHA |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C4 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOHB |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C4 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOJA |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C5 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOJB |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C5 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOKA |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOKB |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOLA |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C7 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3UOLB |
Inactive |
DFGinter |
None |
out-out |
out-out |
0C7 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3FDNA |
Inactive |
DFGinter |
None |
out-out |
out-out |
MMH |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3K5UA |
Inactive |
DFGinter |
None |
out-out |
out-out |
PFQ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4JBQA |
Inactive |
DFGinter |
None |
out-out |
out-out |
VX6 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3LAUA |
Inactive |
DFGinter |
None |
out-out |
none-none |
OFI |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4UZHA |
Inactive |
DFGinter |
None |
out-out |
none-none |
JVE |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H0YA |
Inactive |
DFGinter |
None |
out-out |
none-none |
48B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H10A |
Inactive |
DFGinter |
None |
out-out |
out-out |
97B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H10B |
Inactive |
DFGinter |
None |
out-out |
out-out |
97B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H10D |
Inactive |
DFGinter |
None |
out-out |
out-none |
97B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3P9JA |
Inactive |
DFGinter |
None |
out-out |
out-out |
P9J |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W10A |
Inactive |
DFGinter |
None |
out-out |
out-out |
RO9 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3R22A |
Inactive |
DFGinter |
None |
out-out |
out-out |
D37 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2BMCA |
Inactive |
DFGinter |
None |
out-out |
out-none |
MPY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2BMCB |
Inactive |
DFGinter |
None |
out-out |
out-none |
MPY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2BMCC |
Inactive |
DFGinter |
None |
out-out |
out-none |
MPY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2BMCD |
Inactive |
DFGinter |
None |
out-out |
out-none |
MPY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2BMCE |
Inactive |
DFGinter |
None |
out-out |
out-none |
MPY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2BMCF |
Inactive |
DFGinter |
None |
out-out |
out-none |
MPY |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
7FICA |
Inactive |
DFGinter |
None |
out-none |
none-out |
5YZ |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5L8JA |
Inactive |
DFGinter |
None |
out-out |
none-none |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5L8KA |
Inactive |
DFGinter |
None |
out-out |
out-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5L8LA |
Inactive |
DFGinter |
None |
out-out |
out-out |
ADP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4ZTQA |
Inactive |
DFGinter |
None |
out-out |
out-out |
4RM |
Type1.5_Back |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4ZTSA |
Inactive |
DFGinter |
None |
out-out |
none-none |
4RK |
Type1.5_Back |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3EFWA |
Inactive |
DFGinter |
None |
out-none |
none-none |
AK8 |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3EFWB |
Inactive |
DFGinter |
None |
out-out |
none-none |
AK8 |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3O50A |
Inactive |
DFGinter |
None |
out-out |
none-none |
LJE |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3O50B |
Inactive |
DFGinter |
None |
out-out |
none-out |
LJE |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6HJJA |
Inactive |
DFGinter |
None |
out-out |
out-out |
G7T |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2C6EA |
Inactive |
DFGout |
BBAminus |
out-out |
none-out |
HPM |
Type1.5_Back |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPJA |
Inactive |
DFGout |
None |
out-out |
out-out |
ANP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4JAIA |
Inactive |
DFGout |
None |
out-out |
none-none |
XU2 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
7AYHA |
Inactive |
DFGout |
None |
out-out |
none-none |
S9H |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6VPHA |
Inactive |
DFGout |
None |
out-out |
out-out |
ANP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
7O2VA |
Inactive |
DFGout |
None |
out-out |
out-out |
V0K |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3O51A |
Inactive |
DFGout |
None |
out-none |
none-none |
LJF |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6HJKA |
Inactive |
DFGout |
None |
out-none |
out-out |
G7W |
Type1.5_Front |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
5OBRA |
Inactive |
None |
None |
out-out |
out-out |
9QT
SKE
|
Allosteric
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W2CC |
Inactive |
None |
None |
out-out |
none-none |
N15 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W2CE |
Inactive |
None |
None |
out-out |
none-none |
N15 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2X81A |
Inactive |
None |
None |
out-none |
none-out |
ZZL |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W18A |
Inactive |
None |
None |
out-out |
none-out |
N13 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W18B |
Inactive |
None |
None |
none-none |
none-out |
N13 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4B0GA |
Inactive |
None |
None |
out-out |
out-none |
VEK |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
4BYJA |
Inactive |
None |
None |
out-out |
none-none |
FH5 |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
6C83A |
Inactive |
None |
None |
out-none |
none-out |
ACP |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H0ZB |
Inactive |
None |
None |
out-out |
none-none |
45B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3H0ZC |
Inactive |
None |
None |
out-out |
none-none |
45B |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3COHA |
Inactive |
None |
None |
out-out |
none-out |
83H |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3COHB |
Inactive |
None |
None |
out-out |
none-out |
83H |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3QBNA |
Inactive |
None |
None |
out-out |
none-out |
E9Z |
Type1 |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2WQEA |
Inactive |
None |
None |
out-none |
none-out |
ADP
ADP
ADP
|
Type1
Type1
Type1
|
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W2CA |
Inactive |
None |
None |
out-out |
none-none |
N15 |
Type1.5_Back |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
3W2CG |
Inactive |
None |
None |
out-out |
none-none |
N15 |
Type1.5_Back |
CAMK |
AURKA |
AURKA_HUMAN |
Aurora kinase A |
2C6EB |
Inactive |
None |
None |
out-out |
none-in |
HPM |
Type1.5_Front |
CAMK |
AURKB |
AURKB_HUMAN |
Aurora kinase B |
AF-Q96GD4-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
AURKB |
AURKB_HUMAN |
Aurora kinase B |
4AF3A |
Inactive |
DFGinter |
None |
out-out |
none-none |
VX6 |
Type1 |
CAMK |
AURKC |
AURKC_HUMAN |
Aurora kinase C |
6GR9A |
Inactive |
DFGin |
ABAminus |
out-out |
in-in |
VX6 |
Type1 |
CAMK |
AURKC |
AURKC_HUMAN |
Aurora kinase C |
6GR8A |
Inactive |
DFGin |
ABAminus |
out-out |
in-in |
F8Z |
Type1.5_Front |
CAMK |
AURKC |
AURKC_HUMAN |
Aurora kinase C |
AF-Q9UQB9-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
BRSK1 |
BRSK1_HUMAN |
Serine/threonine-protein kinase BRSK1 |
AF-Q8TDC3-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
BRSK2 |
BRSK2_HUMAN |
Serine/threonine-protein kinase BRSK2 |
AF-Q8IWQ3-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
AF-Q14012-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
4FG7A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
ATP |
Type1 |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
4FGBA |
Inactive |
DFGinter |
None |
out-out |
out-out |
No_ligand |
No_ligand |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
4FG9A |
Inactive |
DFGinter |
None |
out-out |
none-none |
ATP |
Type1 |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
4FG9B |
Inactive |
DFGinter |
None |
out-none |
none-out |
ATP |
Type1 |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
4FG8A |
Inactive |
None |
None |
out-none |
none-none |
ATP |
Type1 |
CAMK |
CAMK1 |
KCC1A_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1 |
4FG8B |
Inactive |
None |
None |
out-none |
none-out |
ATP |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
AF-Q8IU85-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
6QP5A |
Inactive |
DFGin |
None |
out-out |
none-none |
No_ligand |
No_ligand |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
6T28AAA |
Inactive |
DFGin |
None |
out-out |
none-none |
M92 |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
8BFSA |
Inactive |
DFGin |
None |
out-out |
none-none |
QNR |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
8BFMA |
Inactive |
DFGin |
None |
out-none |
none-none |
QI6
QI6
|
Type1
Type3
|
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
6T6FA |
Inactive |
DFGinter |
None |
out-out |
none-none |
MMW |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
6T6FB |
Inactive |
DFGinter |
None |
out-out |
none-none |
MMW |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
6T29AAA |
Inactive |
DFGinter |
None |
out-out |
none-none |
M8Z |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
2JC6A |
Inactive |
None |
None |
out-none |
none-none |
QPP |
Type1 |
CAMK |
CAMK1D |
KCC1D_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1D |
2JC6C |
Inactive |
None |
None |
out-none |
none-none |
QPP |
Type1 |
CAMK |
CAMK1G |
KCC1G_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1G |
AF-Q96NX5-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK1G |
KCC1G_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1G |
2JAMA |
Inactive |
DFGin |
None |
out-out |
out-out |
J60 |
Type1 |
CAMK |
CAMK1G |
KCC1G_HUMAN |
Calcium/calmodulin-dependent protein kinase type 1G |
2JAMB |
Inactive |
DFGin |
None |
out-out |
out-out |
J60 |
Type1 |
CAMK |
CAMK2A |
KCC2A_HUMAN |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
AF-Q9UQM7-K1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK2A |
KCC2A_HUMAN |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
7UJRA |
Inactive |
DFGin |
BLAminus |
out-out |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK2A |
KCC2A_HUMAN |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
6VZKA |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK2A |
KCC2A_HUMAN |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
6X5QA |
Inactive |
DFGin |
BLAminus |
out-out |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK2A |
KCC2A_HUMAN |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
7KL1A |
Active |
DFGin |
BLAminus |
in-in |
in-in |
No_ligand |
No_ligand |
CAMK |
CAMK2A |
KCC2A_HUMAN |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
7KL1B |